FI111078B - Menetelmä mometasonifuroaattimonohydraatin valmistamiseksi - Google Patents

Menetelmä mometasonifuroaattimonohydraatin valmistamiseksi Download PDF

Info

Publication number: FI111078B
Authority: FI; Finland
Prior art keywords: mometasone furoate; water; monohydrate; organic solvent; furoate monohydrate
Prior art date: 1990-09-10

Application number

FI931031A

Other languages

English (en)

Finnish (fi)

Swedish (sv)

Other versions

FI931031A0 (fi

FI931031A (fi

Inventor

Pui-Ho Yuen

Charles Eckhart

Teresa Etlinger

Nancy Levine

Original Assignee

Schering Corp

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-09-10

Filing date

1993-03-09

Publication date

2003-05-30

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24320279&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI111078(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1993-03-09 Application filed by Schering Corp filed Critical Schering Corp

1993-03-09 Publication of FI931031A0 publication Critical patent/FI931031A0/fi

1993-03-09 Publication of FI931031A publication Critical patent/FI931031A/fi

2003-05-30 Application granted granted Critical

2003-05-30 Publication of FI111078B publication Critical patent/FI111078B/fi

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07J—STEROIDS
- C07J17/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, having an oxygen-containing hetero ring not condensed with the cyclopenta(a)hydrophenanthrene skeleton
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0043—Nose

Landscapes

Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Rheumatology (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Steroid Compounds (AREA)
Measuring Or Testing Involving Enzymes Or Micro-Organisms (AREA)
Medicinal Preparation (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

FI931031A 1990-09-10 1993-03-09 Menetelmä mometasonifuroaattimonohydraatin valmistamiseksi FI111078B (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
US58023990A	1990-09-10	1990-09-10
US58023990		1990-09-10
PCT/US1991/006249 WO1992004365A1 (en)	1990-09-10	1991-09-06	Mometasone furoate monohydrate, process for making same and pharmaceutical compositions
US9106249		1991-09-06

Publications (3)

Publication Number	Publication Date
FI931031A0 FI931031A0 (fi)	1993-03-09
FI931031A FI931031A (fi)	1993-03-09
FI111078B true FI111078B (fi)	2003-05-30

Family

ID=24320279

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
FI931031A FI111078B (fi)	1990-09-10	1993-03-09	Menetelmä mometasonifuroaattimonohydraatin valmistamiseksi

Country Status (35)

Country	Link
US (1)	US6180781B1 (sl)
EP (1)	EP0548114B1 (sl)
JP (1)	JPH0725789B2 (sl)
KR (1)	KR960013445B1 (sl)
CN (1)	CN1030920C (sl)
AT (1)	ATE113604T1 (sl)
AU (1)	AU663471B2 (sl)
BG (1)	BG60755B2 (sl)
CA (1)	CA2091360C (sl)
CZ (1)	CZ281318B6 (sl)
DE (2)	DE69104991T2 (sl)
DK (1)	DK0548114T5 (sl)
EE (1)	EE02962B1 (sl)
ES (1)	ES2065701T3 (sl)
FI (1)	FI111078B (sl)
HK (1)	HK185996A (sl)
HR (1)	HRP920383B1 (sl)
HU (1)	HU213401B (sl)
IE (1)	IE67056B1 (sl)
IL (1)	IL99437A (sl)
LU (1)	LU90366I2 (sl)
MX (2)	MX9203396A (sl)
MY (1)	MY106644A (sl)
NL (1)	NL980012I2 (sl)
NO (1)	NO300548B1 (sl)
NZ (1)	NZ239711A (sl)
OA (1)	OA09772A (sl)
PH (1)	PH30443A (sl)
PL (1)	PL165803B1 (sl)
PT (1)	PT98905B (sl)
SI (1)	SI9111497A (sl)
TW (2)	TW229208B (sl)
WO (1)	WO1992004365A1 (sl)
YU (1)	YU48666B (sl)
ZA (1)	ZA917148B (sl)

