NO157738C - ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES. - Google Patents

ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES.

Info

Publication number: NO157738C
Authority: NO; Norway
Prior art keywords: benzocsazolinones; benzocsazinones; preparation; therapeutically active; analogue procedure
Prior art date: 1981-09-01

Application number

NO822932A

Other languages

Norwegian (no)

Other versions

NO157738B (en

NO822932L (en

Inventor

Kurt Schromm

Anton Mentrup

Ernst-Otto Renth

Armin Fugner

Original Assignee

Boehringer Ingelheim Kg

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-09-01

Filing date

1982-08-31

Publication date

1988-05-11

1982-08-31 Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg

1983-03-02 Publication of NO822932L publication Critical patent/NO822932L/en

1988-02-01 Publication of NO157738B publication Critical patent/NO157738B/en

1988-05-11 Publication of NO157738C publication Critical patent/NO157738C/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
- C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
- C07D265/36—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings condensed with one six-membered ring
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Pulmonology (AREA)
Endocrinology (AREA)
Immunology (AREA)
Reproductive Health (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)
Feed For Specific Animals (AREA)
Fodder In General (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)

NO822932A 1981-09-01 1982-08-31 ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES. NO157738C (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE19813134590 DE3134590A1 (en)	1981-09-01	1981-09-01	NEW BENZO HETEROCYCLES

Publications (3)

Publication Number	Publication Date
NO822932L NO822932L (en)	1983-03-02
NO157738B NO157738B (en)	1988-02-01
NO157738C true NO157738C (en)	1988-05-11

Family

ID=6140603

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO822932A NO157738C (en)	1981-09-01	1982-08-31	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES.

Country Status (25)

Country	Link
EP (1)	EP0073505B1 (en)
JP (1)	JPS5852278A (en)
KR (1)	KR890000380B1 (en)
AR (2)	AR231976A1 (en)
AT (1)	ATE16703T1 (en)
AU (1)	AU553589B2 (en)
CA (1)	CA1180012A (en)
CS (1)	CS236679B2 (en)
DD (1)	DD204477A5 (en)
DE (2)	DE3134590A1 (en)
DK (1)	DK158664C (en)
ES (3)	ES8308318A1 (en)
FI (1)	FI78475C (en)
GB (1)	GB2106105B (en)
GR (1)	GR77275B (en)
HU (1)	HU186112B (en)
IE (1)	IE53615B1 (en)
IL (1)	IL66683A0 (en)
NO (1)	NO157738C (en)
NZ (1)	NZ201777A (en)
PL (1)	PL139375B1 (en)
PT (1)	PT75478A (en)
SU (1)	SU1149876A3 (en)
YU (1)	YU42794B (en)
ZA (1)	ZA826349B (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4554284A (en) *	1984-09-12	1985-11-19	Smithkline Beckman Corporation	7-(2-Aminoethyl)-1,3-benzthia- or oxa-zol-2(3H)-ones
DE3743265A1 (en) *	1987-12-19	1989-06-29	Boehringer Ingelheim Kg	NEW AMMONIUM COMPOUNDS, THEIR MANUFACTURE AND USE
TW372967B (en) *	1994-12-27	1999-11-01	Kanebo Ltd	1,4 benzoxazine derivative, pharmaceutical composition containing the same and use thereof
DE10253282A1 (en) *	2002-11-15	2004-05-27	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration
US7056916B2 (en)	2002-11-15	2006-06-06	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Medicaments for the treatment of chronic obstructive pulmonary disease
PE20040950A1 (en)	2003-02-14	2005-01-01	Theravance Inc	BIPHENYL DERIVATIVES AS AGONISTS OF ß2-ADRENERGIC RECEPTORS AND AS ANTAGONISTS OF MUSCARINAL RECEPTORS
JP4516064B2 (en) *	2003-04-04	2010-08-04	ノバルティスアーゲー	Quinolin-2-one derivatives for the treatment of airway diseases
GB0307856D0 (en) *	2003-04-04	2003-05-14	Novartis Ag	Organic compounds
JP2007537187A (en) *	2004-05-13	2007-12-20	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	Hydroxy-substituted benzofused heterocyclic compounds for use as beta agonists in the treatment of respiratory diseases
US7307076B2 (en)	2004-05-13	2007-12-11	Boehringer Ingelheim International Gmbh	Beta agonists for the treatment of respiratory diseases
DE102004024453A1 (en) *	2004-05-14	2006-01-05	Boehringer Ingelheim Pharma Gmbh & Co. Kg	New long-acting bronchodilators for the treatment of respiratory diseases
DE102004024454A1 (en) *	2004-05-14	2005-12-08	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Novel enantiomerically pure beta agonists, process for their preparation and their use as pharmaceuticals
DE102004024452A1 (en) *	2004-05-14	2005-12-08	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Aerosol formulation for the inhalation of beta agonists
US7745621B2 (en)	2004-05-14	2010-06-29	Boehringer Ingelheim International Gmbh	Long acting bronchodilators for the treatment of respiratory diseases
US7220742B2 (en)	2004-05-14	2007-05-22	Boehringer Ingelheim International Gmbh	Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments
DE102004024451A1 (en)	2004-05-14	2005-12-22	Boehringer Ingelheim Pharma Gmbh & Co. Kg	Powder formulations for inhalation containing enantiomerically pure beta agonists
ES2530991T3 (en)	2005-08-15	2015-03-09	Boehringer Ingelheim Int	Procedure for obtaining betamimetics
US20070088030A1 (en)	2005-10-10	2007-04-19	Barbara Niklaus-Humke	Aerosol formulations for the inhalation of beta-agonists
GB0602778D0 (en)	2006-02-10	2006-03-22	Glaxo Group Ltd	Novel compound
JP2010500319A (en) *	2006-08-07	2010-01-07	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	Enantiomerically pure new beta agonists, methods for their preparation and their use as medicaments
UY30543A1 (en) *	2006-08-18	2008-03-31	Boehringer Ingelheim Int	AEROSOL FORMULATION FOR INHALATION OF BETA- AGONISTS
DK2125759T3 (en) *	2007-01-25	2011-09-19	Boehringer Ingelheim Int	Method of Preparation of Beta Mimetics

