BRPI0807799A2 - " derivados de 2-piperazin-1-il-3h-imidazo{4,5-b]piridina". - Google Patents

" derivados de 2-piperazin-1-il-3h-imidazo{4,5-b]piridina".

Info

Publication number: BRPI0807799A2
Authority: BR; Brazil
Prior art keywords: piperazin; imidazo; compounds; pyridine derivatives; concerned
Prior art date: 2007-01-25

Application number

BRPI0807799-1A2A

Other languages

English (en)

Inventor

Frans Eduard Janssens

Jerome Emile Georges Guillemont

Francois Maria Sommen

Jean-Francois Bonfanti

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-01-25

Filing date

2008-01-24

Publication date

2014-06-03

2008-01-24 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2014-06-03 Publication of BRPI0807799A2 publication Critical patent/BRPI0807799A2/pt

2021-04-06 Publication of BRPI0807799B1 publication Critical patent/BRPI0807799B1/pt

2021-05-25 Publication of BRPI0807799B8 publication Critical patent/BRPI0807799B8/pt

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nutrition Science (AREA)
Epidemiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)

BRPI0807799A 2007-01-25 2008-01-24 derivados de 2-piperazin-1-il-3h-imidazo[4,5-b]piridina, composição farmacêutica que os compreende, seu processo de preparação e uso BRPI0807799B8 (pt)

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
EP07101153		2007-01-25
EP07101153.0		2007-01-25
PCT/EP2008/050818 WO2008090200A2 (en)	2007-01-25	2008-01-24	2- piperazin-1-yl-3h-imidazo[4,5-b]pyridine derivatives

Publications (3)

Publication Number	Publication Date
BRPI0807799A2 true BRPI0807799A2 (pt)	2014-06-03
BRPI0807799B1 BRPI0807799B1 (pt)	2021-04-06
BRPI0807799B8 BRPI0807799B8 (pt)	2021-05-25

Family

ID=38179852

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
BRPI0807799A BRPI0807799B8 (pt)	2007-01-25	2008-01-24	derivados de 2-piperazin-1-il-3h-imidazo[4,5-b]piridina, composição farmacêutica que os compreende, seu processo de preparação e uso

Country Status (18)

Country	Link
US (1)	US7994173B2 (pt)
EP (1)	EP2121683B1 (pt)
JP (1)	JP5437814B2 (pt)
KR (1)	KR101484027B1 (pt)
CN (1)	CN101600717B (pt)
AT (1)	ATE522530T1 (pt)
AU (1)	AU2008208820B2 (pt)
BR (1)	BRPI0807799B8 (pt)
CA (1)	CA2671857C (pt)
EA (1)	EA016422B1 (pt)
ES (1)	ES2372433T3 (pt)
HK (1)	HK1136288A1 (pt)
IL (1)	IL199986A (pt)
MX (1)	MX2009007912A (pt)
PL (1)	PL2121683T3 (pt)
UA (1)	UA101149C2 (pt)
WO (1)	WO2008090200A2 (pt)
ZA (1)	ZA200905205B (pt)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP2567959B1 (en)	2011-09-12	2014-04-16	Sanofi	6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8716313D0 (en) *	1987-07-10	1987-08-19	Janssen Pharmaceutica Nv	2-(heterocyclylalkyl)imidazopyridines
ES2038532B1 (es) *	1991-05-10	1994-02-16	Espanola Prod Quimicos	Procedimiento de preparacion de nuevos derivados de 2-piperacinilbecimidazol.
KR100715344B1 (ko) *	1999-11-23	2007-05-08	얀센 파마슈티카 엔.브이.	기저부 이완을 위한 5ｈｔ3 효능제의 용도
TWI225488B (en)	1999-12-21	2004-12-21	Janssen Pharmaceutica Nv	Derivatives of homopiperidinyl substituted benzimidazole analogues

2008
- 2008-01-24 AT AT08708157T patent/ATE522530T1/de not_active IP Right Cessation
- 2008-01-24 UA UAA200906700A patent/UA101149C2/ru unknown
- 2008-01-24 PL PL08708157T patent/PL2121683T3/pl unknown
- 2008-01-24 JP JP2009546755A patent/JP5437814B2/ja not_active Expired - Fee Related
- 2008-01-24 CA CA2671857A patent/CA2671857C/en active Active
- 2008-01-24 CN CN2008800019424A patent/CN101600717B/zh active Active
- 2008-01-24 EA EA200970710A patent/EA016422B1/ru not_active IP Right Cessation
- 2008-01-24 ES ES08708157T patent/ES2372433T3/es active Active
- 2008-01-24 WO PCT/EP2008/050818 patent/WO2008090200A2/en active Application Filing
- 2008-01-24 US US12/523,936 patent/US7994173B2/en not_active Expired - Fee Related
- 2008-01-24 BR BRPI0807799A patent/BRPI0807799B8/pt not_active IP Right Cessation
- 2008-01-24 MX MX2009007912A patent/MX2009007912A/es active IP Right Grant
- 2008-01-24 EP EP08708157A patent/EP2121683B1/en active Active
- 2008-01-24 AU AU2008208820A patent/AU2008208820B2/en not_active Ceased
- 2008-01-24 KR KR1020097014965A patent/KR101484027B1/ko active IP Right Grant
2009
- 2009-07-21 IL IL199986A patent/IL199986A/en active IP Right Grant
- 2009-07-24 ZA ZA200905205A patent/ZA200905205B/xx unknown
2010
- 2010-03-24 HK HK10103088.5A patent/HK1136288A1/xx not_active IP Right Cessation

