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SG10201808053XA - Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders - Google Patents

Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders

Info

Publication number
SG10201808053XA
SG10201808053XA SG10201808053XA SG10201808053XA SG10201808053XA SG 10201808053X A SG10201808053X A SG 10201808053XA SG 10201808053X A SG10201808053X A SG 10201808053XA SG 10201808053X A SG10201808053X A SG 10201808053XA SG 10201808053X A SG10201808053X A SG 10201808053XA
Authority
SG
Singapore
Prior art keywords
treatment
pi3k
mediated disorders
heterocyclic compounds
gamma mediated
Prior art date
Application number
SG10201808053XA
Inventor
Jeffery Kutok
David Winkler
Vito Palombella
Original Assignee
Infinity Pharmaceuticals Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Infinity Pharmaceuticals Inc filed Critical Infinity Pharmaceuticals Inc
Publication of SG10201808053XA publication Critical patent/SG10201808053XA/en

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    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/437Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a five-membered ring having nitrogen as a ring hetero atom, e.g. indolizine, beta-carboline
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    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/535Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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    • A61K31/53771,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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Abstract

HETEROCYCLIC COMPOUNDS FOR USE IN THE TREATMENT OF PI3K- GAMMA MEDIATED DISORDERS Compounds and pharmaceutical compositions that modulate kinase activity, including PI3 kinase activity, and compounds, pharmaceutical compositions, and methods of treatment of diseases and conditions associated with kinase activity, including PI3 kinase activity, are described herein. [FIG.2]
SG10201808053XA 2014-03-19 2015-03-18 Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders SG10201808053XA (en)

Applications Claiming Priority (7)

Application Number Priority Date Filing Date Title
US201461955717P 2014-03-19 2014-03-19
US201461980484P 2014-04-16 2014-04-16
US201462000923P 2014-05-20 2014-05-20
US201462033008P 2014-08-04 2014-08-04
US201462059766P 2014-10-03 2014-10-03
US201462075173P 2014-11-04 2014-11-04
US201562101980P 2015-01-09 2015-01-09

Publications (1)

Publication Number Publication Date
SG10201808053XA true SG10201808053XA (en) 2018-10-30

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SG11201607705XA SG11201607705XA (en) 2014-03-19 2015-03-18 Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders
SG10201808053XA SG10201808053XA (en) 2014-03-19 2015-03-18 Heterocyclic compounds for use in the treatment of pi3k-gamma mediated disorders

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US (4) US9775844B2 (en)
EP (2) EP4066834A1 (en)
JP (1) JP6701088B2 (en)
CN (3) CN113620958A (en)
AU (1) AU2015231413B2 (en)
CA (1) CA2943075C (en)
DK (1) DK3119397T3 (en)
EA (1) EA201691872A1 (en)
ES (1) ES2913486T3 (en)
IL (1) IL247841B (en)
MX (1) MX2016012021A (en)
NZ (1) NZ724368A (en)
PH (1) PH12016501809A1 (en)
PT (1) PT3119397T (en)
SG (2) SG11201607705XA (en)
WO (1) WO2015143012A1 (en)

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