ATE151760T1 - Thiazolidin-derivate - Google Patents

Thiazolidin-derivate

Info

Publication number: ATE151760T1
Authority: AT; Austria
Prior art keywords: group; carbon atom; general formula; atom; single bond
Prior art date: 1987-02-23

Application number

AT91111866T

Other languages

English (en)

Inventor

Masaaki Toda

Shuichi Ohuchida

Hiroyuki Ohno

Original Assignee

Ono Pharmaceutical Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-02-23

Filing date

1988-02-16

Publication date

1997-05-15

1988-02-16 Application filed by Ono Pharmaceutical Co filed Critical Ono Pharmaceutical Co

1997-05-15 Application granted granted Critical

1997-05-15 Publication of ATE151760T1 publication Critical patent/ATE151760T1/de

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/04—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Pyrrole Compounds (AREA)

AT91111866T 1987-02-23 1988-02-16 Thiazolidin-derivate ATE151760T1 (de)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
JP3784487		1987-02-23

Publications (1)

Publication Number	Publication Date
ATE151760T1 true ATE151760T1 (de)	1997-05-15

Family

ID=12508841

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT91111866T ATE151760T1 (de)	1987-02-23	1988-02-16	Thiazolidin-derivate

Country Status (7)

Country	Link
US (1)	US4857537A (de)
EP (2)	EP0461677B1 (de)
KR (1)	KR960001205B1 (de)
AT (1)	ATE151760T1 (de)
DE (2)	DE3875361T2 (de)
ES (2)	ES2103287T3 (de)
GR (1)	GR3006406T3 (de)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPH01250370A (ja) *	1987-12-23	1989-10-05	Zeria Pharmaceut Co Ltd	新規アミノ酸イミド誘導体、製法ならびに用途
JP2515568B2 (ja) *	1987-12-25	1996-07-10	株式会社ヤクルト本社	新規なチアゾリジン誘導体
US5053414A (en) *	1988-04-08	1991-10-01	Ono Pharmaceutical Co., Ltd.	Heterocyclic compounds
US5212191A (en) *	1988-04-08	1993-05-18	Ono Pharmaceutical Co., Ltd.	Heterocyclic compounds
CA2004028C (en) *	1988-12-08	1998-09-22	Motoki Torizuka	Condensed benzene derivative
WO1990012005A1 (en) *	1989-04-13	1990-10-18	Japan Tobacco Inc.	New amino acid derivatives having prolylendopeptidase inhibitor activity
US5073549A (en) *	1990-03-22	1991-12-17	Bristol-Myers Squibb Company	BU-4164E - A and B, prolyl endopeptidase inhibitors and their methods of use
US4999349A (en) *	1990-03-22	1991-03-12	Bristol-Myers Squibb Co.	BU-4164E - A and B, prolyl endopeptidase inhibitors
JP2511605B2 (ja) *	1990-06-04	1996-07-03	ファイザー・インコーポレーテッド	芳香性ピロリジンおよびチアゾリヂンアミド類
US5506256A (en) *	1990-07-27	1996-04-09	Yoshitomi Pharmaceutical Industries, Ltd.	Proline derivatives possessing prolyl endopeptidase-inhibitory activity
IT1283782B1 (it) *	1996-08-09	1998-04-30	Ct Lab Farm Srl	Uso di ammidi dell'acido gamma-idrossibutirrico nel trattamento di tossicodipendenze,ed in particolare sell'alcolismo
US6419857B1 (en) *	1999-12-06	2002-07-16	Baker Hughes Incorporated	Thiazolidines and use thereof for corrosion inhibition
ATE462432T1 (de)	2003-05-05	2010-04-15	Probiodrug Ag	Glutaminylcyclase-hemmer
WO2005049027A2 (en)	2003-11-03	2005-06-02	Probiodrug Ag	Combinations useful for the treatment of neuronal disorders
WO2005075436A2 (en)	2004-02-05	2005-08-18	Probiodrug Ag	Novel inhibitors of glutaminyl cyclase
EP1760076A1 (de)	2005-09-02	2007-03-07	Ferring B.V.	FAP Inhibitoren
EP2089383B1 (de)	2006-11-09	2015-09-16	Probiodrug AG	3-hydroxy-1,5-dihydropyrrol-2-one derivate als inhibitoren von glutaminylcyclase zur behandlung von geschwüren, krebs und anderen krankheiten
JP5523107B2 (ja)	2006-11-30	2014-06-18	プロビオドルグエージー	グルタミニルシクラーゼの新規阻害剤
EP2117540A1 (de)	2007-03-01	2009-11-18	Probiodrug AG	Neue verwendung von glutaminyl-cyclase-hemmern
US9656991B2 (en)	2007-04-18	2017-05-23	Probiodrug Ag	Inhibitors of glutaminyl cyclase
AU2010294214B2 (en)	2009-09-11	2015-05-07	Vivoryon Therapeutics N.V.	Heterocylcic derivatives as inhibitors of glutaminyl cyclase
JP6026284B2 (ja)	2010-03-03	2016-11-16	プロビオドルグエージー	グルタミニルシクラーゼの阻害剤
KR101790806B1 (ko)	2010-03-10	2017-11-20	프로비오드룩 아게	글루타미닐 사이클라제(ｑｃ, ｅｃ 2.3.2.5)의 헤테로사이클릭 억제제
WO2011131748A2 (en)	2010-04-21	2011-10-27	Probiodrug Ag	Novel inhibitors
DK2686313T3 (en)	2011-03-16	2016-05-02	Probiodrug Ag	Benzimidazole derivatives as inhibitors of glutaminyl cyclase
DK3461819T3 (da)	2017-09-29	2020-08-10	Probiodrug Ag	Inhibitorer af glutaminylcyklase

