NO20032667D0 - Cykliseringsfremgangsmåtetrinn for fremstilling av kinoloner og naftyridiner - Google Patents
Cykliseringsfremgangsmåtetrinn for fremstilling av kinoloner og naftyridinerInfo
- Publication number
- NO20032667D0 NO20032667D0 NO20032667A NO20032667A NO20032667D0 NO 20032667 D0 NO20032667 D0 NO 20032667D0 NO 20032667 A NO20032667 A NO 20032667A NO 20032667 A NO20032667 A NO 20032667A NO 20032667 D0 NO20032667 D0 NO 20032667D0
- Authority
- NO
- Norway
- Prior art keywords
- naphthyridines
- quinolones
- preparation
- process steps
- cyclization process
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
- C07D491/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
- C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
- C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D513/04—Ortho-condensed systems
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Virology (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Molecular Biology (AREA)
- AIDS & HIV (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Quinoline Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US25563300P | 2000-12-14 | 2000-12-14 | |
PCT/US2001/048536 WO2002048113A1 (en) | 2000-12-14 | 2001-12-07 | Cyclization process step in the making of quinolones and naphthyridines |
Publications (3)
Publication Number | Publication Date |
---|---|
NO20032667D0 true NO20032667D0 (no) | 2003-06-12 |
NO20032667L NO20032667L (no) | 2003-08-14 |
NO325236B1 NO325236B1 (no) | 2008-03-03 |
Family
ID=22969207
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
NO20032667A NO325236B1 (no) | 2000-12-14 | 2003-06-12 | Cykliseringsfremgangsmatetrinn for fremstilling av kinoloner og naftyridiner |
Country Status (19)
Country | Link |
---|---|
EP (1) | EP1343766B1 (no) |
JP (2) | JP4417007B2 (no) |
KR (1) | KR100603163B1 (no) |
CN (1) | CN1232508C (no) |
AT (1) | ATE300522T1 (no) |
AU (2) | AU2002229057B2 (no) |
BR (1) | BR0116229A (no) |
CA (1) | CA2427831C (no) |
CZ (1) | CZ20031379A3 (no) |
DE (1) | DE60112325T2 (no) |
DK (1) | DK1343766T3 (no) |
ES (1) | ES2247190T3 (no) |
HU (1) | HUP0303991A3 (no) |
IL (2) | IL155677A0 (no) |
MX (1) | MXPA03005338A (no) |
NO (1) | NO325236B1 (no) |
NZ (1) | NZ525569A (no) |
PL (1) | PL207394B1 (no) |
WO (1) | WO2002048113A1 (no) |
Families Citing this family (11)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6803469B2 (en) * | 2002-08-05 | 2004-10-12 | The Procter & Gamble Company | Process for preparing quinolone antibiotic intermediates |
KR100735587B1 (ko) * | 2002-08-05 | 2007-07-04 | 더 프록터 앤드 갬블 캄파니 | 퀴놀론계 항생제 중간체의 제조 방법 |
ATE443048T1 (de) * | 2002-11-20 | 2009-10-15 | Japan Tobacco Inc | 4-oxochinolinverbindungen und deren verwendung als hiv-integrase-inhibitoren |
US7402674B2 (en) | 2004-01-31 | 2008-07-22 | Sanofi-Aventis Deutschland Gmbh, | 7-Phenylamino-4-quinolone-3-carboxylic acid derivatives, process for their preparation and their use as medicaments |
RS54047B1 (en) | 2006-03-06 | 2015-10-30 | Japan Tobacco Inc. | PROCEDURE FOR OBTAINING 4-OXOCHINOLINE COMPOUNDS |
CN101437801B (zh) | 2006-03-06 | 2013-02-06 | 日本烟草产业株式会社 | 制备4-氧代喹啉化合物的方法 |
NZ575542A (en) * | 2006-09-12 | 2012-03-30 | Gilead Sciences Inc | Process and intermediates for preparing 4-oxoquinolone integrase inhibitors |
US8658183B2 (en) | 2007-08-09 | 2014-02-25 | Taigen Biotechnology Company, Ltd. | Antimicrobial parenteral formulation |
AR068403A1 (es) * | 2007-09-11 | 2009-11-18 | Gilead Sciences Inc | Proceso e intermediarios para la preparacion de inhibidores de integrasa |
