NO914775D0 - Fremgangsmaate for fremstilling av en 3-alkylert indol - Google Patents

Fremgangsmaate for fremstilling av en 3-alkylert indol

Info

Publication number: NO914775D0
Authority: NO; Norway
Prior art keywords: preparation; alkyled; indol; procedure; afford
Prior art date: 1990-12-05

Application number

NO914775A

Other languages

English (en)

Other versions

NO914775L (no

NO175680B (no

NO175680C (no

Inventor

Robert Toms Jacobs

Gerard Francis Costello

Stephen Alan Brook

Peter John Harrison

Original Assignee

Ici Plc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-12-05

Filing date

1991-12-04

Publication date

1991-12-04

1991-12-04 Application filed by Ici Plc filed Critical Ici Plc

1991-12-04 Publication of NO914775D0 publication Critical patent/NO914775D0/no

1992-06-09 Publication of NO914775L publication Critical patent/NO914775L/no

1994-08-08 Publication of NO175680B publication Critical patent/NO175680B/no

1994-11-16 Publication of NO175680C publication Critical patent/NO175680C/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C07D209/24—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals with an alkyl or cycloalkyl radical attached to the ring nitrogen atom
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C201/00—Preparation of esters of nitric or nitrous acid or of compounds containing nitro or nitroso groups bound to a carbon skeleton
- C07C201/06—Preparation of nitro compounds
- C07C201/12—Preparation of nitro compounds by reactions not involving the formation of nitro groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C227/00—Preparation of compounds containing amino and carboxyl groups bound to the same carbon skeleton
- C07C227/04—Formation of amino groups in compounds containing carboxyl groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
- C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Ophthalmology & Optometry (AREA)
Pulmonology (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Immunology (AREA)
Dermatology (AREA)
Indole Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)
Saccharide Compounds (AREA)
Physical Or Chemical Processes And Apparatus (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO914775A 1990-12-05 1991-12-04 Fremgangsmåte for fremstilling av en 3-alkylert indol NO175680C (no)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB909026427A GB9026427D0 (en)	1990-12-05	1990-12-05	Chemical process

Publications (4)

Publication Number	Publication Date
NO914775D0 true NO914775D0 (no)	1991-12-04
NO914775L NO914775L (no)	1992-06-09
NO175680B NO175680B (no)	1994-08-08
NO175680C NO175680C (no)	1994-11-16

Family

ID=10686509

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO914775A NO175680C (no)	1990-12-05	1991-12-04	Fremgangsmåte for fremstilling av en 3-alkylert indol

Country Status (22)

Country	Link
US (1)	US5280125A (no)
EP (1)	EP0489547B1 (no)
JP (1)	JP3160040B2 (no)
KR (1)	KR100228328B1 (no)
AT (1)	ATE168998T1 (no)
AU (1)	AU652002B2 (no)
CA (1)	CA2056065C (no)
CZ (1)	CZ282019B6 (no)
DE (1)	DE69129894T2 (no)
DK (1)	DK0489547T3 (no)
ES (1)	ES2118743T3 (no)
FI (1)	FI102170B1 (no)
GB (1)	GB9026427D0 (no)
HU (1)	HU222123B1 (no)
IE (1)	IE913936A1 (no)
IL (1)	IL100055A (no)
NO (1)	NO175680C (no)
NZ (1)	NZ240624A (no)
PT (1)	PT99683B (no)
RU (1)	RU2054417C1 (no)
SK (1)	SK278987B6 (no)
ZA (1)	ZA919079B (no)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9119001D0 (en) *	1991-09-05	1991-10-23	Ici Plc	Pharmaceutical agents
AU4400597A (en) *	1996-10-08	1998-05-05	Fujisawa Pharmaceutical Co., Ltd.	Indole derivatives
CN112457235B (zh) *	2020-12-02	2023-04-25	烟台凯博医药科技有限公司	一种7-甲基吲哚的制备方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3732245A (en) *	1970-11-04	1973-05-08	Hoffmann La Roche	Process and intermediates for the preparation of indoles from ortho-nitrotoluenes
US3976639A (en) *	1970-11-04	1976-08-24	Hoffmann-La Roche Inc.	Intermediates for indoles
US3979410A (en) *	1974-01-21	1976-09-07	Hoffmann-La Roche Inc.	Intermediate α-acyl-β-dialkylamino-2-nitrostyrenes
US4137404A (en) *	1977-12-20	1979-01-30	Hoffmann-La Roche Inc.	Synthesis of tryptophans
US4665087A (en) *	1982-02-22	1987-05-12	Ciba-Geigy Corporation	1-(carbamyl, thiocarbamyl, and iminocarbamyl)-indoline derivatives
GB8607294D0 (en) *	1985-04-17	1986-04-30	Ici America Inc	Heterocyclic amide derivatives
GB8623429D0 (en) *	1985-10-17	1986-11-05	Ici America Inc	Carboximide derivatives
US5180728A (en) *	1989-09-25	1993-01-19	Fujisawa Pharmaceutical Company, Ltd.	Pyrimidoindole derivatives and processes for preparation thereof
GB8927981D0 (en) *	1989-12-11	1990-02-14	Ici Plc	Carbamoyl derivative
GB9026425D0 (en) *	1990-12-05	1991-01-23	Ici Plc	Process

