EP0239062A3 - N2-(1-carboxy-3-oxo-3-phenylpropyl)-l-lysine compounds and their derivatives - Google Patents

N2-(1-carboxy-3-oxo-3-phenylpropyl)-l-lysine compounds and their derivatives Download PDF

Info

Publication number: EP0239062A3
Authority: EP; European Patent Office
Prior art keywords: phenylpropyl; oxo; carboxy; derivatives; lysine compounds
Prior art date: 1986-03-27
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

EP87104291A

Other versions

EP0239062A2 (en

EP0239062B1 (en

Inventor

Kazuhiko Yamada

Kenji Inoue

Satomi Takahashi

Takehisa Ohashi

Kiyoshi Watanabe

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

Kanegafuchi Chemical Industry Co Ltd

Original Assignee

Kanegafuchi Chemical Industry Co Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-03-27

Filing date

1987-03-24

Publication date

1988-03-02

1987-03-24 Application filed by Kanegafuchi Chemical Industry Co Ltd filed Critical Kanegafuchi Chemical Industry Co Ltd

1987-09-30 Publication of EP0239062A2 publication Critical patent/EP0239062A2/en

1988-03-02 Publication of EP0239062A3 publication Critical patent/EP0239062A3/en

1991-05-29 Application granted granted Critical

1991-05-29 Publication of EP0239062B1 publication Critical patent/EP0239062B1/en

2007-03-24 Anticipated expiration legal-status Critical

Status Expired - Lifetime legal-status Critical Current

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C233/00—Carboxylic acid amides
- C07C233/01—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms
- C07C233/45—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups
- C07C233/46—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a hydrocarbon radical substituted by carboxyl groups with the substituted hydrocarbon radical bound to the nitrogen atom of the carboxamide group by an acyclic carbon atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C271/00—Derivatives of carbamic acids, i.e. compounds containing any of the groups, the nitrogen atom not being part of nitro or nitroso groups
- C07C271/06—Esters of carbamic acids
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

EP87104291A 1986-03-27 1987-03-24 N2-(1-carboxy-3-oxo-3-phenylpropyl)-l-lysine compounds and their derivatives Expired - Lifetime EP0239062B1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP68970/86		1986-03-27
JP6897086		1986-03-27

Publications (3)

Publication Number	Publication Date
EP0239062A2 EP0239062A2 (en)	1987-09-30
EP0239062A3 true EP0239062A3 (en)	1988-03-02
EP0239062B1 EP0239062B1 (en)	1991-05-29

Family

ID=13389036

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EP87104291A Expired - Lifetime EP0239062B1 (en)	1986-03-27	1987-03-24	N2-(1-carboxy-3-oxo-3-phenylpropyl)-l-lysine compounds and their derivatives

Country Status (4)

Country	Link
EP (1)	EP0239062B1 (en)
CA (1)	CA1277993C (en)
DE (1)	DE3770301D1 (en)
ES (1)	ES2028812T3 (en)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU198446B (en) *	1987-09-25	1989-10-30	Richter Gedeon Vegyeszet	Process for production of new amids of buten acid and medical compositions containing such active substances
HU214581B (en) *	1995-03-14	1998-04-28	Richter Gedeon Vegyészeti Gyár Rt.	N2-(1s)-(1-ethoxycarbonyl-3-phenylpropyl)-n6-trifluoro-acetyl-l-lysyl-l-proline-benzilester and process for producing it
JP3792777B2 (en) *	1996-05-10	2006-07-05	株式会社カネカ	Method for producing 1-alkoxycarbonyl-3-phenylpropyl derivative
US5945457A (en) *	1997-10-01	1999-08-31	A.V. Topchiev Institute Of Petrochemical Synthesis, Russian Academy Of Science	Process for preparing biologically compatible polymers and their use in medical devices
JP2003026644A (en)	2001-07-11	2003-01-29	Kanegafuchi Chem Ind Co Ltd	Purification process of n2-[1(s)-ethoxy-carbonyl-3- phenylpropyl]-n6-trifluoroacetyl-l-lysine

Citations (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0150263A1 (en) *	1981-11-05	1985-08-07	Hoechst Aktiengesellschaft	Derivatives of cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acid, process for their preparation, medicaments containing them, and their use
US4626545A (en) *	1984-08-27	1986-12-02	Merck & Co., Inc.	Amino acid derivatives as enzyme inhibitors

1987
- 1987-03-24 ES ES198787104291T patent/ES2028812T3/en not_active Expired - Lifetime
- 1987-03-24 CA CA000532830A patent/CA1277993C/en not_active Expired - Lifetime
- 1987-03-24 EP EP87104291A patent/EP0239062B1/en not_active Expired - Lifetime
- 1987-03-24 DE DE8787104291T patent/DE3770301D1/en not_active Expired - Lifetime

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0150263A1 (en) *	1981-11-05	1985-08-07	Hoechst Aktiengesellschaft	Derivatives of cis, endo-2-azabicyclo-[3.3.0]-octane-3-carboxylic acid, process for their preparation, medicaments containing them, and their use
US4626545A (en) *	1984-08-27	1986-12-02	Merck & Co., Inc.	Amino acid derivatives as enzyme inhibitors

Non-Patent Citations (2)

