AU2001269063A1 - Shortened synthesis of 3,3-diarylpropylamine derivatives - Google Patents

Shortened synthesis of 3,3-diarylpropylamine derivatives

Info

Publication number: AU2001269063A1
Authority: AU; Australia
Prior art keywords: shortened synthesis; diarylpropylamine; derivatives; diarylpropylamine derivatives; shortened
Prior art date: 2000-06-14
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Granted

Application number

AU2001269063A

Other versions

AU2001269063B2 (en

Inventor

Claus Meese

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

UCB Pharma GmbH

Original Assignee

Schwarz Pharma AG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-06-14

Filing date

2001-06-11

Publication date

2002-03-14

2000-06-14 Priority claimed from DE10028443A external-priority patent/DE10028443C1/en

2001-06-11 Application filed by Schwarz Pharma AG filed Critical Schwarz Pharma AG

2002-03-14 Publication of AU2001269063A1 publication Critical patent/AU2001269063A1/en

2005-03-24 Application granted granted Critical

2005-03-24 Publication of AU2001269063B2 publication Critical patent/AU2001269063B2/en

2021-06-11 Anticipated expiration legal-status Critical

Status Ceased legal-status Critical Current

Applications Claiming Priority (3)

Application Number	Priority Date	Filing Date	Title
DE10028443.4		2000-06-14
DE10028443A DE10028443C1 (en)	2000-06-14	2000-06-14	Production of optically active 3,3-diaryl-propylamine derivatives comprises six step process from 4-hydroxybenzoic acid or alkyl 4-hydroxybenzoate and cinnamic acid
PCT/EP2001/006577 WO2001096279A1 (en)	2000-06-14	2001-06-11	Shortened synthesis of 3,3-diarylpropylamine derivatives

Publications (2)

Publication Number	Publication Date
AU2001269063A1 true AU2001269063A1 (en)	2002-03-14
AU2001269063B2 AU2001269063B2 (en)	2005-03-24

Family

ID=7645152

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
AU6906301A Pending AU6906301A (en)	2000-06-14	2001-06-11	Shortened synthesis of 3,3-diarylpropylamine derivatives
AU2001269063A Ceased AU2001269063B2 (en)	2000-06-14	2001-06-11	Shortened synthesis of 3,3-diarylpropylamine derivatives

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
AU6906301A Pending AU6906301A (en)	2000-06-14	2001-06-11	Shortened synthesis of 3,3-diarylpropylamine derivatives

Country Status (24)

Country	Link
US (1)	US6809214B2 (en)
EP (1)	EP1289929B1 (en)
JP (2)	JP4002180B2 (en)
KR (1)	KR100580568B1 (en)
CN (1)	CN1234679C (en)
AT (1)	ATE368640T1 (en)
AU (2)	AU6906301A (en)
BR (1)	BR0111266A (en)
CA (1)	CA2412047C (en)
CZ (1)	CZ20023665A3 (en)
DE (2)	DE10028443C1 (en)
ES (1)	ES2290153T3 (en)
HK (1)	HK1050518A1 (en)
HU (1)	HUP0204563A3 (en)
IL (2)	IL151595A0 (en)
IS (1)	IS6534A (en)
MX (1)	MXPA02009643A (en)
NO (1)	NO20025967L (en)
NZ (1)	NZ521265A (en)
PL (1)	PL360845A1 (en)
RU (1)	RU2270188C2 (en)
SK (1)	SK142003A3 (en)
WO (1)	WO2001096279A1 (en)
ZA (1)	ZA200207204B (en)

Families Citing this family (19)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
EP0957073A1 (en)	1998-05-12	1999-11-17	Schwarz Pharma Ag	Novel derivatives of 3,3-diphenylpropylamines
DE10315917A1 (en) *	2003-04-08	2004-11-18	Schwarz Pharma Ag	Highly pure bases of 3,3-diphenylpropylamine monoesters
WO2005012227A2 (en) *	2003-08-05	2005-02-10	Ranbaxy Laboratories Limited	Process for preparation of 2-(3-diisopropylamino-1-phenylpropyl)-4-hydroxymethyl-phenol, a metabolite of tolterodine
JP4513535B2 (en) *	2004-12-03	2010-07-28	住友化学株式会社	Method for producing tolterodine
EP1843999A1 (en) *	2005-01-10	2007-10-17	Teva Pharmaceutical Industries Ltd	Process for preparing tolterodine tartrate
US8344176B2 (en) *	2006-05-31	2013-01-01	Schwarz Pharma Ltd.	Synthesis of substituted hydroxymethyl phenols
PL2027103T3 (en)	2006-06-12	2014-12-31	Ucb Pharma Gmbh	New chiral intermediate, process for producing the same and its use in the manufacture of tolterodine, fesoterodine, or the active metabolite thereof
SI2281801T1 (en) *	2009-07-27	2014-04-30	Crystal Pharma, S.A.U.	Process for obtaining 3,3-diphenylpropylamines
IT1396373B1 (en) *	2009-10-29	2012-11-19	Dipharma Francis Srl	PROCEDURE FOR THE PREPARATION OF FESOTERODINE.
EP2364966A1 (en)	2010-03-09	2011-09-14	LEK Pharmaceuticals d.d.	Process for preparation of 3-(2-hydroxy-5-substituted phenyl)-3-phenylpropylamines, intermediates for making hydroxytolterodine
US20110282094A1 (en)	2010-05-11	2011-11-17	Intas Pharmaceuticals Limited	Process for preparation of phenolic monoesters of hydroxymethyl phenols
IT1401451B1 (en)	2010-06-10	2013-07-26	Chemi Spa	NEW PROCESS OF PREPARATION OF 2-HYDROXY-4-PHENYL-3,4-DIHYDRO-2H-CHROMEN-6-IL-METHANOL E (R) -2- [3- (DIISOPROPYLAMINOUS) -1-PHENYLPROPYL] -4- ( hydroxymethyl) Phenol.
WO2011158257A1 (en) *	2010-06-18	2011-12-22	Panacea Biotec Ltd	Preparation process of fesoterodine and intermediates
IT1403094B1 (en)	2010-12-09	2013-10-04	Dipharma Francis Srl	PROCEDURE FOR THE PREPARATION OF FESOTERODINA OR ITS SALT
JP6234999B2 (en)	2012-05-04	2017-11-22	クリスタルファルマ、エセ、ア、ウＣｒｙｓｔａｌＰｈａｒｍａ，Ｓ．Ａ．Ｕ．	Process for preparing optically active 3,3-diphenylpropylamine
ES2569201T3 (en)	2012-06-14	2016-05-09	Ratiopharm Gmbh	Desfesoterodine salts
ITMI20121232A1 (en)	2012-07-16	2014-01-17	Cambrex Profarmaco Milano Srl	PROCEDURE FOR THE PREPARATION OF 2- (3-N, N-DIISOPROPYLAMINO-1-PHENYLPROPYL) -4-HYDROXYMETHYL-PHENOL AND ITS DERIVATIVES
CN103193747A (en) *	2013-04-18	2013-07-10	中国药科大学	Method for preparing fesoterodine fumarate intermediate
WO2017137955A1 (en)	2016-02-14	2017-08-17	Celestis Pharmaceuticals Pvt. Ltd.	Novel (r) and rac 3-(2-(allyloxy)-5-methylphenyl)-n,n-diisopropyl-3- phenylpropan-1-amine and its use for synthesis of (r) and rac-2-(3- (diisopropylamino)-1-phenylpropyl)-4-(hydroxymethyl)phenol

