BR0002577A - Suspensões orais de trovafloxacina - Google Patents
Suspensões orais de trovafloxacinaInfo
- Publication number
- BR0002577A BR0002577A BR0002577-1A BR0002577A BR0002577A BR 0002577 A BR0002577 A BR 0002577A BR 0002577 A BR0002577 A BR 0002577A BR 0002577 A BR0002577 A BR 0002577A
- Authority
- BR
- Brazil
- Prior art keywords
- crystals
- trovafloxacin
- novel
- suspensions
- oral suspensions
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Cosmetics (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Patente de Invenção:<B>"SUSPENSõES ORAIS DE TROVAFLOXACINA"<D>. A invenção refere-se a suspensões para administração oral compreendendo novos cristais zwitteriónicos de trovafloxacina, e a processos para preparação dos referidos cristais. Esta invenção refere-se ainda a outras composições farmacêuticas compreendendo os referidos novos cristais, e aos métodos de utilização dessas suspensões, e dos novos cristais, em tais outras formas de dosagem, para tratar infecções bacterianas em mamíferos.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US13746399P | 1999-06-04 | 1999-06-04 |
Publications (1)
Publication Number | Publication Date |
---|---|
BR0002577A true BR0002577A (pt) | 2001-01-02 |
Family
ID=22477550
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR0002577-1A BR0002577A (pt) | 1999-06-04 | 2000-06-05 | Suspensões orais de trovafloxacina |
Country Status (10)
Country | Link |
---|---|
US (1) | US6239141B1 (pt) |
EP (1) | EP1057828B1 (pt) |
JP (1) | JP3465820B2 (pt) |
AT (1) | ATE234835T1 (pt) |
BR (1) | BR0002577A (pt) |
CA (1) | CA2311112A1 (pt) |
DE (1) | DE60001687T2 (pt) |
DK (1) | DK1057828T3 (pt) |
ES (1) | ES2194677T3 (pt) |
PT (1) | PT1057828E (pt) |
Families Citing this family (18)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1226138B1 (en) * | 1999-10-08 | 2004-12-29 | Affinium Pharmaceuticals, Inc. | Fab i inhibitors |
EP1372662A1 (en) * | 2001-03-05 | 2004-01-02 | Ortho-Mcneil Pharmaceutical, Inc. | Taste masked liquid pharmaceutical compositions |
EP1560584B1 (en) * | 2001-04-06 | 2009-01-14 | Affinium Pharmaceuticals, Inc. | Fab i inhibitors |
US20030068829A1 (en) * | 2001-06-25 | 2003-04-10 | Symyx Technologies, Inc. | High throughput crystallographic screening of materials |
CA2453182A1 (en) * | 2001-07-10 | 2003-01-23 | Meredith L. Greene | Crystalline thiazine oxazolidinones |
PL216524B1 (pl) | 2001-08-15 | 2014-04-30 | Upjohn Co | Kryształ obejmujący sól N-[2-(dietyloamino) etylo]-5-[(5-fluoro-1,2-dihydro-2-okso-3H-indolo-3-ylideno) metylo]-2,4-dimetylo-1H-pirolo-3-karboksyamidu z kwasem L-jabłkowym i zawierająca go kompozycja |
CN100337630C (zh) * | 2002-03-12 | 2007-09-19 | 布里斯托尔-迈尔斯斯奎布公司 | 可口的口服悬浮液及其制备方法 |
WO2003093322A2 (en) * | 2002-04-30 | 2003-11-13 | The Population Council, Inc. | Carrageenan based antimicrobial compositions |
US8367098B2 (en) * | 2002-04-30 | 2013-02-05 | The Population Council, Inc. | Unique combinations of antimicrobial compositions |
DK1575951T3 (da) | 2002-12-06 | 2014-09-15 | Debiopharm Int Sa | Heterocykliske forbindelser, fremgangsmåder til fremstilling deraf og deres anvendelse i terapi |
CA2519429C (en) | 2003-03-17 | 2013-08-06 | Affinium Pharmaceuticals, Inc. | Pharmaceutical compositions comprising inhibitors of fab i and further antibiotics |