* Cited by examiner, † Cited by third party
Title
CHEMICAL ABSTRACTS, vol. 107, no. 7, 17th August 1987, page 781, column 1, abstract no. 59477s, Columbus, Ohio, US; & ES - A - 544 465 (INKA S.A.) 01-03-1986 *
CHEMICAL ABSTRACTS, vol. 89, no. 25, 18th December 1978, page 630, column 2, abstract no. 215732p, Columbus, Ohio, US; AGBALYAN et al.: "Addition of aliphatic amino acids to beta-aroyl acrylic acids", ARM. KHIM. ZH. 1978, 31(4), 273-275 *

Also Published As

Publication number	Publication date
EP0239062A2 (en)	1987-09-30
DE3770301D1 (en)	1991-07-04
ES2028812T3 (en)	1992-07-16
CA1277993C (en)	1990-12-18
EP0239062B1 (en)	1991-05-29

Publication	Publication Date	Title
NZ220880A (en)	1990-10-26	Di-tert-butyl-phenol derivatives and pharmaceutical compositions
NZ220345A (en)	1990-10-26	Imidazoquinolinylether derivatives and pharmaceutical compositions containing them
NZ221996A (en)	1989-08-29	Imidazo-pyridine derivatives and pharmaceutical compositions
PH24049A (en)	1990-03-05	Substituted benzamide derivatives and pharmaceutical compositions containing the same
NZ220171A (en)	1990-05-28	Dihydro-benzopyran derivatives and pharmaceutical compositions
CS8700282A2 (en)	1991-07-16	Nicorandil-containing stable pharmaceutical
IL82205A (en)	1991-05-12	Substituted alkane-sulfonamidophenyl derivatives and pharmaceutical compositions containing them
EG18368A (en)	1992-10-30	Benzoyl-urea derivatives and its use as pesticide
NZ219161A (en)	1989-03-29	Propylamine derivatives and pharmaceutical compositions
GB2200352B (en)	1990-07-25	5-fluorouracil derivatives
NZ220486A (en)	1989-06-28	Substituted 3-amino-2-benzoylcyclohex-2-enone derivatives and herbicidal compositions
ZA879235B (en)	1988-06-24	Peridone derivatives,and their preparation and use
NZ223051A (en)	1990-06-26	Carbamoyloxylabdane derivatives and pharmaceutical compositions
EP0239062A3 (en)	1988-03-02	N2-(1-carboxy-3-oxo-3-phenylpropyl)-l-lysine compounds and their derivatives
PH23398A (en)	1989-07-26	Indenopyrimidine derivatives and pharmaceutical formulation containing the same
EP0238357A3 (en)	1988-10-05	1,2,4-triazinone derivatives, their preparation and use
PH22967A (en)	1989-02-10	Bis-tert.-butylamino-substituted 1,3,5-triazine derivatives, medidaments containing these compounds and their use
DK624587D0 (en)	1987-11-27	PHARMACEUTICAL PREPARATION CONTAINING IMIDAZOLD DERIVATIVES
NZ222683A (en)	1989-11-28	Substituted heterocyclic derivatives and pharmaceutical compositions
GB8706972D0 (en)	1987-04-29	5-fluorouracil derivatives
KR900700471A (en)	1990-08-13	New 2,3-thiomorpholine dione-2-oxime derivatives, pharmaceutical compositions and preparations containing them
NZ220383A (en)	1990-07-26	Pyrroloisoquinoline derivatives and pharmaceutical compositions
IL80010A0 (en)	1986-12-31	1-amino-3-phenylpropan-2-ol derivatives,their preparation and their use as microbicides
ZA875281B (en)	1988-03-30	Zylometzoline-containing pharmaceutical preparations
PH22830A (en)	1989-01-19	Novel quinaldinamide derivatives and their preparations

Legal Events

Date	Code	Title	Description
1987-08-15	PUAI	Public reference made under article 153(3) epc to a published international application that has entered the european phase	Free format text: ORIGINAL CODE: 0009012
1987-09-30	AK	Designated contracting states	Kind code of ref document: A2 Designated state(s): BE CH DE ES FR GB IT LI NL SE
1988-01-12	PUAL	Search report despatched	Free format text: ORIGINAL CODE: 0009013
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1988-10-19	17P	Request for examination filed	Effective date: 19880824
1989-11-08	17Q	First examination report despatched	Effective date: 19890926
1991-04-12	GRAA	(expected) grant	Free format text: ORIGINAL CODE: 0009210
1991-05-29	AK	Designated contracting states	Kind code of ref document: B1 Designated state(s): BE CH DE ES FR GB IT LI NL SE
1991-07-04	REF	Corresponds to:	Ref document number: 3770301 Country of ref document: DE Date of ref document: 19910704
1991-08-02	ET	Fr: translation filed
1991-08-26	ITF	It: translation for a ep patent filed
1992-04-02	PLBE	No opposition filed within time limit	Free format text: ORIGINAL CODE: 0009261
1992-04-02	STAA	Information on the status of an ep patent application or granted ep patent	Free format text: STATUS: NO OPPOSITION FILED WITHIN TIME LIMIT
1992-05-20	26N	No opposition filed
1992-07-16	REG	Reference to a national code	Ref country code: ES Ref legal event code: FG2A Ref document number: 2028812 Country of ref document: ES Kind code of ref document: T3
1995-01-31	EAL	Se: european patent in force in sweden	Ref document number: 87104291.7
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2007-12-31	BE20	Be: patent expired	Owner name: KANEGAFUCHI KAGAKU KOGYO K.K. Effective date*: 20070324
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