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DK1713805T3 - Kinaseinhibitorer - Google Patents

Kinaseinhibitorer

Info

Publication number
DK1713805T3
DK1713805T3 DK05704878T DK05704878T DK1713805T3 DK 1713805 T3 DK1713805 T3 DK 1713805T3 DK 05704878 T DK05704878 T DK 05704878T DK 05704878 T DK05704878 T DK 05704878T DK 1713805 T3 DK1713805 T3 DK 1713805T3
Authority
DK
Denmark
Prior art keywords
kinase inhibitors
kinase
inhibitors
Prior art date
Application number
DK05704878T
Other languages
English (en)
Inventor
Rosanne Bonjouklian
Chafiq Hamdouchi
Chuan Shih
Dios Alfonso De
Prado Miriam Filadelfa Del
Aguado Carlos Jaramillo
Pramila Kotiyan
Mary Margaret Mader
Sheila Pleite Selgas
Concepcion Sanchez-Martinez
Original Assignee
Lilly Co Eli
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34837430&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK1713805(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Lilly Co Eli filed Critical Lilly Co Eli
Application granted granted Critical
Publication of DK1713805T3 publication Critical patent/DK1713805T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Rheumatology (AREA)
  • Pain & Pain Management (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK05704878T 2004-01-30 2005-01-25 Kinaseinhibitorer DK1713805T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US54083004P 2004-01-30 2004-01-30
PCT/US2005/000025 WO2005075478A1 (en) 2004-01-30 2005-01-25 Kinase inhibitors

Publications (1)

Publication Number Publication Date
DK1713805T3 true DK1713805T3 (da) 2009-08-17

Family

ID=34837430

Family Applications (1)

Application Number Title Priority Date Filing Date
DK05704878T DK1713805T3 (da) 2004-01-30 2005-01-25 Kinaseinhibitorer

Country Status (26)

Country Link
US (2) US7582652B2 (da)
EP (1) EP1713805B1 (da)
CN (1) CN100516064C (da)
AR (1) AR047466A1 (da)
AT (1) ATE433449T1 (da)
AU (1) AU2005210459B2 (da)
CA (1) CA2559128C (da)
CY (1) CY1109234T1 (da)
DE (1) DE602005014848D1 (da)
DK (1) DK1713805T3 (da)
DO (1) DOP2005000010A (da)
ES (1) ES2326819T3 (da)
HK (1) HK1100141A1 (da)
IL (1) IL178103A (da)
MY (1) MY143516A (da)
NZ (1) NZ549780A (da)
PE (1) PE20050689A1 (da)
PL (1) PL1713805T3 (da)
PT (1) PT1713805E (da)
RU (1) RU2348635C2 (da)
SI (1) SI1713805T1 (da)
SV (1) SV2006002001A (da)
TW (1) TWI332003B (da)
UA (1) UA85505C2 (da)
WO (1) WO2005075478A1 (da)
ZA (1) ZA200607648B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TWI332003B (en) * 2004-01-30 2010-10-21 Lilly Co Eli Kinase inhibitors
US7776869B2 (en) * 2004-10-18 2010-08-17 Amgen Inc. Heteroaryl-substituted alkyne compounds and method of use
EP1992344A1 (en) 2007-05-18 2008-11-19 Institut Curie P38 alpha as a therapeutic target in pathologies linked to FGFR3 mutation
DK2571878T3 (da) * 2010-05-17 2019-02-11 Indian Incozen Therapeutics Pvt Ltd Hidtil ukendte 3,5-disubstituerede-3h-imidazo[4,5-b]pyridin- og 3,5- disubstituerede -3h-[1,2,3]triazol[4,5-b]pyridinforbindelser som modulatorer af proteinkinaser
AR083868A1 (es) * 2010-12-03 2013-03-27 Lilly Co Eli Compuestos de oxazol[5,4-b]piridin-5-ilo
HUE037928T2 (hu) * 2011-11-11 2018-09-28 Lilly Co Eli Kombinációs terápia petefészekrák ellen
US9587069B2 (en) * 2012-07-23 2017-03-07 The University Of Akron Polyisobutylene-based polyurethanes containing organically modified montmorillonite
US9067914B1 (en) 2013-12-10 2015-06-30 Genzyme Corporation Tropomyosin-related kinase (TRK) inhibitors
TN2017000234A1 (en) 2014-12-18 2018-10-19 Genzyme Corp Pharmaceutical formulations of tropomyosin related kinase (trk) inhibitors
MA41179A (fr) 2014-12-19 2017-10-24 Cancer Research Tech Ltd Composés inhibiteurs de parg
US9884868B2 (en) * 2015-03-02 2018-02-06 Rigel Pharmaceuticals, Inc. TGF-beta inhibitors
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
HRP20221196T1 (hr) 2017-10-05 2022-12-09 Fulcrum Therapeutics, Inc. Inhibitori p38 kinaze smanjuju ekspresiju dux4 i nizvodnih gena u cilju liječenja fshd
US10899869B2 (en) 2019-01-24 2021-01-26 The University Of Akron Glycerol containing polyurethanes and polyurethane nanocomposites
TW202112368A (zh) 2019-06-13 2021-04-01 荷蘭商法西歐知識產權股份有限公司 用於治療有關dux4表現之疾病的抑制劑組合