1990
- 1990-12-05 GB GB909026427A patent/GB9026427D0/en active Pending
1991
- 1991-11-12 IE IE393691A patent/IE913936A1/en not_active IP Right Cessation
- 1991-11-14 IL IL10005591A patent/IL100055A/en active IP Right Grant
- 1991-11-15 ZA ZA919079A patent/ZA919079B/xx unknown
- 1991-11-18 NZ NZ240624A patent/NZ240624A/en not_active IP Right Cessation
- 1991-11-19 AU AU87946/91A patent/AU652002B2/en not_active Ceased
- 1991-11-22 CA CA002056065A patent/CA2056065C/en not_active Expired - Fee Related
- 1991-11-29 ES ES91311072T patent/ES2118743T3/es not_active Expired - Lifetime
- 1991-11-29 AT AT91311072T patent/ATE168998T1/de not_active IP Right Cessation
- 1991-11-29 DK DK91311072T patent/DK0489547T3/da active
- 1991-11-29 SK SK3633-91A patent/SK278987B6/sk unknown
- 1991-11-29 EP EP91311072A patent/EP0489547B1/en not_active Expired - Lifetime
- 1991-11-29 DE DE69129894T patent/DE69129894T2/de not_active Expired - Fee Related
- 1991-11-29 CZ CS913633A patent/CZ282019B6/cs not_active IP Right Cessation
- 1991-12-02 HU HU9103759A patent/HU222123B1/hu not_active IP Right Cessation
- 1991-12-04 US US07/803,315 patent/US5280125A/en not_active Expired - Fee Related
- 1991-12-04 PT PT99683A patent/PT99683B/pt not_active IP Right Cessation
- 1991-12-04 NO NO914775A patent/NO175680C/no unknown
- 1991-12-04 KR KR1019910022262A patent/KR100228328B1/ko not_active IP Right Cessation
- 1991-12-04 RU SU915010306A patent/RU2054417C1/ru not_active IP Right Cessation
- 1991-12-05 FI FI915735A patent/FI102170B1/fi not_active IP Right Cessation
- 1991-12-05 JP JP32180091A patent/JP3160040B2/ja not_active Expired - Fee Related

Also Published As

Publication number	Publication date
NO914775L (no)	1992-06-09
ZA919079B (en)	1992-09-30
JPH04266870A (ja)	1992-09-22
DK0489547T3 (da)	1999-04-26
EP0489547A1 (en)	1992-06-10
CS363391A3 (en)	1992-06-17
AU652002B2 (en)	1994-08-11
US5280125A (en)	1994-01-18
HU222123B1 (hu)	2003-04-28
FI102170B (fi)	1998-10-30
PT99683B (pt)	1999-05-31
JP3160040B2 (ja)	2001-04-23
FI915735A0 (fi)	1991-12-05
KR100228328B1 (ko)	1999-11-01
CZ282019B6 (cs)	1997-04-16
RU2054417C1 (ru)	1996-02-20
HU913759D0 (en)	1992-02-28
IE913936A1 (en)	1992-06-17
PT99683A (pt)	1992-10-30
NO175680B (no)	1994-08-08
AU8794691A (en)	1992-06-11
DE69129894D1 (de)	1998-09-03
NZ240624A (en)	1994-01-26
GB9026427D0 (en)	1991-01-23
KR920012029A (ko)	1992-07-25
HUT60716A (en)	1992-10-28
FI915735A (fi)	1992-06-06
IL100055A0 (en)	1992-08-18
ES2118743T3 (es)	1998-10-01
SK278987B6 (sk)	1998-05-06
EP0489547B1 (en)	1998-07-29
FI102170B1 (fi)	1998-10-30
NO175680C (no)	1994-11-16
DE69129894T2 (de)	1998-12-10
ATE168998T1 (de)	1998-08-15
CA2056065A1 (en)	1992-06-06
IL100055A (en)	1996-12-05
CA2056065C (en)	2003-07-29

