Nothing Special   »   [go: up one dir, main page]

Metformin rescues Parkinson's disease phenotypes caused by hyperactive mitochondria

Proc Natl Acad Sci U S A. 2020 Oct 20;117(42):26438-26447. doi: 10.1073/pnas.2009838117. Epub 2020 Oct 6.

Abstract

Metabolic dysfunction occurs in many age-related neurodegenerative diseases, yet its role in disease etiology remains poorly understood. We recently discovered a potential causal link between the branched-chain amino acid transferase BCAT-1 and the neurodegenerative movement disorder Parkinson's disease (PD). RNAi-mediated knockdown of Caenorhabditis elegans bcat-1 is known to recapitulate PD-like features, including progressive motor deficits and neurodegeneration with age, yet the underlying mechanisms have remained unknown. Using transcriptomic, metabolomic, and imaging approaches, we show here that bcat-1 knockdown increases mitochondrial respiration and induces oxidative damage in neurons through mammalian target of rapamycin-independent mechanisms. Increased mitochondrial respiration, or "mitochondrial hyperactivity," is required for bcat-1(RNAi) neurotoxicity. Moreover, we show that post-disease-onset administration of the type 2 diabetes medication metformin reduces mitochondrial respiration to control levels and significantly improves both motor function and neuronal viability. Taken together, our findings suggest that mitochondrial hyperactivity may be an early event in the pathogenesis of PD, and that strategies aimed at reducing mitochondrial respiration may constitute a surprising new avenue for PD treatment.

Keywords: Caenorhabditis elegans; Parkinson’s disease; branched-chain amino acid metabolism; metformin; mitochondria.

Publication types

  • Research Support, N.I.H., Extramural
  • Research Support, Non-U.S. Gov't

MeSH terms

  • Amino Acids, Branched-Chain / metabolism
  • Amino Acids, Branched-Chain / physiology
  • Animals
  • Caenorhabditis elegans / metabolism
  • Caenorhabditis elegans Proteins / metabolism
  • Disease Models, Animal
  • Metformin / metabolism
  • Metformin / pharmacology*
  • Mitochondria / drug effects*
  • Neurons / drug effects
  • Parkinson Disease / drug therapy*
  • Parkinson Disease / metabolism
  • Phenotype

Substances

  • Amino Acids, Branched-Chain
  • Caenorhabditis elegans Proteins
  • Metformin

Associated data

  • Dryad/10.5061/dryad.5mkkwh72q