DK412474A - - Google Patents

Info

Publication number: DK412474A
Authority: DK; Denmark

Application number

DK412474A

Other languages

Danish (da)

Other versions

DK146298B (en

DK146298C (en

Inventor

M J Weinstein

P J L Daniels

G H Wagman

R Testa

A K Mallams

J J Wright

T L Nagabhushan

Original Assignee

Scherico Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1973-08-06

Filing date

1974-08-01

Publication date

1975-04-01

1974-03-19 Priority claimed from US05/452,586 external-priority patent/US4029882A/en

1974-08-01 Application filed by Scherico Ltd filed Critical Scherico Ltd

1975-04-01 Publication of DK412474A publication Critical patent/DK412474A/da

1979-02-08 Priority to DK52879A priority Critical patent/DK52879A/en

1983-08-29 Publication of DK146298B publication Critical patent/DK146298B/en

1984-02-06 Application granted granted Critical

1984-02-06 Publication of DK146298C publication Critical patent/DK146298C/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- C07H15/236—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2 a saccharide radical being substituted by an alkylamino radical in position 3 and by two substituents different from hydrogen in position 4, e.g. gentamicin complex, sisomicin, verdamycin
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Engineering & Computer Science (AREA)
Health & Medical Sciences (AREA)
Biochemistry (AREA)
Biotechnology (AREA)
General Health & Medical Sciences (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Life Sciences & Earth Sciences (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Polysaccharides And Polysaccharide Derivatives (AREA)

DK412474A 1973-08-06 1974-08-01 ANALOGY PROCEDURE FOR PREPARING 1-N-SUBSTITUTED DERIVATIVES OF 4,6-DI- (AMINOGLYCOSYL) -1,3-DIAMINOCYCLITOLS OR ACID ADDITION SALTS THEREOF DK146298C (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
DK52879A DK52879A (en)	1974-03-19	1979-02-08	PROCEDURE FOR THE PREPARATION OF 1-N-SUBSTITUTED DERIVATIVES OF 4,6-DI- (AMINOGLYCOSYL) -1,3-DIAMINOCYCLOTOLS OR ACID ADDITIONAL SALTS THEREOF

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
US38575173A	1973-08-06	1973-08-06
US38575173		1973-08-06
US45260074A	1974-03-19	1974-03-19
US45260074		1974-03-19
US05/452,586 US4029882A (en)	1974-03-19	1974-03-19	Selective acylation of the C-1 amino group of aminoglycoside antibiotics
US45258674		1974-03-19

Publications (3)

Publication Number	Publication Date
DK412474A true DK412474A (en)	1975-04-01
DK146298B DK146298B (en)	1983-08-29
DK146298C DK146298C (en)	1984-02-06

Family

ID=27409729

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK412474A DK146298C (en)	1973-08-06	1974-08-01	ANALOGY PROCEDURE FOR PREPARING 1-N-SUBSTITUTED DERIVATIVES OF 4,6-DI- (AMINOGLYCOSYL) -1,3-DIAMINOCYCLITOLS OR ACID ADDITION SALTS THEREOF

Country Status (20)

Country	Link
AR (1)	AR215834A1 (en)
BE (1)	BE818431A (en)
BG (1)	BG25804A3 (en)
CH (1)	CH606076A5 (en)
CY (1)	CY1018A (en)
DD (1)	DD119037A5 (en)
DE (2)	DE2462485C2 (en)
DK (1)	DK146298C (en)
FI (1)	FI62100C (en)
FR (1)	FR2240015B1 (en)
GB (1)	GB1473733A (en)
HK (1)	HK55179A (en)
IE (1)	IE40437B1 (en)
IL (1)	IL45385A (en)
KE (1)	KE2981A (en)
LU (1)	LU70661A1 (en)
MY (1)	MY8000090A (en)
NL (1)	NL171587C (en)
NO (1)	NO139483C (en)
SE (1)	SE424994B (en)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4217446A (en)	1974-10-26	1980-08-12	Pfizer Inc.	ωAmino-2-hydroxyalkyl derivatives of aminoglycoside antibiotics
GB1464401A (en) *	1974-10-26	1977-02-16	Pfizer Ltd	Aminoglycosides
FR2405266A1 (en) *	1975-09-08	1979-05-04	Scherico Ltd	Antibacterial desoxystreptamines - esp 5-epi-4,6-di-(aminoglycosyl)-2-desoxystreptamines and 5-epi-(amino or azido)-5-desoxy derivs
EP0000057B1 (en) *	1977-06-10	1982-07-14	Bayer Ag	Selectively protected 4,6-di-o-(aminoglycosyl)-1,3-diamino-cyclitols
US4282350A (en) *	1977-08-05	1981-08-04	Schering Corporation	Selective 3"-N-acylation of 1,3"-di-N-unprotected-poly-N-protected-4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols
JPS5492951A (en) *	1977-12-29	1979-07-23	Shionogi & Co Ltd	Novel aminoglycoside derivative
JPS5538345A (en) *	1978-09-11	1980-03-17	Shionogi & Co Ltd	Novel aminoglycoside derivative
DE2840907A1 (en) *	1978-09-20	1980-04-03	Bayer Ag	SELECTIVELY PROTECTED 4,6-DI-O- (AMINOGLYKOSYL) -1,3-DIAMINOCYCLITOLE
DE2928183A1 (en) *	1979-07-12	1981-01-29	Bayer Ag	1-N-ALKYLSISOMICIN DERIVATIVES, METHOD FOR THE PRODUCTION THEREOF AND THEIR USE AS MEDICINAL PRODUCTS
CN1040177C (en) *	1993-04-23	1998-10-14	江苏省微生物研究所	1-N-ethyl gentamicin derivative and its preparing method
LT2217610T (en)	2007-11-21	2017-02-27	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132757A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132765A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132760A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of tobramycin
WO2010132768A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of sisomicin
WO2010132759A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of dibekacin
CN101575311B (en) *	2009-06-19	2011-05-04	无锡好芳德药业有限公司	Method for preparing epiphysin

