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DK2820006T3 - Pyrazol-1-yl benzen sulfonamider som ccr9 antagonister - Google Patents

Pyrazol-1-yl benzen sulfonamider som ccr9 antagonister

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Publication number
DK2820006T3
DK2820006T3 DK13708633.6T DK13708633T DK2820006T3 DK 2820006 T3 DK2820006 T3 DK 2820006T3 DK 13708633 T DK13708633 T DK 13708633T DK 2820006 T3 DK2820006 T3 DK 2820006T3
Authority
DK
Denmark
Prior art keywords
benzen
sulphonamides
pyrazol
ccr9 antagonists
ccr9
Prior art date
Application number
DK13708633.6T
Other languages
English (en)
Inventor
Xi Chen
Pingchen Fan
Antoni Krasinski
Lianfa Li
Jeffrey P Mcmahon
Jay P Powers
Yibin Zeng
Penglie Zhang
Rebecca M Lui
Junfa Fan
Original Assignee
Chemocentryx Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chemocentryx Inc filed Critical Chemocentryx Inc
Application granted granted Critical
Publication of DK2820006T3 publication Critical patent/DK2820006T3/da

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    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4151,2-Diazoles
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    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/472Non-condensed isoquinolines, e.g. papaverine
    • A61K31/4725Non-condensed isoquinolines, e.g. papaverine containing further heterocyclic rings
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    • C07D231/10Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D231/14Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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    • C07D231/42Benzene-sulfonamido pyrazoles
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    • A61K31/50Pyridazines; Hydrogenated pyridazines
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    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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DK13708633.6T 2012-02-29 2013-02-28 Pyrazol-1-yl benzen sulfonamider som ccr9 antagonister DK2820006T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201261604998P 2012-02-29 2012-02-29
PCT/US2013/028328 WO2013130811A1 (en) 2012-02-29 2013-02-28 Pyrazol-1-yl benzene sulfonamides as ccr9 antagonists

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DK2820006T3 true DK2820006T3 (da) 2017-11-06

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DK17184205.7T DK3263564T3 (da) 2012-02-29 2013-02-28 Aza-aryl-1h-pyrazol-1-yl-benzen-sulfonamider som ccr(9)- antagonister
DK13708633.6T DK2820006T3 (da) 2012-02-29 2013-02-28 Pyrazol-1-yl benzen sulfonamider som ccr9 antagonister

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US (5) US8916601B2 (da)
EP (3) EP3263564B1 (da)
JP (3) JP6249966B2 (da)
KR (1) KR102083693B1 (da)
CN (2) CN107266425B (da)
AU (3) AU2013225938B2 (da)
BR (1) BR112014021148B1 (da)
CA (1) CA2865714C (da)
DK (2) DK3263564T3 (da)
ES (2) ES2816060T3 (da)
HK (3) HK1206012A1 (da)
MX (1) MX2014010340A (da)
PL (2) PL3263564T3 (da)
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AU2017209023B2 (en) * 2016-01-20 2021-06-17 Chemocentryx, Inc. 2-oxindole compounds
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PL3634417T3 (pl) 2017-05-17 2023-09-25 Arcus Biosciences, Inc. Pochodne chinazolino-pirazolowe do leczenia chorób związanych z nowotworem
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