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NO893240L - USE OF ALFA-AMINOBORIC ACID DERIVATIVES FOR PROPHYLACTIC AND TREATMENT OF VIRUSAL DISEASES. - Google Patents

USE OF ALFA-AMINOBORIC ACID DERIVATIVES FOR PROPHYLACTIC AND TREATMENT OF VIRUSAL DISEASES.

Info

Publication number
NO893240L
NO893240L NO89893240A NO893240A NO893240L NO 893240 L NO893240 L NO 893240L NO 89893240 A NO89893240 A NO 89893240A NO 893240 A NO893240 A NO 893240A NO 893240 L NO893240 L NO 893240L
Authority
NO
Norway
Prior art keywords
virusal
alfa
prophylactic
diseases
treatment
Prior art date
Application number
NO89893240A
Other languages
Norwegian (no)
Other versions
NO893240D0 (en
Inventor
Karin Moelling
Heinz-Werner Kleemann
Hansjoerg Urbach
Wolfgang Koenig
Dieter Ruppert
Irvin Winkler
Arnold Paessens
Original Assignee
Hoechst Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoechst Ag filed Critical Hoechst Ag
Publication of NO893240D0 publication Critical patent/NO893240D0/en
Publication of NO893240L publication Critical patent/NO893240L/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • A61K38/16Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/55Protease inhibitors
    • A61K38/553Renin inhibitors
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/69Boron compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Oncology (AREA)
  • Immunology (AREA)
  • Communicable Diseases (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Virology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
NO89893240A 1988-08-12 1989-08-11 USE OF ALFA-AMINOBORIC ACID DERIVATIVES FOR PROPHYLACTIC AND TREATMENT OF VIRUSAL DISEASES. NO893240L (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE3827340A DE3827340A1 (en) 1988-08-12 1988-08-12 USE OF (ALPHA) -AMINOBORONIC ACID DERIVATIVES FOR THE PROPHYLAXIS AND TREATMENT OF VIRUS DISEASES

Publications (2)

Publication Number Publication Date
NO893240D0 NO893240D0 (en) 1989-08-11
NO893240L true NO893240L (en) 1990-03-27

Family

ID=6360676

Family Applications (1)

Application Number Title Priority Date Filing Date
NO89893240A NO893240L (en) 1988-08-12 1989-08-11 USE OF ALFA-AMINOBORIC ACID DERIVATIVES FOR PROPHYLACTIC AND TREATMENT OF VIRUSAL DISEASES.

Country Status (10)

Country Link
EP (1) EP0354522A1 (en)
JP (1) JPH0291023A (en)
KR (1) KR900002766A (en)
AU (1) AU3951389A (en)
DE (1) DE3827340A1 (en)
DK (1) DK395789A (en)
IL (1) IL91276A0 (en)
NO (1) NO893240L (en)
PT (1) PT91426A (en)
ZA (1) ZA896150B (en)