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1235311B (en)	1963-03-25	1967-03-02	Roussel Uclaf	Process for the production of N-monophenylaethylneomycin B or its therapeutically acceptable salts

1974
- 1974-07-31 CH CH1060274A patent/CH606076A5/xx not_active IP Right Cessation
- 1974-08-01 SE SE7409946A patent/SE424994B/en not_active IP Right Cessation
- 1974-08-01 FR FR7426815A patent/FR2240015B1/fr not_active Expired
- 1974-08-01 AR AR255007A patent/AR215834A1/en active
- 1974-08-01 NL NLAANVRAGE7410363,A patent/NL171587C/en not_active IP Right Cessation
- 1974-08-01 DK DK412474A patent/DK146298C/en not_active IP Right Cessation
- 1974-08-01 GB GB3396874A patent/GB1473733A/en not_active Expired
- 1974-08-01 IE IE1638/74A patent/IE40437B1/en not_active IP Right Cessation
- 1974-08-01 DE DE2462485A patent/DE2462485C2/en not_active Expired
- 1974-08-01 CY CY1018A patent/CY1018A/en unknown
- 1974-08-01 NO NO742787A patent/NO139483C/en unknown
- 1974-08-01 FI FI2304/74A patent/FI62100C/en active
- 1974-08-01 DE DE2437160A patent/DE2437160C3/en not_active Expired
- 1974-08-02 IL IL45385A patent/IL45385A/en unknown
- 1974-08-02 BE BE147234A patent/BE818431A/en not_active IP Right Cessation
- 1974-08-02 LU LU70661A patent/LU70661A1/xx unknown
- 1974-08-05 DD DD180344A patent/DD119037A5/xx unknown
- 1974-08-06 BG BG027440A patent/BG25804A3/en unknown
1979
- 1979-07-09 KE KE2981A patent/KE2981A/en unknown
- 1979-08-09 HK HK551/79A patent/HK55179A/en unknown
1980
- 1980-12-30 MY MY90/80A patent/MY8000090A/en unknown

Also Published As

Publication number	Publication date
FI230474A (en)	1975-02-07
KE2981A (en)	1979-07-20
MY8000090A (en)	1980-12-31
FI62100B (en)	1982-07-30
NO742787L (en)	1975-03-03
DK146298B (en)	1983-08-29
LU70661A1 (en)	1975-05-21
DE2462485C2 (en)	1987-04-09
AR215834A1 (en)	1979-11-15
NO139483C (en)	1979-03-21
BE818431A (en)	1975-02-03
CH606076A5 (en)	1978-10-13
DE2462485A1 (en)	1977-04-21
DE2437160B2 (en)	1979-01-04
NL7410363A (en)	1975-02-10
IE40437B1 (en)	1979-06-06
SE424994B (en)	1982-08-23
IE40437L (en)	1975-02-06
BG25804A3 (en)	1978-12-12
DE2437160C3 (en)	1979-08-30
DD119037A5 (en)	1976-04-05
NO139483B (en)	1978-12-11
NL171587C (en)	1983-04-18
CY1018A (en)	1979-11-23
AU7194274A (en)	1976-02-05
DE2437160A1 (en)	1975-02-20
NL171587B (en)	1982-11-16
FI62100C (en)	1982-11-10
IL45385A (en)	1978-10-31
FR2240015B1 (en)	1978-08-18
HK55179A (en)	1979-08-17
IL45385A0 (en)	1974-11-29
SE7409946L (en)	1975-02-07
FR2240015A1 (en)	1975-03-07
DK146298C (en)	1984-02-06
GB1473733A (en)	1977-05-18

Publication	Publication Date	Title
AR201758A1 (en)	1975-04-15
AU476761B2 (en)	1976-09-30
AU465372B2 (en)	1975-09-25
AR201235Q (en)	1975-02-21
AR201231Q (en)	1975-02-21
AU474593B2 (en)	1976-07-29
AU474511B2 (en)	1976-07-22
AU474838B2 (en)	1976-08-05
AU471343B2 (en)	1976-04-15
FR2240015A1 (en)	1975-03-07
AU465453B2 (en)	1975-09-25
AU465434B2 (en)	1975-09-25
AU450229B2 (en)	1974-07-04
AU476714B2 (en)	1976-09-30
AR201229Q (en)	1975-02-21
AU466283B2 (en)	1975-10-23
AU472848B2 (en)	1976-06-03
AU476696B2 (en)	1976-09-30
AR199451A1 (en)	1974-08-30
AU477823B2 (en)	1975-06-19
AR195948A1 (en)	1973-11-15
AR196382A1 (en)	1973-12-18
AU477824B2 (en)	1975-07-17
AR195311A1 (en)	1973-09-28
AR200256A1 (en)	1974-10-31

Legal Events

Date	Code	Title	Description
1994-09-12	PUP	Patent expired