Family Cites Families (20)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
MX9300141A (es) * 1992-01-13 1994-07-29 Smithkline Beecham Corp Compuestos de imidazol novedosos, procedimiento para su preparacion y composiciones farmaceuticas que lo contienen.
DE19503806A1 (de) * 1994-02-11 1995-08-17 Bernhardt Apparatebau Gmbh Co Vorrichtung zum Aufblasen eines Behälters oder eines Schwimmkörpers, insbesondere einer Schwimmweste
US6426360B1 (en) * 1994-07-28 2002-07-30 G D Searle & Co. 4,5-substituted imidazolyl compounds for the treatment of inflammation
US5620999A (en) 1994-07-28 1997-04-15 Weier; Richard M. Benzenesulfonamide subtituted imidazolyl compounds for the treatment of inflammation
US5717100A (en) * 1995-10-06 1998-02-10 Merck & Co., Inc. Substituted imidazoles having anti-cancer and cytokine inhibitory activity
WO1998007425A1 (en) * 1996-08-21 1998-02-26 Smithkline Beecham Corporation Imidazole compounds, compositions and use
US6087496A (en) * 1998-05-22 2000-07-11 G. D. Searle & Co. Substituted pyrazoles suitable as p38 kinase inhibitors
US6180632B1 (en) * 1997-05-28 2001-01-30 Aventis Pharmaceuticals Products Inc. Quinoline and quinoxaline compounds which inhibit platelet-derived growth factor and/or p56lck tyrosine kinases
WO1999000130A1 (en) 1997-06-30 1999-01-07 Temple University - Of The Commonwealth System Of Higher Education Method for treating vulvar vestibulitis
AR016294A1 (es) * 1997-07-02 2001-07-04 Smithkline Beecham Corp Compuesto de imidazol sustituido, composicion farmaceutica que la contiene, su uso en la fabricacion de un medicamento y procedimiento para supreparacion
CA2314980A1 (en) * 1997-12-19 1999-07-01 Smithkline Beecham Corporation Compounds of heteroaryl substituted imidazole, their pharmaceutical compositions and uses
US6207687B1 (en) 1998-07-31 2001-03-27 Merck & Co., Inc. Substituted imidazoles having cytokine inhibitory activity
US6291457B1 (en) 1999-07-01 2001-09-18 Merck & Co., Inc. Compounds having cytokine inhibitory activity
US6608072B1 (en) * 1999-10-27 2003-08-19 Novartis Ag Thiazole compounds and their pharmaceutical use
GB0007405D0 (en) * 2000-03-27 2000-05-17 Smithkline Beecham Corp Compounds
BR0207990A (pt) 2001-03-09 2004-04-27 Pfizer Prod Inc Compostos antinflamatórios de triazolopiridinas
CA2444596A1 (en) 2001-04-16 2002-10-24 Tanabe Seiyaku Co., Ltd. Large conductance calcium-activated k channel opener
WO2003062215A1 (en) 2002-01-25 2003-07-31 Kylix Pharmaceuticals B.V. 4(hetero-) aryl substituted (thia-/oxa-/pyra) zoles for inhibition of tie-2
ATE323702T1 (de) 2002-08-06 2006-05-15 Astrazeneca Ab Kondensierte pyridine und pyrimidine mit tie2 (tek) aktivität
TWI332003B (en) * 2004-01-30 2010-10-21 Lilly Co Eli Kinase inhibitors

Also Published As

Publication number Publication date
EP1713805A1 (en) 2006-10-25
DOP2005000010A (es) 2005-11-15
NZ549780A (en) 2010-01-29
US20090036445A1 (en) 2009-02-05
WO2005075478A1 (en) 2005-08-18
CN1938302A (zh) 2007-03-28
CA2559128C (en) 2013-04-16
RU2006138606A (ru) 2008-05-10
ATE433449T1 (de) 2009-06-15
DE602005014848D1 (de) 2009-07-23
PL1713805T3 (pl) 2009-10-30
CA2559128A1 (en) 2005-08-18
RU2348635C2 (ru) 2009-03-10
US20090318443A1 (en) 2009-12-24
IL178103A (en) 2011-04-28
CY1109234T1 (el) 2014-07-02
TW200526660A (en) 2005-08-16
TWI332003B (en) 2010-10-21
AU2005210459B2 (en) 2010-10-21
ZA200607648B (en) 2008-06-25
PE20050689A1 (es) 2005-09-27
CN100516064C (zh) 2009-07-22
PT1713805E (pt) 2009-08-20
EP1713805B1 (en) 2009-06-10
AU2005210459A1 (en) 2005-08-18
US7582652B2 (en) 2009-09-01
SI1713805T1 (sl) 2009-10-31
ES2326819T3 (es) 2009-10-20
AR047466A1 (es) 2006-01-18
MY143516A (en) 2011-05-31
HK1100141A1 (en) 2007-09-07
UA85505C2 (en) 2009-01-26
SV2006002001A (es) 2006-02-15

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