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DE60134338D1 - Piperazin-derivate - Google Patents

Piperazin-derivate

Info

Publication number
DE60134338D1
DE60134338D1 DE60134338T DE60134338T DE60134338D1 DE 60134338 D1 DE60134338 D1 DE 60134338D1 DE 60134338 T DE60134338 T DE 60134338T DE 60134338 T DE60134338 T DE 60134338T DE 60134338 D1 DE60134338 D1 DE 60134338D1
Authority
DE
Germany
Prior art keywords
piperazin derivatives
piperazin
derivatives
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
DE60134338T
Other languages
English (en)
Inventor
David Reginald Adams
Jonathan Mark Bentley
James Edward Davidson
Claire Elizabeth Dawson
Ashley Roger George
Howard Langham Mansell
Patrizio Mattei
Jacques Mizrahi
Matthias Heinrich Nettekoven
Robert Mark Pratt
Jonathan Richard Roffey
Stephan Roever
Jean-Luc Specklin
Henri Stalder
Kerry Harrison
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Ligand UK Research Ltd
Original Assignee
F Hoffmann La Roche AG
Vernalis Research Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG, Vernalis Research Ltd filed Critical F Hoffmann La Roche AG
Application granted granted Critical
Publication of DE60134338D1 publication Critical patent/DE60134338D1/de
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/325—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
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    • C07D295/20—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carbonic acid, or sulfur or nitrogen analogues thereof
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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KR100623833B1 (ko) 2006-09-18
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BR0116201A (pt) 2004-03-02
US20020143020A1 (en) 2002-10-03
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GB0030710D0 (en) 2001-01-31
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ZA200304346B (en) 2004-09-03
JP4047724B2 (ja) 2008-02-13
CN1533382A (zh) 2004-09-29
ATE397595T1 (de) 2008-06-15
CA2430601C (en) 2008-05-06
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WO2002048124A3 (en) 2003-06-05
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AR035517A1 (es) 2004-06-02
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