JPS5671084A - 5,8,11,14,17-eicosapentaenoic acid alpha-tocopherol ester and its preparation - Google Patents
5,8,11,14,17-eicosapentaenoic acid alpha-tocopherol ester and its preparationInfo
- Publication number
- JPS5671084A JPS5671084A JP14774179A JP14774179A JPS5671084A JP S5671084 A JPS5671084 A JP S5671084A JP 14774179 A JP14774179 A JP 14774179A JP 14774179 A JP14774179 A JP 14774179A JP S5671084 A JPS5671084 A JP S5671084A
- Authority
- JP
- Japan
- Prior art keywords
- eicosapentaenoic acid
- preparation
- tocopherol ester
- acid
- tocopherol
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrane Compounds (AREA)
Abstract
NEW MATERIAL:5,8,11,14,17-Eicosapentaenoic acid α-tocopherol ester.
USE: Blood platelet coagulation inhibitor: it is more stable and absorbable than 5,8, 11,14,17-eicosapentaenoic acid.
PREPARATION: 5,8,11,14,17-Eicosapentaenoic acid or its reactive derivative such as its acid halide or acid anhydride and α-tocopherol are made to react in an inert solvent such as water or dichloromethane at room temperature to refluxing one of the solvent for 1W20hr to give 5,8,11,14,17-eicosapentaenoic acid α-tocopherol ester. When 5,8,11,14,17-eicosapentaenoic acid is used directly, the reaction preferably is effected in the presence of N,N-dicyclohexylcarbodiimide or 2-substituted pyridinium salt and a base.
COPYRIGHT: (C)1981,JPO&Japio
Priority Applications (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14774179A JPS5671084A (en) | 1979-11-16 | 1979-11-16 | 5,8,11,14,17-eicosapentaenoic acid alpha-tocopherol ester and its preparation |
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP14774179A JPS5671084A (en) | 1979-11-16 | 1979-11-16 | 5,8,11,14,17-eicosapentaenoic acid alpha-tocopherol ester and its preparation |
Publications (2)
Publication Number | Publication Date |
---|---|
JPS5671084A true JPS5671084A (en) | 1981-06-13 |
JPS6332071B2 JPS6332071B2 (en) | 1988-06-28 |
Family
ID=15437087
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
JP14774179A Granted JPS5671084A (en) | 1979-11-16 | 1979-11-16 | 5,8,11,14,17-eicosapentaenoic acid alpha-tocopherol ester and its preparation |
Country Status (1)
Country | Link |
---|---|
JP (1) | JPS5671084A (en) |
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59222487A (en) * | 1983-06-02 | 1984-12-14 | Terumo Corp | Unsaturated fatty acid derivative |
FR2825088A1 (en) * | 2001-05-25 | 2002-11-29 | Derma Dev | NOVEL TOCOPHEROL ESTERS, PROCESSES FOR OBTAINING SAME AND USES THEREOF |
-
1979
- 1979-11-16 JP JP14774179A patent/JPS5671084A/en active Granted
Cited By (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS59222487A (en) * | 1983-06-02 | 1984-12-14 | Terumo Corp | Unsaturated fatty acid derivative |
FR2825088A1 (en) * | 2001-05-25 | 2002-11-29 | Derma Dev | NOVEL TOCOPHEROL ESTERS, PROCESSES FOR OBTAINING SAME AND USES THEREOF |
Also Published As
Publication number | Publication date |
---|---|
JPS6332071B2 (en) | 1988-06-28 |
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