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CA978946A - .alpha.-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES - Google Patents

.alpha.-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES

Info

Publication number
CA978946A
CA978946A CA161,413A CA161413A CA978946A CA 978946 A CA978946 A CA 978946A CA 161413 A CA161413 A CA 161413A CA 978946 A CA978946 A CA 978946A
Authority
CA
Canada
Prior art keywords
aryl
alpha
piperidinoalkanol derivatives
substituted
substituted piperidinoalkanol
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA161,413A
Other languages
English (en)
Other versions
CA161413S (en
Inventor
C. Richard Kinsolving
Albert A. Carr
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Richardson Vicks Ltd Canada
Original Assignee
Richardson Merrell Canada Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22829539&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CA978946(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Richardson Merrell Canada Ltd filed Critical Richardson Merrell Canada Ltd
Application granted granted Critical
Publication of CA978946A publication Critical patent/CA978946A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/68—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D211/70—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/10—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms
    • C07D211/14—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with radicals containing only carbon and hydrogen atoms attached to ring carbon atoms with hydrocarbon or substituted hydrocarbon radicals attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D211/00—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings
    • C07D211/04—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D211/06—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D211/08—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms
    • C07D211/18—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D211/20—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms
    • C07D211/22—Heterocyclic compounds containing hydrogenated pyridine rings, not condensed with other rings with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon or substituted hydrocarbon radicals directly attached to ring carbon atoms with substituted hydrocarbon radicals attached to ring carbon atoms with hydrocarbon radicals, substituted by singly bound oxygen or sulphur atoms by oxygen atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
CA161,413A 1972-01-28 1973-01-16 .alpha.-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES Expired CA978946A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US22182172A 1972-01-28 1972-01-28

Publications (1)

Publication Number Publication Date
CA978946A true CA978946A (en) 1975-12-02

Family

ID=22829539

Family Applications (1)

Application Number Title Priority Date Filing Date
CA161,413A Expired CA978946A (en) 1972-01-28 1973-01-16 .alpha.-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES

Country Status (26)

Country Link
JP (1) JPS5115035B2 (cs)
AR (1) AR195314A1 (cs)
AT (2) AT321917B (cs)
AU (1) AU467361B2 (cs)
BE (1) BE794597A (cs)
CA (1) CA978946A (cs)
CH (2) CH587820A5 (cs)
CS (1) CS177834B2 (cs)
DD (1) DD103239A5 (cs)
DE (1) DE2303306C3 (cs)
DK (1) DK136713B (cs)
ES (1) ES410731A1 (cs)
FR (1) FR2181690B1 (cs)
GB (1) GB1413138A (cs)
HU (1) HU166477B (cs)
IE (1) IE36983B1 (cs)
IL (1) IL41060A (cs)
LU (1) LU66916A1 (cs)
NL (1) NL175410C (cs)
NO (1) NO140057C (cs)
PH (1) PH10264A (cs)
PL (1) PL89095B1 (cs)
SE (1) SE382058B (cs)
SU (1) SU464997A3 (cs)
YU (1) YU36013B (cs)
ZA (1) ZA728544B (cs)

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8067605B2 (en) * 2004-09-17 2011-11-29 Albany Molecular Research, Inc. Process for production of piperidine derivatives