Families Citing this family (26)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5142056A (en) * 1989-05-23 1992-08-25 Abbott Laboratories Retroviral protease inhibiting compounds
EP0315574A3 (en) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin inhibitors
US4983589A (en) * 1989-12-14 1991-01-08 Chevron Research And Technology Company Fungicidal imidazole diphenylaliphaticboranes and derivatives thereof
GB9017694D0 (en) * 1990-08-13 1990-09-26 Sandoz Ltd Improvements in or relating to organic chemistry
GB9024775D0 (en) * 1990-11-14 1991-01-02 Axis Research Chemical compounds
US5554728A (en) * 1991-07-23 1996-09-10 Nexstar Pharmaceuticals, Inc. Lipid conjugates of therapeutic peptides and protease inhibitors
DE4126485A1 (en) * 1991-08-10 1993-02-11 Bayer Ag TRIFLUOROMETHYL-CONTAINING PSEUDOPEPTIDE
US5693617A (en) * 1994-03-15 1997-12-02 Proscript, Inc. Inhibitors of the 26s proteolytic complex and the 20s proteasome contained therein
US6083903A (en) 1994-10-28 2000-07-04 Leukosite, Inc. Boronic ester and acid compounds, synthesis and uses
DE4441483C1 (en) * 1994-11-22 1996-04-04 Gsf Forschungszentrum Umwelt Use of bio-assimilated boron cpds.
US7576206B2 (en) 2003-08-14 2009-08-18 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7223745B2 (en) 2003-08-14 2007-05-29 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7468383B2 (en) 2005-02-11 2008-12-23 Cephalon, Inc. Proteasome inhibitors and methods of using the same
US7442830B1 (en) 2007-08-06 2008-10-28 Millenium Pharmaceuticals, Inc. Proteasome inhibitors
US7838673B2 (en) 2007-10-16 2010-11-23 Millennium Pharmaceuticals, Inc. Proteasome inhibitors
CN107266480A (en) 2008-06-17 2017-10-20 米伦纽姆医药公司 Boric acid ester compound and its medical composition
AR075090A1 (en) 2008-09-29 2011-03-09 Millennium Pharm Inc ACID DERIVATIVES 1-AMINO-2-CYCLLOBUTILETILBORONICO PROTEOSOMA INHIBITORS, USEFUL AS ANTI-BANKER AGENTS, AND PHARMACEUTICAL COMPOSITIONS THAT UNDERSTAND THEM.
CN102725300B (en) 2009-12-22 2015-03-11 赛福伦公司 Proteasome inhibitors and processes for their preparation, purification and use
BR112012022060A2 (en) * 2010-03-01 2018-05-08 Onyx Therapeutics Inc compound for inhibition of immunoproteasome
KR20130036228A (en) 2010-03-31 2013-04-11 밀레니엄 파머슈티컬스 인코퍼레이티드 Derivatives of 1-amino-2-cyclopropylethylboronic acid
CN103483363B (en) * 2012-06-13 2016-12-21 上海赛迦化工产品有限公司 Multifarious chiral aminoboronic acid and its preparation method and application
CN103396426B (en) * 2013-07-12 2016-09-28 上海工程技术大学 Chirality boronic acid derivatives and its preparation method and application
CN103408572B (en) * 2013-07-12 2015-12-02 上海工程技术大学 Chiral aminoboronic acid derivative and its preparation method and application
KR102481856B1 (en) 2014-05-20 2022-12-26 밀레니엄 파머슈티컬스 인코퍼레이티드 Boron-containing proteasome inhibitors for use after primary cancer therapy
US10526315B2 (en) 2016-06-21 2020-01-07 Orion Ophthalmology LLC Carbocyclic prolinamide derivatives
HUE064412T2 (en) 2016-06-21 2024-03-28 Orion Ophthalmology LLC Heterocyclic prolinamide derivatives

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4499082A (en) * 1983-12-05 1985-02-12 E. I. Du Pont De Nemours And Company α-Aminoboronic acid peptides
US4537773A (en) * 1983-12-05 1985-08-27 E. I. Du Pont De Nemours And Company α-Aminoboronic acid derivatives
US5187157A (en) * 1987-06-05 1993-02-16 Du Pont Merck Pharmaceutical Company Peptide boronic acid inhibitors of trypsin-like proteases
EP0315574A3 (en) * 1987-11-05 1990-08-22 Hoechst Aktiengesellschaft Renin inhibitors

Also Published As

Publication number Publication date
KR900002766A (en) 1990-03-31
DE3827340A1 (en) 1990-02-15
IL91276A0 (en) 1990-03-19
DK395789A (en) 1990-02-13
EP0354522A1 (en) 1990-02-14
DK395789D0 (en) 1989-08-11
JPH0291023A (en) 1990-03-30
PT91426A (en) 1990-03-08
ZA896150B (en) 1991-01-30
NO893240D0 (en) 1989-08-11
AU3951389A (en) 1990-03-29

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