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EA200600787A1 - Антагонисты мускариновых ацетилхолиновых рецепторов - Google Patents

Антагонисты мускариновых ацетилхолиновых рецепторов

Info

Publication number
EA200600787A1
EA200600787A1 EA200600787A EA200600787A EA200600787A1 EA 200600787 A1 EA200600787 A1 EA 200600787A1 EA 200600787 A EA200600787 A EA 200600787A EA 200600787 A EA200600787 A EA 200600787A EA 200600787 A1 EA200600787 A1 EA 200600787A1
Authority
EA
Eurasian Patent Office
Prior art keywords
antagonists
muscarine
acetyl choline
choline receptors
receptors
Prior art date
Application number
EA200600787A
Other languages
English (en)
Inventor
Майкл Р. Палович
Цзехун Вань
Чунцзе Чжу
Original Assignee
Глэксо Груп Лимитед
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Глэксо Груп Лимитед filed Critical Глэксо Груп Лимитед
Publication of EA200600787A1 publication Critical patent/EA200600787A1/ru

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/02—Nasal agents, e.g. decongestants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/06—Antiasthmatics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A61P11/08—Bronchodilators
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Pulmonology (AREA)
  • Immunology (AREA)
  • Urology & Nephrology (AREA)
  • Otolaryngology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Описаны антагонисты мускариновых ацетилхолиновых рецепторов и способы их использования.
EA200600787A 2003-10-17 2004-10-15 Антагонисты мускариновых ацетилхолиновых рецепторов EA200600787A1 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US51216103P 2003-10-17 2003-10-17
PCT/US2004/034234 WO2005037224A2 (en) 2003-10-17 2004-10-15 Muscarinic acetylcholine receptor antagonists

Publications (1)

Publication Number Publication Date
EA200600787A1 true EA200600787A1 (ru) 2006-08-25

Family

ID=34465319

Family Applications (1)

Application Number Title Priority Date Filing Date
EA200600787A EA200600787A1 (ru) 2003-10-17 2004-10-15 Антагонисты мускариновых ацетилхолиновых рецепторов

Country Status (22)

Country Link
US (1) US7507747B2 (ru)
EP (1) EP1677796A4 (ru)
JP (1) JP2007509061A (ru)
CN (1) CN1897947A (ru)
AP (1) AP2006003575A0 (ru)
AR (1) AR046114A1 (ru)
AU (1) AU2004281167A1 (ru)
BR (1) BRPI0415281A (ru)
CA (1) CA2542636A1 (ru)
EA (1) EA200600787A1 (ru)
EC (1) ECSP066486A (ru)
IL (1) IL174846A0 (ru)
IS (1) IS8440A (ru)
MA (1) MA28109A1 (ru)
MX (1) MXPA06004242A (ru)
NO (1) NO20062071L (ru)
OA (1) OA13270A (ru)
PE (1) PE20050442A1 (ru)
TW (1) TW200528448A (ru)
UY (1) UY28567A1 (ru)
WO (1) WO2005037224A2 (ru)
ZA (1) ZA200602783B (ru)

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PE20050489A1 (es) * 2003-11-04 2005-09-02 Glaxo Group Ltd Antagonistas de receptores de acetilcolina muscarinicos
JP2007528420A (ja) * 2004-03-11 2007-10-11 グラクソ　グループ　リミテッド 新規ｍ３ムスカリン性アセチルコリン受容体アンタゴニスト
WO2005095407A1 (en) * 2004-03-17 2005-10-13 Glaxo Group Limited M3 muscarinic acetylcholine receptor antagonists
JP2007529511A (ja) * 2004-03-17 2007-10-25 グラクソ　グループ　リミテッド Ｍ３ムスカリン性アセチルコリン受容体アンタゴニスト
AR050902A1 (es) 2004-04-27 2006-12-06 Glaxo Group Ltd Compuesto de quinuclidina, composicion farmaceutica que lo comprende y su usopara preparar dicha composicion
WO2005112644A2 (en) * 2004-05-13 2005-12-01 Glaxo Group Limited Muscarinic acetylcholine receptor antagonists
EP1957075A4 (en) * 2004-11-15 2009-11-18 Glaxo Group Ltd NOVEL ANTAGONISTS OF ACETYLCHOLINE M3 TYPE MUSCARINIC RECEPTORS
WO2007016639A2 (en) * 2005-08-02 2007-02-08 Glaxo Group Limited M3 muscarinic acetylcholine receptor antagonists
US7767691B2 (en) * 2005-08-18 2010-08-03 Glaxo Group Limited Muscarinic acetylcholine receptor antagonists containing an azoniabiocyclo[2.2.1] heptane ring system
UY31635A1 (es) 2008-02-06 2009-08-31 Farmacóforos duales-antagonistas muscarínicos de pde4
CL2009000250A1 (es) 2008-02-06 2009-09-11 Glaxo Group Ltd Compuestos derivados de pirazolo[3,4-b]piridina carboxamida; composicion farmaceutica que los comprende; y su uso en el tratamiento del asma, epoc y rinitis.
AR070563A1 (es) 2008-02-06 2010-04-21 Glaxo Group Ltd Compuesto de un biciclo condensado pirazol-piridin-amina, composicion farmaceutica que lo comprende y su uso para preparar un medicamento util para el tratamiento de enfermedades respiratorias.
WO2010094643A1 (en) 2009-02-17 2010-08-26 Glaxo Group Limited Quinoline derivatives and their uses for rhinitis and urticaria

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Also Published As

Publication number Publication date
EP1677796A2 (en) 2006-07-12
MXPA06004242A (es) 2006-06-28
AP2006003575A0 (en) 2006-04-30
AU2004281167A1 (en) 2005-04-28
WO2005037224A3 (en) 2005-06-23
TW200528448A (en) 2005-09-01
UY28567A1 (es) 2005-05-31
BRPI0415281A (pt) 2006-12-19
CA2542636A1 (en) 2005-04-28
PE20050442A1 (es) 2005-07-09
US7507747B2 (en) 2009-03-24
IS8440A (is) 2006-05-05
ZA200602783B (en) 2007-11-28
AR046114A1 (es) 2005-11-23
EP1677796A4 (en) 2006-12-27
OA13270A (en) 2007-01-31
US20070135478A1 (en) 2007-06-14
CN1897947A (zh) 2007-01-17
JP2007509061A (ja) 2007-04-12
WO2005037224A2 (en) 2005-04-28
NO20062071L (no) 2006-05-08
MA28109A1 (fr) 2006-08-01
ECSP066486A (es) 2006-10-10
IL174846A0 (en) 2006-08-20

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