Families Citing this family (35)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
ATE113604T1 (de) *	1990-09-10	1994-11-15	Schering Corp	Mometason-furoate-monohydrat, verfahren zu seiner herstellung und das enthaltende pharmazeutische zusammensetzungen.
PE44995A1 (es) *	1994-01-27	1995-12-18	Schering Corp	Furoato de mometasona para el tratamiento de las enfermedades pulmonares y de las vias respiratorias
US5837699A (en) *	1994-01-27	1998-11-17	Schering Corporation	Use of mometasone furoate for treating upper airway passage diseases
US5886200A (en) *	1996-07-01	1999-03-23	Schering Corporation	Process for the preparation of 17-esters of 9 α, 21-dihalo-pregnane-11 β, 17 α-diol-20-ones
US5976573A (en)	1996-07-03	1999-11-02	Rorer Pharmaceutical Products Inc.	Aqueous-based pharmaceutical composition
CN1059476C (zh) *	1996-08-21	2000-12-13	邓维鹏	金黄色铝合金硒盐电解着色方法
AU9674398A (en) *	1997-10-09	1999-05-03	Schering Corporation	Mometasone furoate suspensions for nebulization
US6187765B1 (en) *	1997-10-09	2001-02-13	Schering Corporation	Mometasone furoate suspensions for nebulization
MY133181A (en) *	1998-09-10	2007-10-31	Schering Corp	Methods and compositions for treating sinusitis, otitis media and other related disorders using antihistamines
GB0207906D0 (en) *	2002-04-05	2002-05-15	3M Innovative Properties Co	Formoterol and mometasone aerosol formulations
US8912174B2 (en) *	2003-04-16	2014-12-16	Mylan Pharmaceuticals Inc.	Formulations and methods for treating rhinosinusitis
US9808471B2 (en)	2003-04-16	2017-11-07	Mylan Specialty Lp	Nasal pharmaceutical formulations and methods of using the same
US7811606B2 (en)	2003-04-16	2010-10-12	Dey, L.P.	Nasal pharmaceutical formulations and methods of using the same
AR045536A1 (es) *	2003-08-29	2005-11-02	Ranbaxy Lab Ltd	Inhibidores de la fosfodiesterasa tipo -iv
WO2005051931A2 (en) *	2003-11-26	2005-06-09	Ranbaxy Laboratories Limited	Phosphodiesterase inhibitors
US7491725B2 (en)	2004-02-06	2009-02-17	Bristol-Myers Squibb Company	Process for preparing 2-aminothiazole-5-aromatic carboxamides as kinase inhibitors
EP1934219A1 (en)	2005-09-16	2008-06-25	Ranbaxy Laboratories Limited	Substituted pyrazolo [3,4-b] pyridines as phosphodiesterase inhibitors
US20070099883A1 (en) *	2005-10-07	2007-05-03	Cheryl Lynn Calis	Anhydrous mometasone furoate formulation
RU2008119322A (ru) *	2005-10-19	2009-11-27	Рэнбакси Лабораториз Лимитед (In)	Композиции ингибиторов фосфодиэстеразы iv типа
EP1948164A1 (en)	2005-10-19	2008-07-30	Ranbaxy Laboratories, Ltd.	Pharmaceutical compositions of muscarinic receptor antagonists
CN100436473C (zh) *	2005-12-09	2008-11-26	天津药业集团有限公司	糠酸莫美他松中间体21-酯及制法
CN100389121C (zh) *	2005-12-09	2008-05-21	天津药业集团有限公司	糠酸莫美他松中间体21-羟的制备方法
DE102006034883A1 (de) *	2006-07-25	2008-01-31	Hermal Kurt Herrmann Gmbh & Co. Ohg	Pharmazeutische Zusammensetzung enthaltend Mometasonfuroat
KR20090069309A (ko) *	2006-09-22	2009-06-30	랜박시 래보러터리스 리미티드	포스포디에스터라제 타입-ⅳ의 저해제
US20100029728A1 (en) *	2006-09-22	2010-02-04	Ranbaxy Laboratories Limited	Phosphodiesterase inhibitors
EP1958947A1 (en)	2007-02-15	2008-08-20	Ranbaxy Laboratories Limited	Inhibitors of phosphodiesterase type 4
AP2453A (en)	2007-03-14	2012-08-31	Ranbaxy Lab Ltd	Pyrazolo(3,4-B) pyridine derivatives as phosphodiesterase inhibitors
EP2124943A1 (en) *	2007-03-14	2009-12-02	Ranbaxy Laboratories Limited	Pyrazolo [3, 4-b]pyridine derivatives as phosphodiesterase inhibitors
EP2111861A1 (en)	2008-04-21	2009-10-28	Ranbaxy Laboratories Limited	Compositions of phosphodiesterase type IV inhibitors
DK2435024T3 (en)	2009-05-29	2016-10-24	Pearl Therapeutics Inc	Compositions for the respiratory delivery of active agents and related methods and systems
US8815258B2 (en) *	2009-05-29	2014-08-26	Pearl Therapeutics, Inc.	Compositions, methods and systems for respiratory delivery of two or more active agents
PT105058B (pt)	2010-04-21	2013-04-17	Hovione Farmaciencia S A	Processo para processamento de partículas de ingredientes activos farmacêuticos
CA2905542C (en)	2013-03-15	2022-05-03	Pearl Therapeutics, Inc.	Methods and systems for conditioning of particulate crystalline materials
CN107266518B (zh) *	2016-04-08	2021-03-30	天津金耀集团有限公司	一种糠酸莫米松晶型及其制备方法
CN107260671B (zh) *	2016-04-08	2021-03-26	天津金耀集团有限公司	一种糠酸莫米松混悬鼻喷剂组合物