JP2006528182A (ja) * | 2003-07-18 | 2006-12-14 | サンタラス インコーポレイティッド | 薬学的製剤および酸に起因する消化器疾患の治療法 |
US8450307B2 (en) * | 2004-06-04 | 2013-05-28 | Affinium Pharmaceuticals, Inc. | Therapeutic agents, and methods of making and using the same |
US20090156578A1 (en) * | 2005-12-05 | 2009-06-18 | PAULS Henry | 3-Heterocyclylacrylamide Compounds as Fab I Inhibitors and Antibacterial Agents |
WO2008009122A1 (en) | 2006-07-20 | 2008-01-24 | Affinium Pharmaceuticals, Inc. | Acrylamide derivatives as fab i inhibitors |
EP3255045A1 (en) | 2007-02-16 | 2017-12-13 | Debiopharm International SA | Salts, prodrugs and polymorphs of fab i inhibitors |
ME03392B (me) | 2012-06-19 | 2020-01-20 | Debiopharm Int Sa | Prolek derivati (e)-n-meтil-n-( (з-метi lbenzofuran-2-il)meтil)-3-(7 -okso-5 ,6, 7,8-тетrанidr0-1,8-nafтiridin-3-il)akrilamida |
CN108778286A (zh) | 2016-02-26 | 2018-11-09 | 德彪药业国际股份公司 | 用于治疗糖尿病足感染的药物 |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US5164402A (en) | 1989-08-16 | 1992-11-17 | Pfizer Inc | Azabicyclo quinolone and naphthyridinone carboxylic acids |
US5266559A (en) | 1989-10-27 | 1993-11-30 | Firmenich S.A. | Use of unsaturated macrocyclic lactones as perfuming ingredients |
US5391763A (en) | 1990-07-11 | 1995-02-21 | Pfizer Inc. | 3-aza-bicyclo[3.1.0]hexanes which are intermediates for anti-bacterial azabicyclo quinolone carboxylic acids |
TW271400B (pt) | 1992-07-30 | 1996-03-01 | Pfizer | |
JP3145715B2 (ja) | 1995-06-06 | 2001-03-12 | ファイザー・インコーポレーテッド | 無水7−([1α,5α,6α]−6−アミノ−3−アザビシクロ[3.1.0]ヘキサ−3−イル)−6−フルオロ−1−(2,4−ジフルオロフェニル)−1,4−ジヒドロ−4−オキソ−1,8−ナフチリディン−3−カルボン酸メタンスルホン酸塩の新規な結晶形態 |
TR199800339T1 (xx) * | 1995-08-29 | 1998-06-22 | Pfizer Inc. | Trovafloksasinin melez iyonik bi�imleri. |
RU2151152C1 (ru) * | 1995-08-29 | 2000-06-20 | Пфайзер Инк. | Полиморфы 6-n-(l-ala-l-ala)-тровафлоксацина |
US6114531A (en) * | 1998-07-28 | 2000-09-05 | Pfizer Inc. | Process for preparing quinolone and naphthyridone carboxylic acids |
-
2000
- 2000-05-05 US US09/565,420 patent/US6239141B1/en not_active Expired - Fee Related
- 2000-05-16 JP JP2000142971A patent/JP3465820B2/ja not_active Expired - Fee Related
- 2000-05-30 ES ES00304550T patent/ES2194677T3/es not_active Expired - Lifetime
- 2000-05-30 EP EP00304550A patent/EP1057828B1/en not_active Expired - Lifetime
- 2000-05-30 DK DK00304550T patent/DK1057828T3/da active
- 2000-05-30 DE DE60001687T patent/DE60001687T2/de not_active Expired - Fee Related
- 2000-05-30 AT AT00304550T patent/ATE234835T1/de not_active IP Right Cessation
- 2000-05-30 PT PT00304550T patent/PT1057828E/pt unknown
- 2000-06-02 CA CA002311112A patent/CA2311112A1/en not_active Abandoned
- 2000-06-05 BR BR0002577-1A patent/BR0002577A/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
DE60001687T2 (de) | 2003-12-18 |
DE60001687D1 (de) | 2003-04-24 |
PT1057828E (pt) | 2003-07-31 |
ATE234835T1 (de) | 2003-04-15 |
DK1057828T3 (da) | 2003-07-14 |
EP1057828A3 (en) | 2001-05-16 |
EP1057828B1 (en) | 2003-03-19 |
EP1057828A2 (en) | 2000-12-06 |
US6239141B1 (en) | 2001-05-29 |
ES2194677T3 (es) | 2003-12-01 |
CA2311112A1 (en) | 2000-12-04 |
JP3465820B2 (ja) | 2003-11-10 |
JP2000344770A (ja) | 2000-12-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 5A, 6A E 7A ANUIDADES. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1913 DE 04/09/2007. |