3-Metiltiofentanil

3-Metiltiofentanil
(IUPAC) ime
	(RS)-N3-metil-1-[2-(2-tienil)etil]piperidin-4-ilN-fenilpropanamid
Klinički podaci
Identifikatori
CAS broj	86052-04-2
ATC kod	nije dodeljen
PubChem	62296
DrugBank	DB01439
ChemSpider	56092
ChEBI	CHEBI:53763
Hemijski podaci
Formula	C21H28N2OS
Mol. masa	356,526 g/mol
SMILES	eMolekuli & PubHem
InChI
	InChI=1S/C21H28N2OS/c1-3-21(24)23(18-8-5-4-6-9-18)20-12-14-22(16-17(20)2)13-11-19-10-7-15-25-19/h4-10,15,17,20H,3,11-14,16H2,1-2H3 ; Key: SRARDYUHGVMEQI-UHFFFAOYSA-N
Sinonimi	N-[3-metil-1-(2-tiofen-2-iletil)-4-piperidil]-N-fenil-propanamid; 3-metil-tiofentanil
Farmakoinformacioni podaci
Trudnoća	?
Pravni status	? (CA) ? (UK) ? (SAD)

3-Metiltiofentanil je opioidni analgetik koji je analog fentanila.

3-Metiltiofentanil je bio tokom kraćeg perioda u prodaji na crno u Americi tokom 1980-tih, pre nego što je uveden zakon kojim se kontrolišu čitave familije lekova po osnovi njihove strukturne sličnosti.^[4]

3-Metiltiofentanil ima slično dejstvo sa fentanilom. Nuspojave fentanilnih analoga su slične nuspojavama fentanila, i obuhvataju svrab, mučninu i potencijalno ozbiljnu respiratornu derpesiju koja može da dovede do smrtnog slučaja.

Reference

↑ Li Q, Cheng T, Wang Y, Bryant SH (2010). „PubChem as a public resource for drug discovery.”. Drug Discov Today 15 (23-24): 1052-7. DOI:10.1016/j.drudis.2010.10.003. PMID 20970519. edit
↑ Evan E. Bolton, Yanli Wang, Paul A. Thiessen, Stephen H. Bryant (2008). „Chapter 12 PubChem: Integrated Platform of Small Molecules and Biological Activities”. Annual Reports in Computational Chemistry 4: 217-241. DOI:10.1016/S1574-1400(08)00012-1.
↑ Hettne KM, Williams AJ, van Mulligen EM, Kleinjans J, Tkachenko V, Kors JA. (2010). „Automatic vs. manual curation of a multi-source chemical dictionary: the impact on text mining”. J Cheminform 2 (1): 3. DOI:10.1186/1758-2946-2-3. PMID 20331846. edit
↑ Henderson GL. Designer Drugs: Past History and Future Prospects. Journal of Forensic Sciences 1988; 33(2):569-575.

[1] Li Q, Cheng T, Wang Y, Bryant SH (2010). „PubChem as a public resource for drug discovery.”. Drug Discov Today 15 (23-24): 1052-7. DOI:10.1016/j.drudis.2010.10.003. PMID 20970519. edit

[2] Evan E. Bolton, Yanli Wang, Paul A. Thiessen, Stephen H. Bryant (2008). „Chapter 12 PubChem: Integrated Platform of Small Molecules and Biological Activities”. Annual Reports in Computational Chemistry 4: 217-241. DOI:10.1016/S1574-1400(08)00012-1.

[3] Hettne KM, Williams AJ, van Mulligen EM, Kleinjans J, Tkachenko V, Kors JA. (2010). „Automatic vs. manual curation of a multi-source chemical dictionary: the impact on text mining”. J Cheminform 2 (1): 3. DOI:10.1186/1758-2946-2-3. PMID 20331846. edit

[4] Henderson GL. Designer Drugs: Past History and Future Prospects. Journal of Forensic Sciences 1988; 33(2):569-575.

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