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ES2008420A6 - PROCEDURE FOR OBTAINING A DRY PREPARATION SUITABLE FOR THE MANUFACTURE OF A WATER SUSPENSION OF A DICLOFENAC SALT - Google Patents

PROCEDURE FOR OBTAINING A DRY PREPARATION SUITABLE FOR THE MANUFACTURE OF A WATER SUSPENSION OF A DICLOFENAC SALT

Info

Publication number
ES2008420A6
ES2008420A6 ES8800262A ES8800262A ES2008420A6 ES 2008420 A6 ES2008420 A6 ES 2008420A6 ES 8800262 A ES8800262 A ES 8800262A ES 8800262 A ES8800262 A ES 8800262A ES 2008420 A6 ES2008420 A6 ES 2008420A6
Authority
ES
Spain
Prior art keywords
procedure
manufacture
obtaining
water suspension
dry preparation
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES8800262A
Other languages
Spanish (es)
Inventor
Leo Geller
Peter Glanzmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Publication of ES2008420A6 publication Critical patent/ES2008420A6/en
Expired legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/14Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Transition And Organic Metals Composition Catalysts For Addition Polymerization (AREA)
  • Blow-Moulding Or Thermoforming Of Plastics Or The Like (AREA)

Abstract

A dry formulation, in particular obtainable by lyophilisation, which is suitable for the preparation of a stable, aqueous suspension for the parenteral administration of a diclofenac salt contains a pharmaceutically acceptable and micronised salt of diclofenac and optional pharmaceutically acceptable adjuvants.
ES8800262A 1987-01-30 1988-01-29 PROCEDURE FOR OBTAINING A DRY PREPARATION SUITABLE FOR THE MANUFACTURE OF A WATER SUSPENSION OF A DICLOFENAC SALT Expired ES2008420A6 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
CH350/87A CH673395A5 (en) 1987-01-30 1987-01-30

Publications (1)

Publication Number Publication Date
ES2008420A6 true ES2008420A6 (en) 1989-07-16

Family

ID=4185019

Family Applications (1)

Application Number Title Priority Date Filing Date
ES8800262A Expired ES2008420A6 (en) 1987-01-30 1988-01-29 PROCEDURE FOR OBTAINING A DRY PREPARATION SUITABLE FOR THE MANUFACTURE OF A WATER SUSPENSION OF A DICLOFENAC SALT

Country Status (26)

Country Link
JP (1) JPS63192716A (en)
KR (1) KR880008808A (en)
AT (1) AT397460B (en)
AU (1) AU612343B2 (en)
BE (1) BE1000442A4 (en)
CA (1) CA1305058C (en)
CH (1) CH673395A5 (en)
DE (1) DE3802357A1 (en)
DK (1) DK45588A (en)
ES (1) ES2008420A6 (en)
FI (1) FI880368A7 (en)
FR (1) FR2611498B1 (en)
GB (1) GB2201089B (en)
GR (1) GR880100041A (en)
IE (1) IE60453B1 (en)
IT (1) IT1224241B (en)
LU (1) LU87115A1 (en)
MY (1) MY102662A (en)
NL (1) NL8800231A (en)
NO (1) NO880403L (en)
NZ (1) NZ223343A (en)
PH (1) PH23652A (en)
PT (1) PT86644B (en)
SE (1) SE8800228L (en)
YU (1) YU15488A (en)
ZA (1) ZA88638B (en)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH675537A5 (en) * 1988-03-25 1990-10-15 Ciba Geigy Ag
MX9201782A (en) * 1991-04-19 1992-10-01 Sandoz Ag PARTICLES OF BIOLOGICALLY ACTIVE SUBSTANCES, SUBSTANTIALLY INSOLUBLE IN WATER, PROCESS FOR THEIR PRODUCTION AND PHARMACEUTICAL COMPOSITION THAT CONTAINS THEM.
DE4140184C2 (en) * 1991-12-05 1995-12-21 Alfatec Pharma Gmbh Acute form for a medicine containing flurbiprofen
DE4140185C2 (en) * 1991-12-05 1996-02-01 Alfatec Pharma Gmbh Medicament containing a 2-arylpropionic acid derivative in nanosol form and its preparation
DE4140183C2 (en) * 1991-12-05 1995-12-21 Alfatec Pharma Gmbh Retard form for a medicine containing flurbiprofen
GB9212450D0 (en) * 1992-06-11 1992-07-22 Indena Spa New derivatives of non-steroidal anti-inflammatory,analgesic and/or antipyretic substances,their use and pharmaceutical formulations containing them
ZA949182B (en) * 1993-12-02 1995-07-26 South African Druggists Ltd Pharmaceutical composition
US6447806B1 (en) 1999-02-25 2002-09-10 Novartis Ag Pharmaceutical compositions comprised of stabilized peptide particles
FR2793418B1 (en) * 1999-05-11 2001-07-27 Synthelabo GALENIC FORMULATIONS OF ANTITHROMBOTIC AGENTS FOR SUBCUTANEOUS ADMINISTRATION
GB0207529D0 (en) * 2002-04-02 2002-05-08 Norbrook Lab Ltd Injectable veterinary composition for small animals
JO3352B1 (en) * 2005-06-17 2019-03-13 Apr Applied Pharma Res Sa Diclofenac formulations and methods of use

