IL150163A - PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS - Google Patents

PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS

Info

Publication number: IL150163A
Authority: IL; Israel
Prior art keywords: pyrazolo; novel; compounds; pharmaceutical compositions; pyrimidine derivatives
Prior art date: 1996-07-24

Application number

IL150163A

Original Assignee

Du Pont Pharm Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1996-07-24

Filing date

2002-06-11

Publication date

2010-12-30

1997-07-23 Priority claimed from US08/899,242 external-priority patent/US6124289A/en

1997-07-23 Priority claimed from PCT/US1997/013072 external-priority patent/WO1998003510A1/en

2002-06-11 Application filed by Du Pont Pharm Co filed Critical Du Pont Pharm Co

2010-12-30 Publication of IL150163A publication Critical patent/IL150163A/en

Links

IL150163A 1996-07-24 2002-06-11 PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS IL150163A (en)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US68604796A	1996-07-24	1996-07-24
US2329096P	1996-07-24	1996-07-24
US08/899,242 US6124289A (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines
PCT/US1997/013072 WO1998003510A1 (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines

Publications (1)

Publication Number	Publication Date
IL150163A true IL150163A (en)	2010-12-30

Family

ID=27362048

Family Applications (4)

Application Number	Title	Priority Date	Filing Date
IL12787197A IL127871A0 (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines
IL127871A IL127871A (en)	1996-07-24	1998-12-30	PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES
IL150163A IL150163A (en)	1996-07-24	2002-06-11	PHARMACEUTICAL COMPOSITIONS COMPRISING PYRAZOLO[1,5-a]PYRIMIDINE DERIVATIVES AND SOME NOVEL SUCH COMPOUNDS
IL164513A IL164513A (en)	1996-07-24	2004-10-12	Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments

Family Applications Before (2)

Application Number	Title	Priority Date	Filing Date
IL12787197A IL127871A0 (en)	1996-07-24	1997-07-23	Azolo triazines and pyrimidines
IL127871A IL127871A (en)	1996-07-24	1998-12-30	PHARMACEUTICAL COMPOSITIONS CONTAINING CRF ANTAGONIST 3-ARYL-PYRAZOLO (AND 1,2,3-TRIAZOLO) [1,5-a]-1,3,5-TRIAZINE DERIVATIVES AND SOME NEW SUCH DERIVATIVES

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
IL164513A IL164513A (en)	1996-07-24	2004-10-12	Pyrazolopyrimidines, pharmaceutical compositions containing them and their use in the preparation of medicaments

Country Status (15)

Country	Link
JP (2)	JP4704521B2 (en)
CN (3)	CN1104432C (en)
AR (1)	AR049583A2 (en)
BR (1)	BR9710544A (en)
CA (1)	CA2259583C (en)
CZ (1)	CZ299451B6 (en)
EA (1)	EA004403B1 (en)
EE (1)	EE04316B1 (en)
HR (1)	HRP970413A2 (en)
IL (4)	IL127871A0 (en)
NO (1)	NO315610B3 (en)
NZ (1)	NZ333777A (en)
PL (1)	PL195762B1 (en)
SI (1)	SI9720045B (en)
SK (1)	SK286461B6 (en)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ES2282401T3 (en) *	2001-03-13	2007-10-16	Bristol-Myers Squibb Pharma Company	4- (2-BUTILAMINO) -2,7-DIMETHYL-8- (2-METHYL-6-METOXIPIRID-3-IL) PIRAZOLO - 1,5-A-1,3,5-TRIAZINE, ITS ENANTIOMERS AND PHARMACEUTICALLY SALTS ACCEPTABLE AS LIGANDS OF THE RECEIVER OF THE CROTICOTROPINE RELEASE FACTOR.
WO2004110454A1 (en) *	2003-06-13	2004-12-23	Ishihara Sangyo Kaisha, Ltd.	COMPOSITION FOR TREATMENT FOR OR PREVENTION OF DISEASE NECESSITATING ADMINISTRATION OF ADENOSINE A2a RECEPTOR AGONIST
US7329662B2 (en) *	2003-10-03	2008-02-12	Hoffmann-La Roche Inc.	Pyrazolo-pyridine
GB0519957D0 (en) *	2005-09-30	2005-11-09	Sb Pharmco Inc	Chemical compound
CA2663511C (en) *	2006-09-20	2012-12-04	Eli Lilly And Company	Thiazole pyrazolopyrimidines as crf1 receptor antagonists
CN103694242B (en) *	2013-12-10	2016-01-06	昆明翔昊科技有限公司	Pyrazolopyrimidines and pharmaceutical composition thereof and its application in pharmacy
EA202090450A1 (en)	2017-08-14	2020-09-24	Спрюс Биосайнсес, Инк.	RECEPTOR ANTAGONISTS OF THE CORTICOTROPIN-RELEASING FACTOR
CN112608316B (en) *	2019-07-30	2022-10-21	厦门宝太生物科技股份有限公司	Pyrazolotriazine adenosine receptor antagonist
JP2023537598A (en)	2020-08-12	2023-09-04	スプルースバイオサイエンシーズ，インク．	Methods and compositions for treating polycystic ovary syndrome
US11708372B2 (en)	2021-11-19	2023-07-25	Spruce Biosciences, Inc.	Crystalline composition of tildacerfont and methods of use and preparation thereof