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3260474D1 (en) *	1981-02-02	1984-09-06	Schering Corp	Aromatic heterocyclic esters of steroids, their preparation and pharmaceutical compositions containing them
US4783444A (en)	1984-09-17	1988-11-08	Schering Corporation	Antiglaucoma compositions and methods
US4808610A (en) *	1986-10-02	1989-02-28	Schering Corporation	Mometasone furoate anti-inflammatory cream composition using hexylene glycol
US4775529A (en) *	1987-05-21	1988-10-04	Schering Corporation	Steroid lotion
ATE113604T1 (de) *	1990-09-10	1994-11-15	Schering Corp	Mometason-furoate-monohydrat, verfahren zu seiner herstellung und das enthaltende pharmazeutische zusammensetzungen.

1991
- 1991-09-06 AT AT91915453T patent/ATE113604T1/de active
- 1991-09-06 KR KR1019930700702A patent/KR960013445B1/ko not_active IP Right Cessation
- 1991-09-06 WO PCT/US1991/006249 patent/WO1992004365A1/en active IP Right Grant
- 1991-09-06 AU AU84974/91A patent/AU663471B2/en not_active Expired
- 1991-09-06 EP EP91915453A patent/EP0548114B1/en not_active Expired - Lifetime
- 1991-09-06 MX MX9203396A patent/MX9203396A/es unknown
- 1991-09-06 CA CA002091360A patent/CA2091360C/en not_active Expired - Lifetime
- 1991-09-06 HU HU9300685A patent/HU213401B/hu unknown
- 1991-09-06 CZ CZ93383A patent/CZ281318B6/cs not_active IP Right Cessation
- 1991-09-06 PL PL91298223A patent/PL165803B1/pl unknown
- 1991-09-06 DK DK91915453.4T patent/DK0548114T5/da active
- 1991-09-06 DE DE69104991T patent/DE69104991T2/de not_active Expired - Lifetime
- 1991-09-06 IL IL9943791A patent/IL99437A/en not_active IP Right Cessation
- 1991-09-06 ES ES91915453T patent/ES2065701T3/es not_active Expired - Lifetime
- 1991-09-06 JP JP3514768A patent/JPH0725789B2/ja not_active Expired - Lifetime
- 1991-09-06 DE DE1991604991 patent/DE19875032I2/de active Active
- 1991-09-09 MX MX9100990A patent/MX9100990A/es unknown
- 1991-09-09 NZ NZ239711A patent/NZ239711A/en not_active IP Right Cessation
- 1991-09-09 PT PT98905A patent/PT98905B/pt not_active IP Right Cessation
- 1991-09-09 SI SI9111497A patent/SI9111497A/sl unknown
- 1991-09-09 TW TW080107102A patent/TW229208B/zh not_active IP Right Cessation
- 1991-09-09 MY MYPI91001630A patent/MY106644A/en unknown
- 1991-09-09 IE IE315591A patent/IE67056B1/en not_active IP Right Cessation
- 1991-09-09 TW TW083106101A patent/TW272195B/zh not_active IP Right Cessation
- 1991-09-09 ZA ZA917148A patent/ZA917148B/xx unknown
- 1991-09-09 YU YU149791A patent/YU48666B/sh unknown
- 1991-09-09 PH PH43072A patent/PH30443A/en unknown
- 1991-09-10 CN CN91108910A patent/CN1030920C/zh not_active Expired - Lifetime
1992
- 1992-09-21 HR HRP-1497/91A patent/HRP920383B1/xx not_active IP Right Cessation
1993
- 1993-02-26 NO NO930693A patent/NO300548B1/no not_active IP Right Cessation
- 1993-03-09 OA OA60348A patent/OA09772A/en unknown
- 1993-03-09 FI FI931031A patent/FI111078B/fi not_active IP Right Cessation
1994
- 1994-02-24 BG BG098564A patent/BG60755B2/bg unknown
- 1994-11-21 EE EE9400388A patent/EE02962B1/xx unknown
1995
- 1995-04-17 US US08/422,479 patent/US6180781B1/en not_active Expired - Lifetime
1996
- 1996-10-03 HK HK185996A patent/HK185996A/xx not_active IP Right Cessation
1998
- 1998-03-12 NL NL980012C patent/NL980012I2/nl unknown
1999
- 1999-03-05 LU LU90366C patent/LU90366I2/xx unknown