NZ588898A (en) | 2008-07-01 | 2012-09-28 | Taigen Biotechnology Co Ltd | Use of nemonoxacin for treating antibiotic-resistant staphylococcus aureus infection |
AU2013296289B2 (en) | 2012-08-03 | 2017-10-05 | Gilead Sciences, Inc. | Process and intermediates for preparing integrase inhibitors |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CA2196539C (en) * | 1994-08-02 | 2001-05-15 | The Procter & Gamble Company | Process for making quinolonyl lactam antimicrobials and novel intermediate compounds |
CA2196538C (en) * | 1994-08-02 | 2000-04-25 | Jared Lynn Randall | Process for making antimicrobial compounds |
-
2001
- 2001-12-07 PL PL363355A patent/PL207394B1/pl not_active IP Right Cessation
- 2001-12-07 JP JP2002549644A patent/JP4417007B2/ja not_active Expired - Fee Related
- 2001-12-07 AT AT01990192T patent/ATE300522T1/de active
- 2001-12-07 HU HU0303991A patent/HUP0303991A3/hu unknown
- 2001-12-07 ES ES01990192T patent/ES2247190T3/es not_active Expired - Lifetime
- 2001-12-07 AU AU2002229057A patent/AU2002229057B2/en not_active Ceased
- 2001-12-07 BR BR0116229-2A patent/BR0116229A/pt not_active IP Right Cessation
- 2001-12-07 WO PCT/US2001/048536 patent/WO2002048113A1/en active IP Right Grant
- 2001-12-07 DK DK01990192T patent/DK1343766T3/da active
- 2001-12-07 AU AU2905702A patent/AU2905702A/xx active Pending
- 2001-12-07 EP EP01990192A patent/EP1343766B1/en not_active Expired - Lifetime
- 2001-12-07 CZ CZ20031379A patent/CZ20031379A3/cs unknown
- 2001-12-07 IL IL15567701A patent/IL155677A0/xx active IP Right Grant
- 2001-12-07 DE DE60112325T patent/DE60112325T2/de not_active Expired - Lifetime
- 2001-12-07 CA CA002427831A patent/CA2427831C/en not_active Expired - Fee Related
- 2001-12-07 MX MXPA03005338A patent/MXPA03005338A/es active IP Right Grant
- 2001-12-07 KR KR1020037007905A patent/KR100603163B1/ko not_active IP Right Cessation
- 2001-12-07 CN CNB018207146A patent/CN1232508C/zh not_active Expired - Lifetime
- 2001-12-07 NZ NZ525569A patent/NZ525569A/en not_active IP Right Cessation
-
2003
- 2003-04-30 IL IL155677A patent/IL155677A/en not_active IP Right Cessation
- 2003-06-12 NO NO20032667A patent/NO325236B1/no not_active IP Right Cessation
-
2009
- 2009-10-05 JP JP2009231801A patent/JP2010001315A/ja not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP1343766B1 (en) | 2005-07-27 |
DK1343766T3 (da) | 2005-10-31 |
NZ525569A (en) | 2004-09-24 |
MXPA03005338A (es) | 2003-10-06 |
HUP0303991A2 (hu) | 2004-04-28 |
WO2002048113A1 (en) | 2002-06-20 |
EP1343766A1 (en) | 2003-09-17 |
NO20032667L (no) | 2003-08-14 |
CA2427831C (en) | 2009-08-18 |
CA2427831A1 (en) | 2002-06-20 |
CN1481365A (zh) | 2004-03-10 |
AU2905702A (en) | 2002-06-24 |
HUP0303991A3 (en) | 2012-09-28 |
ES2247190T3 (es) | 2006-03-01 |
KR20030063420A (ko) | 2003-07-28 |
CZ20031379A3 (cs) | 2003-11-12 |
AU2002229057B2 (en) | 2005-04-21 |
CN1232508C (zh) | 2005-12-21 |
IL155677A (en) | 2009-02-11 |
PL207394B1 (pl) | 2010-12-31 |
DE60112325D1 (de) | 2005-09-01 |
KR100603163B1 (ko) | 2006-07-24 |
NO325236B1 (no) | 2008-03-03 |
JP2004515542A (ja) | 2004-05-27 |
BR0116229A (pt) | 2003-11-04 |
PL363355A1 (en) | 2004-11-15 |
JP4417007B2 (ja) | 2010-02-17 |
DE60112325T2 (de) | 2006-05-24 |
IL155677A0 (en) | 2003-11-23 |
ATE300522T1 (de) | 2005-08-15 |
JP2010001315A (ja) | 2010-01-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MM1K | Lapsed by not paying the annual fees |