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3995039A (en) *	1975-05-27	1976-11-30	Merck & Co., Inc.	Pyrazolo [1,5-a] [1,3,5] triazines
JPS6157587A (en) *	1984-08-29	1986-03-24	Shionogi & Co Ltd	Condensed heterocyclic derivative and antiulcerative
US4824834A (en) *	1986-10-31	1989-04-25	Otsuka Pharmaceutical Company, Limited	Pyrazolotriazine compounds
JP2691317B2 (en) *	1989-08-25	1997-12-17	株式会社大塚製薬工場	4-Hydroxy-8- (3-lower alkoxy-4-phenylsulfinylphenyl) pyrazolo [1,5-a] -1,3,5-triazine optically active salts and process for producing the same
US5420128A (en) *	1990-10-09	1995-05-30	Otsuka Pharmaceutical Co., Ltd.	Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor
CA2107479C (en) *	1991-04-22	1997-12-16	Makoto Inoue	Pyrazolo[1,5-a]pyrimidine derivatives and anti-inflammatory agent containing the same
US5356897A (en) *	1991-09-09	1994-10-18	Fujisawa Pharmaceutical Co., Ltd.	3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines

1997
- 1997-07-23 SI SI9720045A patent/SI9720045B/en active Search and Examination
- 1997-07-23 CA CA002259583A patent/CA2259583C/en not_active Expired - Lifetime
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/en not_active IP Right Cessation
- 1997-07-23 CN CN97196525A patent/CN1104432C/en not_active Expired - Lifetime
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 SK SK97-99A patent/SK286461B6/en not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/en not_active Expired - Fee Related
- 1997-07-23 EA EA199900158A patent/EA004403B1/en not_active IP Right Cessation
- 1997-07-23 EE EEP199900019A patent/EE04316B1/en unknown
- 1997-07-23 BR BR9710544A patent/BR9710544A/en not_active IP Right Cessation
- 1997-07-23 PL PL97331523A patent/PL195762B1/en unknown
- 1997-07-23 IL IL12787197A patent/IL127871A0/en unknown
- 1997-07-24 HR HRP970413 patent/HRP970413A2/en not_active Application Discontinuation
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
1999
- 1999-01-21 NO NO19990264A patent/NO315610B3/en not_active IP Right Cessation
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/en not_active Expired - Lifetime
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/en active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/en not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/en not_active Application Discontinuation

Also Published As

Publication number	Publication date
PL195762B1 (en)	2007-10-31
IL164513A (en)	2010-04-29
NZ333777A (en)	2000-07-28
EA004403B1 (en)	2004-04-29
CN1225637A (en)	1999-08-11
NO990264D0 (en)	1999-01-21
EA199900158A1 (en)	1999-10-28
IL127871A (en)	2010-04-29
IL164513A0 (en)	2005-12-18
SI9720045A (en)	1999-10-31
CA2259583C (en)	2009-11-17
CN1388126A (en)	2003-01-01
JP2005097257A (en)	2005-04-14
NO315610B1 (en)	2003-09-29
SK286461B6 (en)	2008-10-07
BR9710544A (en)	1999-08-17
SK9799A3 (en)	2005-04-01
JP4194539B2 (en)	2008-12-10
JP2002513382A (en)	2002-05-08
CN1327793A (en)	2001-12-26
JP4704521B2 (en)	2011-06-15
NO315610B3 (en)	2003-09-29
SI9720045B (en)	2008-02-29
PL331523A1 (en)	1999-07-19
NO990264L (en)	1999-03-10
CN1250223C (en)	2006-04-12
CN1104432C (en)	2003-04-02
IL127871A0 (en)	1999-10-28
EE04316B1 (en)	2004-06-15
CA2259583A1 (en)	1998-01-29
EE9900019A (en)	1999-08-16
CZ18499A3 (en)	1999-11-17
CZ299451B6 (en)	2008-07-30
HRP970413A2 (en)	1998-10-31
AR049583A2 (en)	2006-08-16

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Legal Events

Date	Code	Title	Description
2015-06-30	KB	Patent renewed
2018-02-28	EXP	Patent expired