ES430202A1 - Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas. - Google Patents

Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.

Info

Publication number: ES430202A1
Authority: ES; Spain
Prior art keywords: methyl; normorphines; norcodeines; desoxy; furyl
Prior art date: 1972-09-14
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.): Expired

Application number

ES430202A

Other languages

Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)

CH Boehringer Sohn AG and Co KG

Original Assignee

CH Boehringer Sohn AG and Co KG

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1972-09-14

Filing date

1974-09-19

Publication date

1976-10-16

1974-09-19 Application filed by CH Boehringer Sohn AG and Co KG filed Critical CH Boehringer Sohn AG and Co KG

1976-10-16 Publication of ES430202A1 publication Critical patent/ES430202A1/es

Status Expired legal-status Critical Current

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/47—Quinolines; Isoquinolines
- A61K31/485—Morphinan derivatives, e.g. morphine, codeine
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Life Sciences & Earth Sciences (AREA)
Emergency Medicine (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Networks Using Active Elements (AREA)

ES430202A 1972-09-14 1974-09-19 Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas. Expired ES430202A1 (es)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE2245141A DE2245141A1 (de)	1972-09-14	1972-09-14	Neue n-(heteroarylmethyl)-desoxynormorphine und -norcodeine, deren saeureadditionssalze, verfahren zu deren herstellung sowie deren verwendung als arzneimittel

Publications (1)

Publication Number	Publication Date
ES430202A1 true ES430202A1 (es)	1976-10-16

Family

ID=5856355

Family Applications (8)

Application Number	Title	Priority Date	Filing Date
ES418563A Expired ES418563A1 (es)	1972-09-14	1973-09-07	Procedimiento para la preparacion de n-(heteroarilmetil)- delta7 - desoxi-normorfinas y -norcodeinas.
ES430202A Expired ES430202A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430198A Expired ES430198A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430199A Expired ES430199A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430200A Expired ES430200A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430197A Expired ES430197A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil) - delta7-desoxi-normorfinas y -norcodeina.
ES430203A Expired ES430203A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430201A Expired ES430201A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.

Family Applications Before (1)

Application Number	Title	Priority Date	Filing Date
ES418563A Expired ES418563A1 (es)	1972-09-14	1973-09-07	Procedimiento para la preparacion de n-(heteroarilmetil)- delta7 - desoxi-normorfinas y -norcodeinas.

Family Applications After (6)

Application Number	Title	Priority Date	Filing Date
ES430198A Expired ES430198A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430199A Expired ES430199A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430200A Expired ES430200A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430197A Expired ES430197A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil) - delta7-desoxi-normorfinas y -norcodeina.
ES430203A Expired ES430203A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES430201A Expired ES430201A1 (es)	1972-09-14	1974-09-19	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.

Country Status (24)

Country	Link
US (1)	US3928359A (es)
JP (1)	JPS4966700A (es)
AT (1)	AT326281B (es)
BE (1)	BE804836A (es)
BG (8)	BG21412A3 (es)
CH (7)	CH589090A5 (es)
CS (8)	CS168674B2 (es)
DD (1)	DD109384A5 (es)
DE (1)	DE2245141A1 (es)
ES (8)	ES418563A1 (es)
FI (1)	FI55512C (es)
FR (1)	FR2199982B1 (es)
GB (1)	GB1449222A (es)
HU (1)	HU166367B (es)
IE (1)	IE38320B1 (es)
IL (1)	IL43216A (es)
NL (1)	NL7312621A (es)
NO (1)	NO139482C (es)
PL (8)	PL87721B1 (es)
RO (2)	RO70193A (es)
SE (1)	SE413510B (es)
SU (8)	SU498911A3 (es)
YU (2)	YU243973A (es)
ZA (1)	ZA737289B (es)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4236008A (en) *	1978-09-19	1980-11-25	E. I. Du Pont De Nemours And Company	Fluorination of precursors for fluorine analogs of hydrocodone and oxycodone
US4241065A (en) *	1979-07-02	1980-12-23	E. I. Du Pont De Nemours And Company	Fluoro analogs of hydrocodone and oxycodone useful as analgesics, narcotic antagonists or both
JP2002501923A (ja) *	1998-01-29	2002-01-22	モナシュユニバーシティ	治療用化合物

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2107989A1 (de) *	1971-02-19	1972-09-07	Boehringer Sohn Ingelheim	N-(Furyl-methy])-morphinane, deren Säureadditionssalze sowie Verfahren zu deren Herstellung