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3941795A (en) 1974-02-08 1976-03-02 Richardson-Merrell Inc. α-ARYL-4-SUBSTITUTED PIPERIDINOALKANOL DERIVATIVES
US4254130A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
US4254129A (en) * 1979-04-10 1981-03-03 Richardson-Merrell Inc. Piperidine derivatives
IT1200123B (it) * 1985-09-27 1989-01-05 Ind Chimica Srl Procedimento per la preparazione di alfa-(p-terbutilfenil)-4-(idrossidifenilmetil)-1-piperidinobutanolo
US4742175A (en) * 1986-05-07 1988-05-03 Merrell Dow Pharmaceuticals Inc. Preparation of polymorphically pure terfenadine
JPS63101760U (cs) * 1986-12-19 1988-07-02
IT1205685B (it) * 1987-05-26 1989-03-31 Erregierre Spa Processo per la preparazione di alfa-(alchilfenil)-4-(idrossi difenilmetil)-1-piperidina butanolo
IL93499A0 (en) * 1989-02-28 1990-11-29 Merrell Dow Pharma Preparation of the low melting polymorphic form of terfenadine
CA2015390A1 (en) * 1989-05-01 1990-11-01 Frederick J. Mccarty Process for the preparation of the high melting polymorphic of terfenadine
DE3917241A1 (de) * 1989-05-26 1990-11-29 Schaper & Bruemmer Gmbh 4-(hydroxydiphenylmethyl)-1-piperidyl-phenylalkan-derivate
EP0596120A4 (en) * 1991-08-09 1994-07-06 Yoshitomi Pharmaceutical Thiophene compound.
HUP9801254A3 (en) * 1995-05-08 1998-09-28 Aventis Pharmaceuticals Inc Br Alpha-(substituted alkylphenyl)-4-(hydroxydiphenylmethyl)-1-piperidine butanol derivatives, their preparation and their use as anti-histamines, anti-allergy agents and bronchodilators
ES2216191T3 (es) * 1997-03-11 2004-10-16 Aventis Pharmaceuticals Inc. Procedimiento para preparar acido 4-(4-(hidroxidifenil)-1-piperidinil)-1-hidroxibutil)-alfa,alfa-dimetilfenilacetico y derivados fosforilados.
US8153385B2 (en) 2004-10-18 2012-04-10 Reverse Proteomics Research Institute Co., Ltd. Target protein and target gene in drug designing and screening method

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3081303A (en) * 1961-10-13 1963-03-12 Searle & Co 1-aminoalkyl-alpha, alpha-diphenylpiperidine-methanols
GB1242169A (en) * 1969-04-09 1971-08-11 Ucb Sa Piperidine derivatives

Cited By (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8067605B2 (en) * 2004-09-17 2011-11-29 Albany Molecular Research, Inc. Process for production of piperidine derivatives

Also Published As

Publication number Publication date
GB1413138A (en) 1975-11-05
FR2181690A1 (cs) 1973-12-07
DE2303306C3 (de) 1979-05-31
JPS4885578A (cs) 1973-11-13
JPS5115035B2 (cs) 1976-05-13
NL7300873A (cs) 1973-07-31
ES410731A1 (es) 1976-04-01
LU66916A1 (cs) 1973-07-27
DE2303306A1 (de) 1973-08-02
YU36013B (en) 1981-11-13
NL175410B (nl) 1984-06-01
ZA728544B (en) 1974-02-27
IE36983B1 (en) 1977-04-13
DD103239A5 (cs) 1974-01-12
DK136713B (da) 1977-11-14
PL89095B1 (cs) 1976-10-30
SE382058B (sv) 1976-01-12
DE2303306B2 (de) 1978-09-28
IL41060A (en) 1975-06-25
SU464997A3 (ru) 1975-03-25
AU467361B2 (en) 1975-11-27
AT323742B (de) 1975-07-25
IE36983L (en) 1973-07-28
BE794597A (fr) 1973-05-16
IL41060A0 (en) 1973-02-28
AR195314A1 (es) 1973-09-28
AT321917B (de) 1975-04-25
NO140057C (no) 1979-07-04
HU166477B (cs) 1975-03-28
YU3473A (en) 1981-02-28
FR2181690B1 (cs) 1976-05-14
AU4989372A (en) 1974-06-13
CH587820A5 (cs) 1977-05-13
DK136713C (cs) 1978-05-01
CH593259A5 (cs) 1977-11-30
NO140057B (no) 1979-03-19
NL175410C (nl) 1984-11-01
CS177834B2 (cs) 1977-08-31
PH10264A (en) 1976-10-20

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