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NO20013150D0 - Fremgangsmåte ved fremstilling av 5-cyanftalid - Google Patents

Fremgangsmåte ved fremstilling av 5-cyanftalid

Info

Publication number
NO20013150D0
NO20013150D0 NO20013150A NO20013150A NO20013150D0 NO 20013150 D0 NO20013150 D0 NO 20013150D0 NO 20013150 A NO20013150 A NO 20013150A NO 20013150 A NO20013150 A NO 20013150A NO 20013150 D0 NO20013150 D0 NO 20013150D0
Authority
NO
Norway
Prior art keywords
cyanophthalide
preparation
Prior art date
Application number
NO20013150A
Other languages
English (en)
Other versions
NO20013150L (no
NO326516B1 (no
Inventor
Hans Petersen
Poul Dahlberg Nielsen
Original Assignee
Lundbeck & Co As H
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lundbeck & Co As H filed Critical Lundbeck & Co As H
Publication of NO20013150D0 publication Critical patent/NO20013150D0/no
Publication of NO20013150L publication Critical patent/NO20013150L/no
Publication of NO326516B1 publication Critical patent/NO326516B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D307/00Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/77Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom ortho- or peri-condensed with carbocyclic rings or ring systems
    • C07D307/87Benzo [c] furans; Hydrogenated benzo [c] furans
    • C07D307/88Benzo [c] furans; Hydrogenated benzo [c] furans with one oxygen atom directly attached in position 1 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Furan Compounds (AREA)
NO20013150A 1998-12-23 2001-06-22 Fremgangsmate ved fremstilling av 5-cyanftalid NO326516B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DKPA199801718 1998-12-23
PCT/DK1999/000728 WO2000039112A1 (en) 1998-12-23 1999-12-22 Method for the preparation of 5-cyanophthalide

Publications (3)

Publication Number Publication Date
NO20013150D0 true NO20013150D0 (no) 2001-06-22
NO20013150L NO20013150L (no) 2001-08-20
NO326516B1 NO326516B1 (no) 2008-12-22

Family

ID=8107494

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20013150A NO326516B1 (no) 1998-12-23 2001-06-22 Fremgangsmate ved fremstilling av 5-cyanftalid

Country Status (31)