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2035749A1 (en) *	1969-02-06	1970-12-24	Bellon Labor Sa Roger
CA1041523A (en) *	1974-06-19	1978-10-31	Queen's University	Preparation of 1-oxapenicillins and novel intermediates therefor

1981
- 1981-09-01 DE DE19813134590 patent/DE3134590A1/en not_active Withdrawn
1982
- 1982-08-27 SU SU823483451A patent/SU1149876A3/en active
- 1982-08-28 DE DE8282107919T patent/DE3267702D1/en not_active Expired
- 1982-08-28 EP EP82107919A patent/EP0073505B1/en not_active Expired
- 1982-08-28 AT AT82107919T patent/ATE16703T1/en not_active IP Right Cessation
- 1982-08-30 PL PL1982238077A patent/PL139375B1/en unknown
- 1982-08-30 PT PT75478A patent/PT75478A/en not_active IP Right Cessation
- 1982-08-30 FI FI822985A patent/FI78475C/en not_active IP Right Cessation
- 1982-08-30 AR AR290473A patent/AR231976A1/en active
- 1982-08-30 DD DD82242881A patent/DD204477A5/en unknown
- 1982-08-30 YU YU1949/82A patent/YU42794B/en unknown
- 1982-08-31 GR GR69166A patent/GR77275B/el unknown
- 1982-08-31 HU HU822793A patent/HU186112B/en not_active IP Right Cessation
- 1982-08-31 IE IE2105/82A patent/IE53615B1/en not_active IP Right Cessation
- 1982-08-31 DK DK389082A patent/DK158664C/en not_active IP Right Cessation
- 1982-08-31 JP JP57151626A patent/JPS5852278A/en active Granted
- 1982-08-31 ZA ZA826349A patent/ZA826349B/en unknown
- 1982-08-31 NO NO822932A patent/NO157738C/en unknown
- 1982-08-31 GB GB08224810A patent/GB2106105B/en not_active Expired
- 1982-08-31 AU AU87874/82A patent/AU553589B2/en not_active Ceased
- 1982-08-31 IL IL66683A patent/IL66683A0/en not_active IP Right Cessation
- 1982-08-31 NZ NZ201777A patent/NZ201777A/en unknown
- 1982-08-31 ES ES515380A patent/ES8308318A1/en not_active Expired
- 1982-08-31 CS CS826329A patent/CS236679B2/en unknown
- 1982-08-31 CA CA000410462A patent/CA1180012A/en not_active Expired
- 1982-09-01 KR KR8203945A patent/KR890000380B1/en active
1983
- 1983-04-27 ES ES521870A patent/ES8402279A1/en not_active Expired
- 1983-04-27 ES ES521871A patent/ES521871A0/en active Granted
- 1983-11-17 AR AR294856A patent/AR231977A1/en active