Also Published As

Publication number	Publication date
ES2372433T3 (es)	2012-01-19
IL199986A0 (en)	2010-04-15
CN101600717A (zh)	2009-12-09
KR20090101464A (ko)	2009-09-28
CA2671857A1 (en)	2008-07-31
JP5437814B2 (ja)	2014-03-12
EP2121683B1 (en)	2011-08-31
CN101600717B (zh)	2013-03-13
BRPI0807799B1 (pt)	2021-04-06
EP2121683A2 (en)	2009-11-25
WO2008090200A2 (en)	2008-07-31
UA101149C2 (en)	2013-03-11
IL199986A (en)	2013-03-24
AU2008208820B2 (en)	2012-09-20
CA2671857C (en)	2013-11-19
MX2009007912A (es)	2009-07-31
ZA200905205B (en)	2010-09-29
KR101484027B1 (ko)	2015-01-19
HK1136288A1 (pt)	2010-06-25
BRPI0807799B8 (pt)	2021-05-25
US7994173B2 (en)	2011-08-09
ATE522530T1 (de)	2011-09-15
JP2010516740A (ja)	2010-05-20
US20100004260A1 (en)	2010-01-07
EA200970710A1 (ru)	2009-12-30
AU2008208820A1 (en)	2008-07-31
PL2121683T3 (pl)	2012-01-31
EA016422B1 (ru)	2012-04-30
WO2008090200A3 (en)	2008-09-04

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Legal Events

Date	Code	Title	Description
2018-04-24	B06F	Objections, documents and/or translations needed after an examination request according [chapter 6.6 patent gazette]
2018-09-18	B06T	Formal requirements before examination [chapter 6.20 patent gazette]
2019-10-01	B07D	Technical examination (opinion) related to article 229 of industrial property law [chapter 7.4 patent gazette]	Free format text: DE ACORDO COM O ARTIGO 229-C DA LEI NO 10196/2001, QUE MODIFICOU A LEI NO 9279/96, A CONCESSAO DA PATENTE ESTA CONDICIONADA A ANUENCIA PREVIA DA ANVISA. CONSIDERANDO A APROVACAO DOS TERMOS DO PARECER NO 337/PGF/EA/2010, BEM COMO A PORTARIA INTERMINISTERIAL NO 1065 DE 24/05/2012, ENCAMINHA-SE O PRESENTE PEDIDO PARA AS PROVIDENCIAS CABIVEIS.
2020-08-11	B07E	Notification of approval relating to section 229 industrial property law [chapter 7.5 patent gazette]
2020-11-10	B06A	Patent application procedure suspended [chapter 6.1 patent gazette]
2021-02-23	B09A	Decision: intention to grant [chapter 9.1 patent gazette]
2021-04-06	B16A	Patent or certificate of addition of invention granted [chapter 16.1 patent gazette]	Free format text: PRAZO DE VALIDADE: 10 (DEZ) ANOS CONTADOS A PARTIR DE 06/04/2021, OBSERVADAS AS CONDICOES LEGAIS.
2021-05-25	B16C	Correction of notification of the grant [chapter 16.3 patent gazette]	Free format text: PRAZO DE VALIDADE: 20 (VINTE) ANOS CONTADOS A PARTIR DE 24/01/2008 OBSERVADAS AS CONDICOES LEGAIS. PATENTE CONCEDIDA CONFORME ADI 5.529/DF
2023-11-14	B21F	Lapse acc. art. 78, item iv - on non-payment of the annual fees in time	Free format text: REFERENTE A 16A ANUIDADE.
2024-03-05	B24J	Lapse because of non-payment of annual fees (definitively: art 78 iv lpi, resolution 113/2013 art. 12)	Free format text: EM VIRTUDE DA EXTINCAO PUBLICADA NA RPI 2758 DE 14-11-2023 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDA A EXTINCAO DA PATENTE E SEUS CERTIFICADOS, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013.