IN2014DN08922A - - Google Patents
Info
- Publication number
- IN2014DN08922A IN2014DN08922A IN8922DEN2014A IN2014DN08922A IN 2014DN08922 A IN2014DN08922 A IN 2014DN08922A IN 8922DEN2014 A IN8922DEN2014 A IN 8922DEN2014A IN 2014DN08922 A IN2014DN08922 A IN 2014DN08922A
- Authority
- IN
- India
- Prior art keywords
- pyrazine
- difluoromethyl
- action
- hibitory
- chloropyrazine
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/24—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Plural Heterocyclic Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US201261639362P | 2012-04-27 | 2012-04-27 | |
| PCT/JP2013/062863 WO2013162065A1 (fr) | 2012-04-27 | 2013-04-25 | Procédé de production d'acide 5-(difluorométhyl)pyrazine-2-carboxylique et d'un intermédiaire pour sa production |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| IN2014DN08922A true IN2014DN08922A (fr) | 2015-05-22 |
Family
ID=49483351
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| IN8922DEN2014 IN2014DN08922A (fr) | 2012-04-27 | 2013-04-25 |
Country Status (14)
| Country | Link |
|---|---|
| US (1) | US9227942B2 (fr) |
| EP (1) | EP2841423B1 (fr) |
| JP (1) | JP6118817B2 (fr) |
| CN (1) | CN104245680B (fr) |
| BR (1) | BR112014026474A2 (fr) |
| CA (1) | CA2871264A1 (fr) |
| ES (1) | ES2615304T3 (fr) |
| HU (1) | HUE030534T2 (fr) |
| IL (1) | IL235161A0 (fr) |
| IN (1) | IN2014DN08922A (fr) |
| MX (1) | MX2014012683A (fr) |
| RU (1) | RU2014142545A (fr) |
| SG (1) | SG11201406589PA (fr) |
| WO (1) | WO2013162065A1 (fr) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JO3318B1 (ar) | 2013-06-18 | 2019-03-13 | Lilly Co Eli | مثبطات bace |
| EP4101843A4 (fr) * | 2020-02-06 | 2024-03-27 | Agc Inc. | Procédé de fabrication de dérivé d'acide difluoroacétique substitué par un hétérocycle aromatique |
| CN112645890B (zh) * | 2020-12-25 | 2022-08-12 | 江苏广域化学有限公司 | 2-吡嗪羧酸酯类化合物的合成方法 |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2007208494A1 (en) | 2006-01-12 | 2007-08-02 | Merck Sharp & Dohme Corp. | Fluorinated arylamide derivatives |
| ES2548774T3 (es) | 2008-01-18 | 2015-10-20 | Eisai R&D Management Co., Ltd. | Derivado de aminodihidrotiazina condensado |
| NZ590320A (en) * | 2008-07-14 | 2012-12-21 | Gilead Sciences Inc | Fused heterocyclyc inhibitors of histone deacetylase and/or cyclin-dependent kinases |
| TW201016708A (en) | 2008-09-30 | 2010-05-01 | Eisai R&D Man Co Ltd | Novel fused aminodihydrothiazine derivative |
| AR077277A1 (es) | 2009-07-09 | 2011-08-17 | Lilly Co Eli | Compuestos de biciclo (1,3)tiazin-2-amina formulacion farmaceutica que lo comprende y su uso para la manufactura de un medicamento util para el tratamiento de la enfermedad de alzheimer |
| GB0912778D0 (en) | 2009-07-22 | 2009-08-26 | Eisai London Res Lab Ltd | Fused aminodihydro-oxazine derivatives |
| GB0912777D0 (en) | 2009-07-22 | 2009-08-26 | Eisai London Res Lab Ltd | Fused aminodihydropyrimidone derivatives |
| JP5696355B2 (ja) * | 2009-11-18 | 2015-04-08 | セントラル硝子株式会社 | 芳香族ジフルオロメチル化合物の製造方法 |
| US8673894B2 (en) | 2010-05-07 | 2014-03-18 | Hoffmann-La Roche Inc. | 2,5,6,7-tetrahydro-[1,4]oxazepin-3-ylamine or 2,3,6,7-tetrahydro-[1,4]oxazepin-5-ylamine compounds |
| JP5679855B2 (ja) | 2011-02-14 | 2015-03-04 | 国立大学法人群馬大学 | ジフルオロメチル化ヘテロアリール化合物の製造方法 |
-
2013
- 2013-04-25 IN IN8922DEN2014 patent/IN2014DN08922A/en unknown
- 2013-04-25 JP JP2014547207A patent/JP6118817B2/ja active Active
- 2013-04-25 SG SG11201406589PA patent/SG11201406589PA/en unknown
- 2013-04-25 MX MX2014012683A patent/MX2014012683A/es unknown
- 2013-04-25 EP EP13781634.4A patent/EP2841423B1/fr active Active
- 2013-04-25 US US14/396,261 patent/US9227942B2/en active Active
- 2013-04-25 HU HUE13781634A patent/HUE030534T2/hu unknown
- 2013-04-25 ES ES13781634.4T patent/ES2615304T3/es active Active
- 2013-04-25 CA CA2871264A patent/CA2871264A1/fr not_active Abandoned
- 2013-04-25 RU RU2014142545A patent/RU2014142545A/ru unknown
- 2013-04-25 BR BR112014026474A patent/BR112014026474A2/pt not_active Application Discontinuation
- 2013-04-25 WO PCT/JP2013/062863 patent/WO2013162065A1/fr active Application Filing
- 2013-04-25 CN CN201380021262.XA patent/CN104245680B/zh active Active
-
2014
- 2014-10-19 IL IL235161A patent/IL235161A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ES2615304T3 (es) | 2017-06-06 |
| JP6118817B2 (ja) | 2017-04-19 |
| EP2841423A4 (fr) | 2015-09-09 |
| EP2841423A1 (fr) | 2015-03-04 |
| SG11201406589PA (en) | 2014-11-27 |
| CN104245680A (zh) | 2014-12-24 |
| IL235161A0 (en) | 2014-12-31 |
| CN104245680B (zh) | 2016-11-23 |
| US20150087836A1 (en) | 2015-03-26 |
| US9227942B2 (en) | 2016-01-05 |
| RU2014142545A (ru) | 2016-06-27 |
| CA2871264A1 (fr) | 2013-10-31 |
| BR112014026474A2 (pt) | 2017-06-27 |
| HUE030534T2 (hu) | 2017-05-29 |
| JP2015514676A (ja) | 2015-05-21 |
| EP2841423B1 (fr) | 2016-11-30 |
| MX2014012683A (es) | 2015-01-16 |
| WO2013162065A1 (fr) | 2013-10-31 |
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