1972
- 1972-09-14 DE DE2245141A patent/DE2245141A1/de active Pending
1973
- 1973-09-03 AT AT761673A patent/AT326281B/de not_active IP Right Cessation
- 1973-09-07 ES ES418563A patent/ES418563A1/es not_active Expired
- 1973-09-11 CH CH207177A patent/CH589090A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH1298673A patent/CH590287A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207077A patent/CH591490A5/xx not_active IP Right Cessation
- 1973-09-11 US US396171A patent/US3928359A/en not_active Expired - Lifetime
- 1973-09-11 CH CH198077A patent/CH589088A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH198177A patent/CH589089A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207377A patent/CH591491A5/xx not_active IP Right Cessation
- 1973-09-11 CH CH207277A patent/CH605958A5/xx not_active IP Right Cessation
- 1973-09-12 DD DD173479A patent/DD109384A5/xx unknown
- 1973-09-12 SU SU1962620A patent/SU498911A3/ru active
- 1973-09-12 HU HUBO1463A patent/HU166367B/hu unknown
- 1973-09-12 CS CS282*[A patent/CS168674B2/cs unknown
- 1973-09-12 BG BG24524A patent/BG21412A3/xx unknown
- 1973-09-12 BG BG025616A patent/BG21227A3/xx unknown
- 1973-09-12 BG BG025613A patent/BG21224A3/xx unknown
- 1973-09-12 CS CS285*[A patent/CS168677B2/cs unknown
- 1973-09-12 BG BG025619A patent/BG21230A3/xx unknown
- 1973-09-12 CS CS6322A patent/CS168673B2/cs unknown
- 1973-09-12 CS CS286*[A patent/CS168678B2/cs unknown
- 1973-09-12 CS CS287*[A patent/CS168679B2/cs unknown
- 1973-09-12 CS CS283*[A patent/CS168675B2/cs unknown
- 1973-09-12 BG BG025618A patent/BG21229A3/xx unknown
- 1973-09-12 BG BG25617A patent/BG21228A3/xx unknown
- 1973-09-12 CS CS288*[A patent/CS168680B2/cs unknown
- 1973-09-12 IE IE1630/73A patent/IE38320B1/xx unknown
- 1973-09-12 BG BG025614A patent/BG21225A3/xx unknown
- 1973-09-12 CS CS284*[A patent/CS168676B2/cs unknown
- 1973-09-13 PL PL1973165187A patent/PL87721B1/pl unknown
- 1973-09-13 NL NL7312621A patent/NL7312621A/xx not_active Application Discontinuation
- 1973-09-13 PL PL1973174968A patent/PL90720B1/pl unknown
- 1973-09-13 RO RO7382817A patent/RO70193A/ro unknown
- 1973-09-13 IL IL43216A patent/IL43216A/en unknown
- 1973-09-13 PL PL1973174974A patent/PL91809B1/pl unknown
- 1973-09-13 JP JP48103716A patent/JPS4966700A/ja active Pending
- 1973-09-13 PL PL1973174971A patent/PL91829B1/pl unknown
- 1973-09-13 PL PL1973174969A patent/PL91837B1/pl unknown
- 1973-09-13 PL PL1973174973A patent/PL91808B1/pl unknown
- 1973-09-13 NO NO3588/73A patent/NO139482C/no unknown
- 1973-09-13 BE BE135636A patent/BE804836A/xx unknown
- 1973-09-13 GB GB4314673A patent/GB1449222A/en not_active Expired
- 1973-09-13 FI FI2853/73A patent/FI55512C/fi active
- 1973-09-13 ZA ZA00737289A patent/ZA737289B/xx unknown
- 1973-09-13 YU YU02439/73A patent/YU243973A/xx unknown
- 1973-09-13 PL PL1973174970A patent/PL91836B1/pl unknown
- 1973-09-13 RO RO7300076068A patent/RO63003A/ro unknown
- 1973-09-13 PL PL1973174972A patent/PL91807B1/pl unknown
- 1973-09-14 FR FR7333092A patent/FR2199982B1/fr not_active Expired
- 1973-09-14 SE SE7312583A patent/SE413510B/xx unknown
1974
- 1974-01-28 BG BG025615A patent/BG21226A3/bg unknown
- 1974-09-19 ES ES430202A patent/ES430202A1/es not_active Expired
- 1974-09-19 ES ES430198A patent/ES430198A1/es not_active Expired
- 1974-09-19 ES ES430199A patent/ES430199A1/es not_active Expired
- 1974-09-19 ES ES430200A patent/ES430200A1/es not_active Expired
- 1974-09-19 ES ES430197A patent/ES430197A1/es not_active Expired
- 1974-09-19 ES ES430203A patent/ES430203A1/es not_active Expired
- 1974-09-19 ES ES430201A patent/ES430201A1/es not_active Expired
- 1974-09-30 SU SU2063985A patent/SU503523A3/ru active
- 1974-09-30 SU SU2063986A patent/SU505366A3/ru active
- 1974-09-30 SU SU2063380A patent/SU503524A3/ru active
- 1974-09-30 SU SU2063984A patent/SU520049A3/ru active
- 1974-09-30 SU SU2063982A patent/SU528878A3/ru active
- 1974-09-30 SU SU2063983A patent/SU509239A3/ru active
- 1974-09-30 SU SU2063987A patent/SU506299A3/ru active
1979
- 1979-10-19 YU YU02548/79A patent/YU254879A/xx unknown