Also Published As

Publication number	Publication date
IE822105L (en)	1983-03-01
CS236679B2 (en)	1985-05-15
YU194982A (en)	1984-12-31
PL238077A1 (en)	1984-04-09
YU42794B (en)	1988-12-31
ES521870A0 (en)	1984-01-16
FI822985A0 (en)	1982-08-30
DE3134590A1 (en)	1983-03-10
DK389082A (en)	1983-03-02
DK158664B (en)	1990-07-02
CA1180012A (en)	1984-12-27
NZ201777A (en)	1985-08-30
ATE16703T1 (en)	1985-12-15
HU186112B (en)	1985-06-28
KR890000380B1 (en)	1989-03-15
PT75478A (en)	1982-09-01
IL66683A0 (en)	1982-12-31
GB2106105B (en)	1985-07-10
ZA826349B (en)	1984-04-25
EP0073505A1 (en)	1983-03-09
GR77275B (en)	1984-09-11
FI78475B (en)	1989-04-28
AR231976A1 (en)	1985-04-30
DK158664C (en)	1991-01-14
GB2106105A (en)	1983-04-07
IE53615B1 (en)	1988-12-21
EP0073505B1 (en)	1985-11-27
JPS5852278A (en)	1983-03-28
AU8787482A (en)	1983-03-10
DE3267702D1 (en)	1986-01-09
DD204477A5 (en)	1983-11-30
AU553589B2 (en)	1986-07-24
FI822985L (en)	1983-03-02
ES515380A0 (en)	1983-08-16
NO157738B (en)	1988-02-01
ES8402279A1 (en)	1984-01-16
KR840001560A (en)	1984-05-07
AR231977A1 (en)	1985-04-30
FI78475C (en)	1989-08-10
NO822932L (en)	1983-03-02
JPH035392B2 (en)	1991-01-25
PL139375B1 (en)	1987-01-31
ES8308318A1 (en)	1983-08-16
ES8405778A1 (en)	1984-06-16
SU1149876A3 (en)	1985-04-07
ES521871A0 (en)	1984-06-16

Publication	Publication Date	Title
NO159016C (en)	1988-11-23	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PHENETANOLAMINE DERIVATIVES.
NO156785B (en)	1987-08-17	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CYCLOBUTAN DERIVATIVES.
NO157738C (en)	1988-05-11	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZOCSAZINONES AND BENZOCSAZOLINONES.
NO164025C (en)	1990-08-22	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 3-IMIDAZOLYLMETHYL-TETRAHYDROCARBAZOLONE DERIVATIVES.
NO154058C (en)	1986-07-09	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE N-HETEROCYCLYL-4-PIPERIDINAMINES.
NO162113C (en)	1989-11-08	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE PHENETANOLAMINE COMPOUNDS.
NO812344L (en)	1982-01-11	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE STEROIDS.
NO165397C (en)	1991-02-06	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOLO COMPOUNDS.
NO161497C (en)	1989-08-23	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE 9A-AZA-9A-HOMOERYTROMYCIN DERIVATIVES.
NO154492C (en)	1986-10-01	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC EFFECTIVE RELATIONS.
NO161317C (en)	1989-08-02	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE OXICAMS.
NO871028D0 (en)	1987-03-12	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE TIAZOL AND OKSAZOL DERIVATIVES.
NO158460C (en)	1988-09-14	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE RELATIONS.
NO164541C (en)	1990-10-17	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE BENZIMIDAZOLD DERIVATIVES.
NO169963C (en)	1992-08-26	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE, SUBSTITUTED 3,4-DIHYDRO-2H-BENZOPYRANES
NO155771C (en)	1987-05-27	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE AMINOPROPANOL DERIVATIVES.
NO163775C (en)	1990-07-18	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE ISOINDOLINYL-ALKYL-PIPERAZINES.
NO158417C (en)	1988-09-07	ANALOGUE PROCEDURE FOR THE PREPARATION OF PHARMACOLOGICALLY ACTIVE URINENTS AND TIOUR INGREDIENTS.
NO163692C (en)	1990-07-04	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE OKSAZAPHOSPHORIN-4-TIO-ALKANSULPHONIC ACIDS AND SALTS THEREOF.
NO162860C (en)	1990-02-28	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE BENZO (PYRANO AND TIOPYRANO) PYRIDINES.
NO167664C (en)	1991-11-27	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE CASTANOSPERMINESTERS AND GLYCOSIDES.
NO159090C (en)	1988-11-30	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE PYRIDOINDOL DERIVATIVES.
NO163570C (en)	1990-06-20	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTIC ACTIVE ACYLAMINOMITOSANES.
NO894949D0 (en)	1989-12-08	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY EFFECTIVE BENZOPYRANYLPYRROLINE UNDIVATIVES.
NO165493C (en)	1991-02-20	ANALOGUE PROCEDURE FOR THE PREPARATION OF THERAPEUTICALLY ACTIVE CHINAZOL INDIA AND PYRIDOPYRIMID INDIA.