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CL2008002717A1 - 3-(1-clorofenil)-7-oxo-6-[4-(2-oxo-1(2h)piridinil)fenil]-4,5,6,7-tetrahidro-1h-pirazolo[3,4-c]piridin-3-carboxamida y 3-(1-hidroxi-1-metil-etil)-1-(a-metoxi-fenil)-6-[4-(2-oxo-2h-piridin-1-il)-fenil]-1,4,5,6-tetrahidro-pirazolo[3,4-c]piridin-7-ona; composicion farmaceutica; combinacion farmaceutica y uso en el tratamiento de un desorden tromboembolico - Google Patents

3-(1-clorofenil)-7-oxo-6-[4-(2-oxo-1(2h)piridinil)fenil]-4,5,6,7-tetrahidro-1h-pirazolo[3,4-c]piridin-3-carboxamida y 3-(1-hidroxi-1-metil-etil)-1-(a-metoxi-fenil)-6-[4-(2-oxo-2h-piridin-1-il)-fenil]-1,4,5,6-tetrahidro-pirazolo[3,4-c]piridin-7-ona; composicion farmaceutica; combinacion farmaceutica y uso en el tratamiento de un desorden tromboembolico

Info

Publication number
CL2008002717A1
CL2008002717A1 CL2008002717A CL2008002717A CL2008002717A1 CL 2008002717 A1 CL2008002717 A1 CL 2008002717A1 CL 2008002717 A CL2008002717 A CL 2008002717A CL 2008002717 A CL2008002717 A CL 2008002717A CL 2008002717 A1 CL2008002717 A1 CL 2008002717A1
Authority
CL
Chile
Prior art keywords
oxo
phenyl
pyrazolo
pyridin
tetrahydro
Prior art date
Application number
CL2008002717A
Other languages
English (en)
Inventor
Li Yun-Long
L Quan Mimi
J Orwat Michael
J Pinto Donald
Han Wei
X Qiao Jennifer
y s lam Patrick
Stephanie
Original Assignee
Bristol Myers Squibb Pharma Company
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=23262376&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2008002717(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bristol Myers Squibb Pharma Company filed Critical Bristol Myers Squibb Pharma Company
Publication of CL2008002717A1 publication Critical patent/CL2008002717A1/es

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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
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    • A61J—CONTAINERS SPECIALLY ADAPTED FOR MEDICAL OR PHARMACEUTICAL PURPOSES; DEVICES OR METHODS SPECIALLY ADAPTED FOR BRINGING PHARMACEUTICAL PRODUCTS INTO PARTICULAR PHYSICAL OR ADMINISTERING FORMS; DEVICES FOR ADMINISTERING FOOD OR MEDICINES ORALLY; BABY COMFORTERS; DEVICES FOR RECEIVING SPITTLE
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    • A61K31/4365—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system having sulfur as a ring hetero atom, e.g. ticlopidine
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    • A61K31/437—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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Abstract

Compuestos derivados de pirazolo[3,4-c]piridina; composición farmacéutica; y uso en el tratamiento de un desorden tromboembólico (Div. Sol. 2175-02).
CL2008002717A 2001-09-21 2008-09-12 3-(1-clorofenil)-7-oxo-6-[4-(2-oxo-1(2h)piridinil)fenil]-4,5,6,7-tetrahidro-1h-pirazolo[3,4-c]piridin-3-carboxamida y 3-(1-hidroxi-1-metil-etil)-1-(a-metoxi-fenil)-6-[4-(2-oxo-2h-piridin-1-il)-fenil]-1,4,5,6-tetrahidro-pirazolo[3,4-c]piridin-7-ona; composicion farmaceutica; combinacion farmaceutica y uso en el tratamiento de un desorden tromboembolico CL2008002717A1 (es)

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