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1373913A (en) * 1970-12-17 1974-11-13 Glaxo Lab Ltd Pharmaceutical compositions
DE2914788A1 (en) * 1979-04-11 1980-10-16 Nattermann A & Cie PARENTERAL APPLICABLE, STABLE DRUG SOLUTIONS WITH ANTI-INFLAMMATORY EFFECT
DE3324193A1 (en) * 1983-07-05 1985-01-17 Troponwerke Gmbh & Co Kg DEPOT ANTIPHLOGISTICS
DE3328401A1 (en) * 1983-08-05 1985-02-21 Merckle GmbH, 7902 Blaubeuren INJECTABLE SOLUTION FOR TREATING INFLAMMATION
EP0152379A3 (en) * 1984-02-15 1986-10-29 Ciba-Geigy Ag Process for preparing pharmaceutical compositions containing unilamellar liposomes
DE3421468A1 (en) * 1984-06-08 1985-12-19 Dr. Rentschler Arzneimittel Gmbh & Co, 7958 Laupheim LIPID NANOPELLETS AS A CARRIER SYSTEM FOR MEDICINAL PRODUCTS FOR PERORAL USE
IE58110B1 (en) * 1984-10-30 1993-07-14 Elan Corp Plc Controlled release powder and process for its preparation
US5002940A (en) * 1984-11-06 1991-03-26 Ciba-Geigy Corporation Solid drug formulations and stable suspensions
DE3446873A1 (en) * 1984-12-21 1986-07-10 Merckle Gmbh LIQUID DICLOFENAC PREPARATIONS
IT1207994B (en) * 1986-01-03 1989-06-01 Therapicon Srl WATER SOLUBLE SALTS OF ANTI-INFLAMMATORY AND ANALGESIC ADAPTITY COMPOUNDS, THEIR PREPARATION AND USE IN PHARMACEUTICAL COMPOSITIONS.
DE3607339A1 (en) * 1986-03-06 1987-09-10 Merck Patent Gmbh PHARMACEUTICAL PREPARATION

Also Published As

Publication number Publication date
AU612343B2 (en) 1991-07-11
GB8801737D0 (en) 1988-02-24
DK45588A (en) 1988-07-31
SE8800228D0 (en) 1988-01-25
KR880008808A (en) 1988-09-13
IE60453B1 (en) 1994-07-13
YU15488A (en) 1989-10-31
JPS63192716A (en) 1988-08-10
GB2201089B (en) 1990-05-16
LU87115A1 (en) 1989-03-08
FR2611498B1 (en) 1991-06-14
CA1305058C (en) 1992-07-14
ZA88638B (en) 1989-10-25
FI880368A0 (en) 1988-01-27
ATA18588A (en) 1993-09-15
SE8800228L (en) 1988-07-31
DE3802357A1 (en) 1988-08-11
DK45588D0 (en) 1988-01-29
NO880403L (en) 1988-08-01
PH23652A (en) 1989-09-27
IT1224241B (en) 1990-09-26
BE1000442A4 (en) 1988-12-06
IE880250L (en) 1988-07-30
GB2201089A (en) 1988-08-24
FR2611498A1 (en) 1988-09-09
NO880403D0 (en) 1988-01-29
NL8800231A (en) 1988-08-16
FI880368L (en) 1988-07-31
FI880368A7 (en) 1988-07-31
MY102662A (en) 1992-08-17
IT8847557A0 (en) 1988-08-21
AT397460B (en) 1994-04-25
GR880100041A (en) 1988-12-16
AU1110288A (en) 1988-08-04
CH673395A5 (en) 1990-03-15
PT86644A (en) 1988-02-01
NZ223343A (en) 1990-03-27
PT86644B (en) 1992-01-31

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 19991102