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MX2015005947A - Formas de dosificacion de ruxolitinib de liberacion sostenida. - Google Patents

Formas de dosificacion de ruxolitinib de liberacion sostenida.

Info

Publication number
MX2015005947A
MX2015005947A MX2015005947A MX2015005947A MX2015005947A MX 2015005947 A MX2015005947 A MX 2015005947A MX 2015005947 A MX2015005947 A MX 2015005947A MX 2015005947 A MX2015005947 A MX 2015005947A MX 2015005947 A MX2015005947 A MX 2015005947A
Authority
MX
Mexico
Prior art keywords
ruxolitinib
sustained
dosage forms
release dosage
useful
Prior art date
Application number
MX2015005947A
Other languages
English (en)
Inventor
Yong Ni
Bhavnish Parikh
Krishnaswamy Yeleswaram
Susan Erickson-Viitanen
William V Williams
Original Assignee
Incyte Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=49681181&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2015005947(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Incyte Corp filed Critical Incyte Corp
Publication of MX2015005947A publication Critical patent/MX2015005947A/es

Links

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Neurology (AREA)
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  • Communicable Diseases (AREA)
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  • Neurosurgery (AREA)
  • Ophthalmology & Optometry (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Nutrition Science (AREA)
  • Pulmonology (AREA)
  • Cardiology (AREA)
  • Reproductive Health (AREA)
  • Child & Adolescent Psychology (AREA)

Abstract

La presente invención se refiere a formulaciones de liberación sostenida y formas de dosificación de ruxolitinib o su sal farmacéuticamente aceptable, que son útiles en el tratamiento de enfermedades relacionadas con las cinasa Janus como trastornos mieloproliferativos.
MX2015005947A 2012-11-15 2013-11-14 Formas de dosificacion de ruxolitinib de liberacion sostenida. MX2015005947A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201261726893P 2012-11-15 2012-11-15
US201361769408P 2013-02-26 2013-02-26
PCT/US2013/070012 WO2014078486A1 (en) 2012-11-15 2013-11-14 Sustained-release dosage forms of ruxolitinib

Publications (1)

Publication Number Publication Date
MX2015005947A true MX2015005947A (es) 2015-09-08

Family

ID=49681181

Family Applications (3)

Application Number Title Priority Date Filing Date
MX2020012676A MX2020012676A (es) 2012-11-15 2013-11-14 Formas de dosificación de ruxolitinib de liberación sostenida.
MX2015005947A MX2015005947A (es) 2012-11-15 2013-11-14 Formas de dosificacion de ruxolitinib de liberacion sostenida.
MX2023000255A MX2023000255A (es) 2012-11-15 2015-05-12 Formas de dosificacion de ruxolitinib de liberacion sostenida.

Family Applications Before (1)

Application Number Title Priority Date Filing Date
MX2020012676A MX2020012676A (es) 2012-11-15 2013-11-14 Formas de dosificación de ruxolitinib de liberación sostenida.

Family Applications After (1)

Application Number Title Priority Date Filing Date
MX2023000255A MX2023000255A (es) 2012-11-15 2015-05-12 Formas de dosificacion de ruxolitinib de liberacion sostenida.

Country Status (35)

Country Link
US (7) US10166191B2 (es)
EP (2) EP2919766B1 (es)
JP (4) JP2015537030A (es)
KR (3) KR20220162825A (es)
CN (3) CN105007901A (es)
AR (1) AR093490A1 (es)
AU (4) AU2013344780B2 (es)
BR (1) BR112015010663B1 (es)
CA (2) CA2890755C (es)
CL (1) CL2015001286A1 (es)
CR (2) CR20190073A (es)
CY (1) CY1124446T1 (es)
DK (1) DK2919766T3 (es)
EA (1) EA201590930A1 (es)
ES (1) ES2880814T3 (es)
HK (1) HK1213796A1 (es)
HR (1) HRP20211158T1 (es)
HU (1) HUE055894T2 (es)
IL (4) IL317061A (es)
LT (1) LT2919766T (es)
MX (3) MX2020012676A (es)
MY (1) MY191357A (es)
NZ (2) NZ708157A (es)
PE (2) PE20200175A1 (es)
PH (2) PH12020551186B1 (es)
PL (1) PL2919766T3 (es)
PT (1) PT2919766T (es)
RS (1) RS62329B1 (es)
SG (3) SG10202111768XA (es)
SI (1) SI2919766T1 (es)
SM (1) SMT202100436T1 (es)
TW (4) TWI761825B (es)
UA (1) UA120834C2 (es)
WO (1) WO2014078486A1 (es)
ZA (1) ZA202202711B (es)

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LT2426129T (lt) 2005-12-13 2017-02-10 Incyte Holdings Corporation Heteroarilu pakeisti pirolo[2,3-b]piridinai ir pirolo[2,3-b]pirimidinai kaip janus kinazės inhibitoriai
RS54878B1 (sr) 2007-06-13 2016-10-31 Incyte Holdings Corp Kristalne soli inhibitora janus kinaze (r)-3-(4-(7h-pirolo[2,3-d]pirimidin-4-il)-1h-pirazol-1-il)-3-ciklopentilpropionitril
WO2010135650A1 (en) 2009-05-22 2010-11-25 Incyte Corporation N-(HETERO)ARYL-PYRROLIDINE DERIVATIVES OF PYRAZOL-4-YL-PYRROLO[2,3-d]PYRIMIDINES AND PYRROL-3-YL-PYRROLO[2,3-d]PYRIMIDINES AS JANUS KINASE INHIBITORS
UA106078C2 (uk) 2009-05-22 2014-07-25 Інсайт Корпорейшн 3-[4-(7H-ПІРОЛО[2,3-d]ПІРИМІДИН-4-ІЛ)-1H-ПІРАЗОЛ-1-ІЛ]ОКТАН- АБО ГЕПТАННІТРИЛ ЯК JAK-ІНГІБІТОРИ
MX364636B (es) 2010-03-10 2019-05-03 Incyte Corp Derivados de piperidin-4-il azetidina como inhibidores de janus cinasa 1 (jak1).
SI2574168T1 (sl) 2010-05-21 2016-07-29 Incyte Holdings Corporation Topična formulacija zaviralca jak
SG190839A1 (en) 2010-11-19 2013-07-31 Incyte Corp Cyclobutyl substituted pyrrolopyridine and pyrrolopyrimidine derivatives as jak inhibitors
AU2012273164B2 (en) 2011-06-20 2015-05-28 Incyte Holdings Corporation Azetidinyl phenyl, pyridyl or pyrazinyl carboxamide derivatives as JAK inhibitors
UA111854C2 (uk) 2011-09-07 2016-06-24 Інсайт Холдінгс Корпорейшн Способи і проміжні сполуки для отримання інгібіторів jak
ES2867048T3 (es) * 2012-06-15 2021-10-20 Concert Pharmaceuticals Inc Derivados deuterados de ruxolitinib
AR093308A1 (es) 2012-11-01 2015-05-27 Incyte Corp Derivados triciclicos fusionados de tiofeno como inhibidores de jak
JP2015537030A (ja) 2012-11-15 2015-12-24 インサイト・コーポレイションＩｎｃｙｔｅ Ｃｏｒｐｏｒａｔｉｏｎ ルキソリチニブの徐放性投薬形態
KR102366356B1 (ko) 2013-03-06 2022-02-23 인사이트 홀딩스 코포레이션 Jak 저해제를 제조하기 위한 방법 및 중간생성물
EA036448B1 (ru) 2013-05-17 2020-11-11 Инсайт Корпорейшн Производные бипиразола в качестве ингибиторов jak
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