Also Published As

Publication number	Publication date
IE67056B1 (en)	1996-02-21
AU663471B2 (en)	1995-10-12
HU9300685D0 (en)	1993-06-28
FI931031A0 (fi)	1993-03-09
ZA917148B (en)	1992-08-26
MX9100990A (es)	1992-05-04
MX9203396A (es)	1992-07-31
SI9111497A (sl)	1998-04-30
US6180781B1 (en)	2001-01-30
PL165803B1 (pl)	1995-02-28
IE913155A1 (en)	1992-03-11
NO930693D0 (no)	1993-02-26
FI931031A (fi)	1993-03-09
ES2065701T3 (es)	1995-02-16
DE69104991T2 (de)	1995-04-20
NL980012I1 (nl)	1998-05-06
HRP920383B1 (en)	2000-04-30
YU48666B (sh)	1999-06-15
CZ38393A3 (en)	1994-01-19
IL99437A (en)	1995-05-29
CN1030920C (zh)	1996-02-07
WO1992004365A1 (en)	1992-03-19
TW272195B (sl)	1996-03-11
CZ281318B6 (cs)	1996-08-14
OA09772A (en)	1993-11-30
AU8497491A (en)	1992-03-30
HRP920383A2 (en)	1998-06-30
CN1059911A (zh)	1992-04-01
DE69104991D1 (de)	1994-12-08
PT98905A (pt)	1992-09-30
IL99437A0 (en)	1992-08-18
NO300548B1 (no)	1997-06-16
ATE113604T1 (de)	1994-11-15
EE02962B1 (et)	1997-02-17
KR960013445B1 (ko)	1996-10-05
TW229208B (sl)	1994-09-01
CA2091360C (en)	1997-04-08
CA2091360A1 (en)	1992-03-11
HU213401B (en)	1997-06-30
DK0548114T5 (da)	1995-01-30
PH30443A (en)	1997-05-09
JPH0725789B2 (ja)	1995-03-22
PT98905B (pt)	1998-08-31
BG60755B2 (bg)	1996-02-29
HK185996A (en)	1996-10-11
NO930693L (no)	1993-02-26
YU149791A (sh)	1994-01-20
NZ239711A (en)	1992-09-25
EP0548114A1 (en)	1993-06-30
JPH05506667A (ja)	1993-09-30
DE19875032I2 (de)	2007-04-19
LU90366I2 (fr)	1999-05-05
MY106644A (en)	1995-07-31
EP0548114B1 (en)	1994-11-02
NL980012I2 (nl)	2004-11-01
HUT64361A (en)	1993-12-28

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Legal Events

Date	Code	Title	Description
2003-07-24	SPCF	Supplementary protection certificate application filed	Spc suppl protection certif: L20030010
2008-06-24	SPCG	Supplementary protection certificate granted	Spc suppl protection certif: 219 Extension date: 20120219
2011-11-25	MA	Patent expired

Date

Code

Title

Description

2003-07-24

SPCF

Supplementary protection certificate application filed

Spc suppl protection certif: L20030010

2008-06-24

SPCG

Supplementary protection certificate granted

Spc suppl protection certif: 219

Extension date: 20120219

2011-11-25

Patent expired