Country Link
US (1) US6392060B2 (no)
EP (1) EP1140886B1 (no)
JP (1) JP2002533450A (no)
KR (1) KR100454008B1 (no)
CN (1) CN1149208C (no)
AR (1) AR019791A1 (no)
AT (1) ATE236145T1 (no)
AU (1) AU764161B2 (no)
BG (1) BG64986B1 (no)
BR (1) BR9916955A (no)
CA (1) CA2356188C (no)
CZ (1) CZ300408B6 (no)
DE (1) DE69906580T2 (no)
DK (1) DK1140886T3 (no)
EA (1) EA003057B1 (no)
ES (1) ES2195644T3 (no)
HK (1) HK1043130B (no)
HU (1) HUP0104856A3 (no)
IL (1) IL143422A0 (no)
IS (1) IS2261B (no)
IT (1) IT1315269B1 (no)
NO (1) NO326516B1 (no)
NZ (1) NZ512073A (no)
PL (1) PL203275B1 (no)
PT (1) PT1140886E (no)
SI (1) SI1140886T1 (no)
SK (1) SK285530B6 (no)
TR (1) TR200101796T2 (no)
UA (1) UA70979C2 (no)
WO (1) WO2000039112A1 (no)
ZA (1) ZA200104262B (no)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO2000023431A1 (en) 1998-10-20 2000-04-27 H. Lundbeck A/S Method for the preparation of citalopram
NZ512073A (en) 1998-12-23 2003-10-31 H Method for the preparation of 5-cyanophthalide and citalopram
AR022329A1 (es) * 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
NZ514671A (en) 1999-04-14 2003-10-31 H Method for the preparation of citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991581A1 (it) * 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
GB2360281B (en) 1999-10-25 2002-01-16 Lundbeck & Co As H Method for the preparation of citalopram
SK287140B6 (sk) 1999-10-25 2010-01-07 H. Lundbeck A/S Spôsob prípravy citalopramu a medziprodukt na jeho výrobu
AR026063A1 (es) 1999-11-01 2002-12-26 Lundbeck & Co As H Metodo para la preparacion de 5-carboxiftalida.
CA2395404A1 (en) 1999-12-28 2001-07-05 H. Lundbeck A/S Method for the preparation of citalopram
SK11052002A3 (sk) 1999-12-30 2003-01-09 H. Lundbeck A/S Spôsob prípravy medziproduktu pri príprave citalopramu
SK286879B6 (sk) 2000-01-14 2009-07-06 H. Lundbeck A/S Spôsob prípravy 5-kyanoftalidu
FR2805812A1 (fr) 2000-02-24 2001-09-07 Lundbeck & Co As H Procede de preparation du citalopram
IES20010157A2 (en) 2000-03-03 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
TR200202195T2 (tr) 2000-03-13 2002-12-23 H. Lundbeck A/S 5-Yer değiştirmiş 1-(4-florofenil)-1,3- dihidroizobenzofuran'ın adım adım alkillenmesi
CA2402388A1 (en) 2000-03-13 2001-09-20 Hans Petersen Method for the preparation of citalopram
IES20010206A2 (en) 2000-03-13 2002-03-06 Lundbeck & Co As H Method for the preparation of citalopram
SK14512002A3 (sk) 2000-03-14 2003-03-04 H. Lundbeck A/S Spôsob výroby citalopramu, medziprodukt a citalopram výrobený týmto spôsobom
CZ20023406A3 (cs) * 2000-03-16 2003-01-15 H. Lundbeck A/S Způsob výroby 5-kyano-1-(4-fluorfenyl)-1,3-dihydroisobenzofuranu
AR032455A1 (es) 2000-05-12 2003-11-12 Lundbeck & Co As H Metodo para la preparacion de citalopram, un intermediario empleado en el metodo, un metodo para la preparacion del intermediario empleado en el metodo y composicion farmaceutica antidepresiva
IL144816A (en) 2000-08-18 2005-09-25 Lundbeck & Co As H Method for the preparation of citalopram
JP3798982B2 (ja) 2000-12-22 2006-07-19 ハー・ルンドベック・アクチエゼルスカベット 純粋なシタロプラムの製造方法
ES2181663T3 (es) 2000-12-28 2003-03-01 Lundbeck & Co As H Procedimiento para la preparacion de citalopram puro.
EP1321464A1 (en) * 2001-12-21 2003-06-25 ICROM S.p.A. Process for the preparation of 5-cyanophthalide and intermediates useful therein
WO2004083197A2 (en) * 2003-03-21 2004-09-30 H. Lundbeck A/S Intermediates for the preparation of citalopram and escitalopram
TR200504022T1 (tr) * 2003-03-24 2006-08-21 Hetero Drugs Limited (S)-sitalopram oksalatın yeni sıvı kristal formları.
EP1777221A1 (en) 2005-10-14 2007-04-25 Adorkem Technology SpA Process for the preparation of 5-cyanophthalide starting from 5-carboxyphthalide

