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CL2016002312A1 - Modulador del receptor de andrógeno y usos de este. - Google Patents

Modulador del receptor de andrógeno y usos de este.

Info

Publication number
CL2016002312A1
CL2016002312A1 CL2016002312A CL2016002312A CL2016002312A1 CL 2016002312 A1 CL2016002312 A1 CL 2016002312A1 CL 2016002312 A CL2016002312 A CL 2016002312A CL 2016002312 A CL2016002312 A CL 2016002312A CL 2016002312 A1 CL2016002312 A1 CL 2016002312A1
Authority
CL
Chile
Prior art keywords
androgen receptor
receptor modulator
metastassic
trifluorometilpiridin
diazaespiro
Prior art date
Application number
CL2016002312A
Other languages
English (en)
Inventor
Nicholas D Smith
Mark R Herbert
Isan Chen
Jeffrey H Hager
Edna Chow Maneval
Original Assignee
Aragon Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=50029265&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2016002312(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Aragon Pharmaceuticals Inc filed Critical Aragon Pharmaceuticals Inc
Publication of CL2016002312A1 publication Critical patent/CL2016002312A1/es

Links

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    • A61K31/337—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having four-membered rings, e.g. taxol
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    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/4025—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil not condensed and containing further heterocyclic rings, e.g. cromakalim
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Abstract

<p>METODO PARA TRATAR CANCER DE PROSTATA RESISTENTE A LA CASTRACIÓN POSTERIOR AL TRATAMIENTO CON ACETATO DE ABIRATERONA, CANCER DE PROSTATA METASTASICO Y NO METASTÁSICO RESISTENTE A LA CASTRACIÓN, ENTRE OTROS, QUE COMPRENDE EL USO DE 4-[7-( 6-CIANO-5-TRIFLUOROMETILPIRIDIN-3-IL)-8-OXO-6-TIOXO-5,7-DIAZAESPIRO[3,4]OCT-5-IL]-2-FLUORO-N-METILBENZAMIDA (DIV. SOL. 1983-15). </p>
CL2016002312A 2013-01-15 2016-09-14 Modulador del receptor de andrógeno y usos de este. CL2016002312A1 (es)

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