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
SE8800207D0 (en) *	1988-01-22	1988-01-22	Kabivitrum Ab	NEW AMINES, THEIR USE AND MANUFACTURING
SE9203318D0 (en) *	1992-11-06	1992-11-06	Kabi Pharmacia Ab	NOVEL 3,3-DIPHENYL PROPYLAMINES, THEIR USE AND PREPARATION
KR20000057548A (en) *	1996-12-13	2000-09-25	알프레드 엘. 미첼슨	Optically transmissive material and bond
SE9701144D0 (en) *	1997-03-27	1997-03-27	Pharmacia & Upjohn Ab	Novel compounds, their use and preparation
JP3913329B2 (en) *	1997-09-11	2007-05-09	株式会社クラレ	Optical resolution method of (±) -chromancarboxylic acid
EP0957073A1 (en) *	1998-05-12	1999-11-17	Schwarz Pharma Ag	Novel derivatives of 3,3-diphenylpropylamines
DE19955190A1 (en) *	1999-11-16	2001-06-21	Sanol Arznei Schwarz Gmbh	Stable salts of novel derivatives of 3,3-diphenylpropylamines

2000
- 2000-06-14 DE DE10028443A patent/DE10028443C1/en not_active Expired - Fee Related
2001
- 2001-06-11 HU HU0204563A patent/HUP0204563A3/en unknown
- 2001-06-11 KR KR1020027013004A patent/KR100580568B1/en not_active IP Right Cessation
- 2001-06-11 AT AT01947355T patent/ATE368640T1/en not_active IP Right Cessation
- 2001-06-11 RU RU2002132900/04A patent/RU2270188C2/en not_active IP Right Cessation
- 2001-06-11 CA CA002412047A patent/CA2412047C/en not_active Expired - Fee Related
- 2001-06-11 DE DE50112793T patent/DE50112793D1/en not_active Expired - Fee Related
- 2001-06-11 IL IL15159501A patent/IL151595A0/en active IP Right Grant
- 2001-06-11 EP EP01947355A patent/EP1289929B1/en not_active Expired - Lifetime
- 2001-06-11 ES ES01947355T patent/ES2290153T3/en not_active Expired - Lifetime
- 2001-06-11 AU AU6906301A patent/AU6906301A/en active Pending
- 2001-06-11 MX MXPA02009643A patent/MXPA02009643A/en active IP Right Grant
- 2001-06-11 CZ CZ20023665A patent/CZ20023665A3/en unknown
- 2001-06-11 SK SK14-2003A patent/SK142003A3/en unknown
- 2001-06-11 BR BR0111266-0A patent/BR0111266A/en not_active IP Right Cessation
- 2001-06-11 AU AU2001269063A patent/AU2001269063B2/en not_active Ceased
- 2001-06-11 WO PCT/EP2001/006577 patent/WO2001096279A1/en active IP Right Grant
- 2001-06-11 US US10/297,778 patent/US6809214B2/en not_active Expired - Fee Related
- 2001-06-11 PL PL36084501A patent/PL360845A1/en unknown
- 2001-06-11 NZ NZ521265A patent/NZ521265A/en unknown
- 2001-06-11 CN CNB018095259A patent/CN1234679C/en not_active Expired - Fee Related
- 2001-06-11 JP JP2002510423A patent/JP4002180B2/en not_active Expired - Fee Related
2002
- 2002-08-30 IS IS6534A patent/IS6534A/en unknown
- 2002-09-04 IL IL151595A patent/IL151595A/en not_active IP Right Cessation
- 2002-09-09 ZA ZA200207204A patent/ZA200207204B/en unknown
- 2002-12-12 NO NO20025967A patent/NO20025967L/en not_active Application Discontinuation
2003
- 2003-04-14 HK HK03102705A patent/HK1050518A1/en not_active IP Right Cessation
2007
- 2007-06-05 JP JP2007149492A patent/JP2007231024A/en active Pending

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