Also Published As

Publication number	Publication date
YU254879A (en)	1983-01-21
CH589088A5 (es)	1977-06-30
PL91807B1 (es)	1977-03-31
PL91808B1 (es)	1977-03-31
CS168675B2 (es)	1976-06-29
CS168676B2 (es)	1976-06-29
DE2245141A1 (de)	1974-03-21
PL91836B1 (es)	1977-03-31
RO63003A (fr)	1978-05-15
US3928359A (en)	1975-12-23
ES430203A1 (es)	1976-10-16
RO70193A (ro)	1981-04-30
FR2199982B1 (es)	1977-01-28
BE804836A (fr)	1974-03-13
CH589089A5 (es)	1977-06-30
JPS4966700A (es)	1974-06-27
CH589090A5 (es)	1977-06-30
PL87721B1 (es)	1976-07-31
ES430198A1 (es)	1976-10-16
GB1449222A (en)	1976-09-15
SU520049A3 (ru)	1976-06-30
SU503523A3 (ru)	1976-02-15
PL90720B1 (es)	1977-01-31
CS168679B2 (es)	1976-06-29
SU509239A3 (ru)	1976-03-30
SU503524A3 (ru)	1976-02-15
CS168678B2 (es)	1976-06-29
CH591491A5 (es)	1977-09-30
ES430197A1 (es)	1976-10-16
NO139482B (no)	1978-12-11
SU498911A3 (ru)	1976-01-05
CS168674B2 (es)	1976-06-29
PL91829B1 (es)	1977-03-31
ZA737289B (en)	1975-05-28
BG21229A3 (bg)	1976-03-20
CS168673B2 (es)	1976-06-29
CH591490A5 (es)	1977-09-30
DD109384A5 (es)	1974-11-05
HU166367B (es)	1975-03-28
SU506299A3 (ru)	1976-03-05
ES430201A1 (es)	1976-10-16
BG21226A3 (bg)	1976-03-20
SU505366A3 (ru)	1976-02-28
SU528878A3 (ru)	1976-09-15
CS168680B2 (es)	1976-06-29
AU6030173A (en)	1975-03-13
ES430199A1 (es)	1976-10-16
SE413510B (sv)	1980-06-02
BG21224A3 (bg)	1976-03-20
FI55512C (fi)	1979-08-10
IL43216A (en)	1976-07-30
YU243973A (en)	1982-05-31
ES430200A1 (es)	1976-10-16
FR2199982A1 (es)	1974-04-19
ATA761673A (de)	1975-02-15
CH590287A5 (es)	1977-07-29
IE38320B1 (en)	1978-02-15
NO139482C (no)	1979-03-21
IE38320L (en)	1974-03-14
CS168677B2 (es)	1976-06-29
AT326281B (de)	1975-12-10
ES418563A1 (es)	1976-05-01
BG21225A3 (bg)	1976-03-20
PL91837B1 (es)	1977-03-31
BG21228A3 (es)	1976-03-20
FI55512B (fi)	1979-04-30
NL7312621A (es)	1974-03-18
CH605958A5 (es)	1978-10-13
IL43216A0 (en)	1973-11-28
BG21412A3 (es)	1976-05-20
PL91809B1 (es)	1977-03-31
BG21227A3 (bg)	1976-03-20
BG21230A3 (bg)	1976-03-20

Publication	Publication Date	Title
ES431515A1 (es)	1976-11-01	Procedimiento para la preparacion de 2 - (heteroaril-metil)-5,9 beta - dialcohil-6,7-benzomorfanos.
ES452768A1 (es)	1977-10-01	Procedimiento para la preparacion de nuevos 2-tetrahidrofur-furil-6, 7-benzomorfanos disustituidos en 5, 9-beta.
ES465525A1 (es)	1978-09-16	Procedimiento para la obtencion de nuevas feniletilaminas.
ES429221A1 (es)	1976-08-16	Procedimiento para la preparacion de nuevas amidas de aci- dos n-(1-omega-fenilalcohil)-piperidil-4) - n-(alfa-piridil)-carboxilicos.
ES439927A1 (es)	1977-06-01	Procedimiento para la obtencion de 7-metoxi-6-tiatetracicli-nas.
ES450897A1 (es)	1977-12-01	Procedimiento para la preparacion de n-(r-tetrahidrofurfu- ril)-noroximorfona y n-(s-tetrahidrofurfuril)-noroximorfona.
ES477785A1 (es)	1980-02-01	Procedimiento para la preparacion de nuevas 2-fenilimino- imidazolidinas sustituidas.
ES430198A1 (es)	1976-10-16	Procedimiento para la preparacion de n-(heteroarilmetil - delta7-desoxi-normorfinas y -norcodeinas.
ES416106A1 (es)	1976-02-16	Procedimiento para la preparacion de n-(heteroaril-metil)- 6,14-endoeteno-7a-hidroxialcohil-tetrahidro-nororipavinas y tebainas.
ES424310A1 (es)	1976-06-16	Procedimiento para la preparacion de n-(heteroarilmetil)-7 acil-6,14-endoetenotetrahidronororipavinas y -tebai nas.
IE41106B1 (en)	1979-10-24	Pharmaceutical compositions containing benzylamines
ES468798A1 (es)	1978-12-01	Procedimiento para la preparacion de nuevos 2'-hidroxi-2-(5-isoxazolilmetil)-6,7-benzomorfanos.
GB1358979A (en)	1974-07-03	Treatment of anaplasmosis in cattle