Family Cites Families (19)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1143702A (no) 1965-03-18
GB1526331A (en) 1976-01-14 1978-09-27 Kefalas As Phthalanes
GB8419963D0 (en) 1984-08-06 1984-09-12 Lundbeck & Co As H Intermediate compound and method
GB8814057D0 (en) 1988-06-14 1988-07-20 Lundbeck & Co As H New enantiomers & their isolation
DK213290D0 (da) 1990-09-06 1990-09-06 Lundbeck & Co As H Treatment of cerebrovascular disorders
DE19626659A1 (de) 1996-07-03 1998-01-08 Basf Ag Verfahren zur Herstellung von Phthaliden
DE19627697A1 (de) 1996-07-10 1998-01-15 Basf Ag Verfahren zur Herstellung von Phthaliden
ZA9711376B (en) 1996-12-20 1998-07-21 Lundbeck & Co As H Indole or dihydroindole derivatives
DE69801764T2 (de) 1997-07-08 2002-07-04 H. Lundbeck A/S, Kobenhavn-Valby Verfahren zur herstellung von citalopram
UA62985C2 (en) 1997-11-10 2004-01-15 Lunnbeck As H A method for the preparation of citalopram
SK283907B6 (sk) 1997-11-11 2004-04-06 H. Lundbeck A/S Spôsob výroby citalopramu a medziprodukty
WO2000023431A1 (en) 1998-10-20 2000-04-27 H. Lundbeck A/S Method for the preparation of citalopram
NZ512073A (en) 1998-12-23 2003-10-31 H Method for the preparation of 5-cyanophthalide and citalopram
AR022329A1 (es) 1999-01-29 2002-09-04 Lundbeck & Co As H Metodo para la preparacion de 5-cianoftalida
NZ514671A (en) 1999-04-14 2003-10-31 H Method for the preparation of citalopram
ITMI991581A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
ITMI991579A1 (it) 1999-06-25 2001-01-15 Lundbeck & Co As H Metodo per la preparazione di citalopram
GB2360281B (en) 1999-10-25 2002-01-16 Lundbeck & Co As H Method for the preparation of citalopram
US6310222B1 (en) 1999-11-01 2001-10-30 Sumika Fine Chemicals Co., Ltd. Production method of 5-phthalancarbonitrile compound, intermediate therefor and production method of the intermediate

Also Published As

Publication number Publication date
JP2002533450A (ja) 2002-10-08
CZ20012335A3 (cs) 2001-12-12
EP1140886A1 (en) 2001-10-10
CA2356188C (en) 2006-05-23
IL143422A0 (en) 2002-04-21
HUP0104856A3 (en) 2003-01-28
DK1140886T3 (da) 2003-07-28
UA70979C2 (uk) 2004-11-15
SK285530B6 (sk) 2007-03-01
WO2000039112A1 (en) 2000-07-06
ITMI992696A1 (it) 2001-06-23
ZA200104262B (en) 2001-12-11
TR200101796T2 (tr) 2001-11-21
CZ300408B6 (cs) 2009-05-13
AR019791A1 (es) 2002-03-13
NZ512073A (en) 2003-10-31
SK8962001A3 (en) 2003-03-04
AU764161B2 (en) 2003-08-14
IS5952A (is) 2001-05-22
KR20010082370A (ko) 2001-08-29
US20020019546A1 (en) 2002-02-14
PL348608A1 (en) 2002-06-03
HK1043130A1 (en) 2002-09-06
NO20013150L (no) 2001-08-20
HK1043130B (zh) 2005-03-04
IS2261B (is) 2007-06-15
ES2195644T3 (es) 2003-12-01
PL203275B1 (pl) 2009-09-30
EP1140886B1 (en) 2003-04-02
CN1149208C (zh) 2004-05-12
NO326516B1 (no) 2008-12-22
AU1774200A (en) 2000-07-31
CN1331686A (zh) 2002-01-16
IT1315269B1 (it) 2003-02-03
BR9916955A (pt) 2001-09-11
HUP0104856A2 (hu) 2002-04-29
DE69906580D1 (de) 2003-05-08
BG64986B1 (bg) 2006-11-30
EA003057B1 (ru) 2002-12-26
ITMI992696A0 (it) 1999-12-23
PT1140886E (pt) 2003-08-29
US6392060B2 (en) 2002-05-21
CA2356188A1 (en) 2000-07-06
SI1140886T1 (en) 2003-08-31
BG105655A (en) 2002-01-31
KR100454008B1 (ko) 2004-10-20
EA200100696A1 (ru) 2001-12-24
DE69906580T2 (de) 2004-02-12
ATE236145T1 (de) 2003-04-15

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Representative=s name: PLOUGMANN & VINGTOFT, POSTBOKS 1003 SENTRUM, 0104

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