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EA201001683A1 - Производные фенил- или пиридинилзамещенных индазолов - Google Patents

Производные фенил- или пиридинилзамещенных индазолов

Info

Publication number
EA201001683A1
EA201001683A1 EA201001683A EA201001683A EA201001683A1 EA 201001683 A1 EA201001683 A1 EA 201001683A1 EA 201001683 A EA201001683 A EA 201001683A EA 201001683 A EA201001683 A EA 201001683A EA 201001683 A1 EA201001683 A1 EA 201001683A1
Authority
EA
Eurasian Patent Office
Prior art keywords
derivatives
indazols
phenyl
pyridinyl substituted
new
Prior art date
Application number
EA201001683A
Other languages
English (en)
Inventor
Маркус Бергер
Ян Дамен
Карл Эдман
Томас Ханссон
Мартин Хеммерлинг
Нафизал Хоссаин
Хенрик ЙОХАНССОН
Матти Лепистё
Стинабритт Нильссон
Хартмут Ревинкель
Original Assignee
Астразенека Аб
Байер Шеринг Фарма Аг
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41340347&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=EA201001683(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Астразенека Аб, Байер Шеринг Фарма Аг filed Critical Астразенека Аб
Publication of EA201001683A1 publication Critical patent/EA201001683A1/ru

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    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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Abstract

Настоящее изобретение относится к новым индазолильным производным соединениям формулы Iaфармацевтическим композициям, содержащим такие производные, способам получения таких новых производных и к применению таких производных в качестве лекарственных средств.
EA201001683A 2008-05-20 2009-05-20 Производные фенил- или пиридинилзамещенных индазолов EA201001683A1 (ru)

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US8211930B2 (en) 2012-07-03
EP2291359A4 (en) 2011-05-11
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CL2009001248A1 (es) 2010-06-11
CR11801A (es) 2011-02-15
JP2011520954A (ja) 2011-07-21
SI2291369T1 (sl) 2016-02-29
CN102099355B (zh) 2014-11-05
ZA201007918B (en) 2011-07-27
HRP20160071T1 (hr) 2016-02-26
BRPI0912855A2 (pt) 2015-10-13
CO6331310A2 (es) 2011-10-20
IL209121A0 (en) 2011-01-31
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US20100087489A1 (en) 2010-04-08
UA102543C2 (ru) 2013-07-25
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US20120302617A1 (en) 2012-11-29
PE20091974A1 (es) 2010-02-05
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JP2011520955A (ja) 2011-07-21
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IL209122A0 (en) 2011-01-31
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CL2009001247A1 (es) 2010-07-23
US20150080434A1 (en) 2015-03-19
NZ588994A (en) 2012-08-31
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