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60188317A (ja) *	1984-03-09	1985-09-25	Yakult Honsha Co Ltd	抗健忘症剤
JPS6137764A (ja) *	1984-07-31	1986-02-22	Suntory Ltd	抗プロリルエンドペプチダ−ゼ活性を有する新規生理活性化合物
JPH0623190B2 (ja) *	1985-04-16	1994-03-30	サントリー株式会社	インヒビタ−活性を有するｎ−アシルピロリジン誘導体及びその製法並びに用途
DE3684633D1 (de) *	1985-04-16	1992-05-07	Suntory Ltd	Dipeptid-derivate von fettsaeure, verfahren zu ihrer herstellung, heilmittel, das sie enthaelt und anwendung.
US4873342A (en) *	1985-04-16	1989-10-10	Suntory Limited	Dipeptide derivative and synthesis and use thereof

1988
- 1988-02-16 DE DE8888102243T patent/DE3875361T2/de not_active Expired - Fee Related
- 1988-02-16 EP EP91111866A patent/EP0461677B1/de not_active Expired - Lifetime
- 1988-02-16 ES ES91111866T patent/ES2103287T3/es not_active Expired - Lifetime
- 1988-02-16 EP EP88102243A patent/EP0280956B1/de not_active Expired - Lifetime
- 1988-02-16 AT AT91111866T patent/ATE151760T1/de not_active IP Right Cessation
- 1988-02-16 DE DE3855875T patent/DE3855875T2/de not_active Expired - Fee Related
- 1988-02-16 ES ES88102243T patent/ES2052619T3/es not_active Expired - Lifetime
- 1988-02-23 KR KR1019880001849A patent/KR960001205B1/ko not_active IP Right Cessation
- 1988-02-23 US US07/159,073 patent/US4857537A/en not_active Expired - Lifetime
1992
- 1992-12-02 GR GR920402770T patent/GR3006406T3/el unknown

Also Published As

Publication number	Publication date
DE3875361T2 (de)	1993-03-25
US4857537A (en)	1989-08-15
ES2103287T3 (es)	1997-09-16
GR3006406T3 (de)	1993-06-21
KR960001205B1 (ko)	1996-01-24
DE3855875T2 (de)	1997-08-28
DE3855875D1 (de)	1997-05-22
KR880009949A (ko)	1988-10-06
ES2052619T3 (es)	1994-07-16
EP0461677B1 (de)	1997-04-16
DE3875361D1 (de)	1992-11-26
EP0280956B1 (de)	1992-10-21
EP0280956A1 (de)	1988-09-07
EP0461677A1 (de)	1991-12-18

Publication	Publication Date	Title
ATE151760T1 (de)	1997-05-15	Thiazolidin-derivate
DE3879522D1 (de)	1993-04-29	Prolinalderivate.
DK0624584T3 (da)	1999-05-25	Piperazinderivater, der er nyttige som calmodulininhibitorer
ATE84787T1 (de)	1993-02-15	Prolin-derivate.
DE68918681D1 (de)	1994-11-10	Glycosidasehemmer.
ES2070135T3 (es)	1995-06-01	Derivados de pirrolidina anti-amnesicos.
DK147588A (da)	1988-09-19	Benzoxazinderivat samt fremgangsmaade til fremstilling deraf
ATE137747T1 (de)	1996-05-15	Aminobenzolverbindungen, herstellung und verwendung
EG19396A (en)	1995-01-31	Pesticidal heterocyclic compounds
DK0658555T3 (da)	1997-12-22	Pyridazinonderivater, fremgangsmåder til fremstilling deraf samt anvendelse deraf
DE69734479D1 (de)	2005-12-01	Herstellung von Thiazolen
ATE143591T1 (de)	1996-10-15	Verwendung von bis-(p- hydroxyphenylthio)methanderivaten zur hemmung der fortschreitenden entwicklung von insulinabhängingem diabetes mellitus
ES445339A1 (es)	1977-06-01	Un procedimiento para la preparacion de derivados pirrolidi-nicos.
HUT39173A (en)	1986-08-28	Process for production of derivatives of 3-hydro-amino-2,3-dihydro-benzoxepin

Legal Events

Date	Code	Title	Description
1997-10-15	UEP	Publication of translation of european patent specification
2003-11-15	REN	Ceased due to non-payment of the annual fee