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DK3399984T3 - Modulatorer af 5'-nukleotidase, ecto og anvendelsen deraf - Google Patents

Modulatorer af 5'-nukleotidase, ecto og anvendelsen deraf Download PDF

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Publication number
DK3399984T3
DK3399984T3 DK17736459.3T DK17736459T DK3399984T3 DK 3399984 T3 DK3399984 T3 DK 3399984T3 DK 17736459 T DK17736459 T DK 17736459T DK 3399984 T3 DK3399984 T3 DK 3399984T3
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Prior art keywords
nucleotidase
ecto
modulators
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DK17736459.3T
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English (en)
Inventor
Laurent Pierre Paul Debien
Juan Carlos Jaen
Jaroslaw Kalisiak
Kenneth V Lawson
Manmohan Reddy Leleti
Erick Allen Lindsey
Dillon Harding Miles
Eric Newcomb
Jay Patrick Powers
Brandon Reid Rosen
Ehesan Ui Sharif
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Arcus Biosciences Inc
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Publication of DK3399984T3 publication Critical patent/DK3399984T3/da

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    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/23Heterocyclic radicals containing two or more heterocyclic rings condensed among themselves or condensed with a common carbocyclic ring system, not provided for in groups C07H19/14 - C07H19/22
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DK17736459.3T 2016-01-08 2017-01-06 Modulatorer af 5'-nukleotidase, ecto og anvendelsen deraf DK3399984T3 (da)

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Application Number Priority Date Filing Date Title
US201662276564P 2016-01-08 2016-01-08
US201662324077P 2016-04-18 2016-04-18
PCT/US2017/012587 WO2017120508A1 (en) 2016-01-08 2017-01-06 Modulators of 5'-nucleotidase, ecto and the use thereof

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JP (3) JP6920344B2 (da)
KR (1) KR20180100638A (da)
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SA (1) SA518391985B1 (da)
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SI (1) SI3399984T1 (da)
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UA (1) UA124529C2 (da)
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Publication number Priority date Publication date Assignee Title
BR112018013827B1 (pt) 2016-01-08 2024-02-20 Arcus Biosciences, Inc Moduladores de 5-nucleotidase, ecto, composição farmacêutica, combinação, kit e uso dos mesmos
US10472364B2 (en) 2016-09-09 2019-11-12 Calithera Biosciences, Inc. Ectonucleotidase inhibitors and methods of use thereof
US11267845B2 (en) 2016-11-18 2022-03-08 Arcus Biosciences, Inc. Inhibitors of CD73-mediated immunosuppression
PT3551627T (pt) 2016-12-08 2022-04-06 H Hoffnabb La Roche Ag Novos derivados de éter isoxazolílico enquanto moduladores alostéricos positivos de gaba a α5
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