Publication	Publication Date	Title
ES2101063T3 (es)	1997-07-01	Derivados monofluorados de n-propargil-1-amino-indano y su utilizacion como inhibidores de la monoamin-oxidasa.
MY131298A (en)	2007-08-30	5-heteroyl indole derivatives
LV10575A (lv)	1995-04-20	Izoksazoi-4-karbonskabes amids un hidroksialkiliden-cianetikskabes amids sos savienojumus saturosi astniecibas lidzekli un to pielietojums
NL300181I1 (nl)	2005-05-02	N-(pyrroloÄ2,3-dÜpyrimidine-3-ylacyl)-glutaminezuurderivaten.
ATE90093T1 (de)	1993-06-15	1,3,4,5-tetrahydrobenz(c,d>indole.
DE3682541D1 (de)	1992-01-02	Herbizid wirkende derivate des n-phenyl-3,4,5,6-tetrahydrophthalsaeureimides.
NO914775L (no)	1992-06-09	Fremgangsmaate for fremstilling av en 3-alkylert indol
NO860733L (no)	1986-08-29	N-(2-klor-4-trifluormethylfenyl)-3-trifluormethyl-benzensulfonamidderivat, fremgangsmaate for fremstilling av dette, og fungicid middel inneholdende dette.
DK218083D0 (da)	1983-05-16	Aminoalkadien-derivater, deres fremstilling og anvendelse
DK0462837T3 (da)	2000-09-11	Fremstilling af indol-derivater
EE03873B1 (et)	2002-10-15	Meetod alküüloksüfuranooni amiinderivaatide valmistamiseks, sel meetodil saadud ühendid ja nende kasutamine
DK34888A (da)	1988-07-28	Fremgangsmaade til fremstilling af n,n-(dibenzohexatrienylen)urinstoffer
NO175899C (no)	1994-12-28	Analogifremgangsmåte for fremstilling av terapeutisk aktive heksahydropyrrolo(2,3-b)indol karbamater-, urea-, -amider og beslektede forbindelser
ATE112272T1 (de)	1994-10-15	Herstellung von n-(3-(((aryl)amino)sulfonyl)-1h- 1,2,4-triazol-5-yl)aminen.
NO165395C (no)	1991-02-06	Fremgangsmaate for fremstilling av n-(sulfonylmetyl)formamider.
NO852418L (no)	1985-12-16	Fremgangsmaate for fremstilling av aminderivater.
NO874136D0 (no)	1987-10-01	Fremgangsmaate for fremstilling av n-(omega-cyanoalkyl)aminofenoler.
ES517874A0 (es)	1983-12-01	Procedimiento de preparacion de derivados de diaza-3,7a-cicloherta-(j,k)-fluorenos.
NO20012538L (no)	2001-07-04	Anvendelse av N-substituerte azabicycloalkanderivater for behandling av forstyrrelser i sentralnervesystemet
AU2175288A (en)	1989-03-02	Production of N-(4-chloro-2-fluoro-5-(n-pentyloxycarbonyl methyloxy) phenyl' 3,4,5,6-tetrahydrophthalimide compounds via aniline derivatives
DK0686641T3 (da)	1998-11-23	2'-Deoxy-5-fluoruridinderivat, farmaceutisk acceptabelt salt deraf, fremgangsmåde til fremstilling deraf, og antitumorlægem
ES8406061A1 (es)	1984-07-01	Un procedimiento para la preparacion de un derivado de naftalenamina.
IT8125591A0 (it)	1981-12-15	Procedimento di purificazione di n-alchil nitro aniline da n-nitroso ammine.
SU1297421A1 (ru)	2016-09-10	ГИДРОХЛОРИДЫ 3-ЗАМЕЩЕННЫХ 2-ЭТИЛ-4-МЕТИЛПИРАЗОЛО(1,5-а)-БЕНЗИМИДАЗОЛА, ОБЛАДАЮЩИЕ АНТИАРИТМИЧЕСКОЙ АКТИВНОСТЬЮ
ATE64377T1 (de)	1991-06-15	Substituierte aminderivate, ihre herstellung und verwendung.