DK249089D0 - Benzamid-forbindelser, der er nyttige som protease-inhibitorer - Google Patents

Benzamid-forbindelser, der er nyttige som protease-inhibitorer

Info

Publication number: DK249089D0
Authority: DK; Denmark
Prior art keywords: protease inhibitors; compounds used; benzamide compounds; benzamide; het
Prior art date: 1988-05-24

Application number

DK249089A

Other languages

English (en)

Other versions

DK249089A (da

Inventor

Anton Franz Josef Fliri

Rodney Caughren Schnur

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-05-24

Filing date

1989-05-23

Publication date

1989-05-23

1989-05-23 Application filed by Pfizer filed Critical Pfizer

1989-05-23 Publication of DK249089D0 publication Critical patent/DK249089D0/da

1989-11-27 Publication of DK249089A publication Critical patent/DK249089A/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/12—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles
- C07D285/125—1,3,4-Thiadiazoles; Hydrogenated 1,3,4-thiadiazoles with oxygen, sulfur or nitrogen atoms, directly attached to ring carbon atoms, the nitrogen atoms not forming part of a nitro radical
- C07D285/135—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/12—Radicals substituted by oxygen atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/04—Antihaemorrhagics; Procoagulants; Haemostatic agents; Antifibrinolytic agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
- C07D209/40—Nitrogen atoms, not forming part of a nitro radical, e.g. isatin semicarbazone
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/72—Nitrogen atoms
- C07D213/75—Amino or imino radicals, acylated by carboxylic or carbonic acids, or by sulfur or nitrogen analogues thereof, e.g. carbamates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/40—Nitrogen atoms attached in position 8
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/54—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings condensed with carbocyclic rings or ring systems
- C07D231/56—Benzopyrazoles; Hydrogenated benzopyrazoles
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/90—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/30—Nitrogen atoms not forming part of a nitro radical
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
- C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
- C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
- C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
- C07D239/32—One oxygen, sulfur or nitrogen atom
- C07D239/42—One nitrogen atom
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
- C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
- C07D241/10—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members
- C07D241/14—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D241/20—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D261/00—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings
- C07D261/02—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings
- C07D261/06—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members
- C07D261/10—Heterocyclic compounds containing 1,2-oxazole or hydrogenated 1,2-oxazole rings not condensed with other rings having two or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D261/14—Nitrogen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
- C07D263/58—Benzoxazoles; Hydrogenated benzoxazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/54—Nitrogen and either oxygen or sulfur atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D285/00—Heterocyclic compounds containing rings having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by groups C07D275/00 - C07D283/00
- C07D285/01—Five-membered rings
- C07D285/02—Thiadiazoles; Hydrogenated thiadiazoles
- C07D285/04—Thiadiazoles; Hydrogenated thiadiazoles not condensed with other rings
- C07D285/08—1,2,4-Thiadiazoles; Hydrogenated 1,2,4-thiadiazoles

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Engineering & Computer Science (AREA)
Diabetes (AREA)
Hematology (AREA)
Obesity (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Plural Heterocyclic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Pyridine Compounds (AREA)
Pyrrole Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Quinoline Compounds (AREA)
Indole Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK249089A 1988-05-24 1989-05-23 Benzamid-forbindelser, der er nyttige som protease-inhibitorer DK249089A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US07/197,927 US4874864A (en)	1988-05-24	1988-05-24	Benzamide protease inhibitors

Publications (2)

Publication Number	Publication Date
DK249089D0 true DK249089D0 (da)	1989-05-23
DK249089A DK249089A (da)	1989-11-27

Family

ID=22731305

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK249089A DK249089A (da)	1988-05-24	1989-05-23	Benzamid-forbindelser, der er nyttige som protease-inhibitorer

Country Status (19)

Country	Link
US (1)	US4874864A (da)
EP (1)	EP0343894B1 (da)
JP (1)	JPH0667905B2 (da)
KR (1)	KR910004207B1 (da)
AT (1)	ATE77083T1 (da)
AU (1)	AU602294B2 (da)
DE (1)	DE68901746T2 (da)
DK (1)	DK249089A (da)
ES (1)	ES2032229T3 (da)
FI (1)	FI91254C (da)
GR (1)	GR3005072T3 (da)
HU (1)	HU201314B (da)
IE (1)	IE61151B1 (da)
IL (1)	IL90336A (da)
MY (1)	MY104021A (da)
NO (1)	NO173867C (da)
NZ (1)	NZ229235A (da)
PT (1)	PT90623B (da)
ZA (1)	ZA893865B (da)

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JPH05201981A (ja) *	1991-08-06	1993-08-10	Ichikawa Gosei Kagaku Kk	２−アミノ−３−ニトロ−５−ハロゲノピリジン類の製造方法
US5290943A (en) *	1991-02-21	1994-03-01	Ichikawa Gosei Chemical Co., Ltd.	Method of producing 2-acyl amino 5-halogenopyridine compounds
JPH08505846A (ja) *	1992-12-29	1996-06-25	スミスクライン・ビーチャム・コーポレイション	血小板凝集阻害用化合物
FR2703995B1 (fr) *	1993-04-16	1995-07-21	Sanofi Elf	5-acylamino 1,2,4-thiadiazoles, leur preparation et compositions pharmaceutiques en contenant.
AU7084294A (en) *	1993-07-14	1995-02-13	Taisho Pharmaceutical Co., Ltd.	5-acetylthiazoline oxime derivative
JPH09512556A (ja) *	1994-04-29	1997-12-16	サノフィウィンスロップ，インコーポレイティド	ＩＬ−１βプロテアーゼ・インヒビターとしてのハロメチル・アミド
US6100423A (en) *	1995-08-30	2000-08-08	G. D. Searle & Co.	Amino benzenepropanoic acid compounds and derivatives thereof
ATE203234T1 (de) *	1995-08-30	2001-08-15	Searle & Co	Meta-guanidine, harnstoff, thioharnstoff oder azacyklische aminobenzoesäure-derivate als integrin antagonisten
IL127559A0 (en) *	1996-06-20	1999-10-28	Univ Texas	Compounds and methods for providing pharmacologically active preparations and uses thereof
US6028087A (en) *	1998-01-21	2000-02-22	Smithkline Beecham Corporation	Platelet aggregation inhibiting compounds
US6162791A (en) *	1998-03-02	2000-12-19	Apotex Inc.	Thiadiazole compounds useful as inhibitors of cysteine activity dependent enzymes
FR2783519B1 (fr) *	1998-09-23	2003-01-24	Sod Conseils Rech Applic	Nouveaux derives d'amidines, leur preparation, leur application a titre de medicaments et les compositions pharmaceutiques les contenant
DZ3415A1 (fr)	2000-08-31	2002-03-07	Chiron Corp	Guanidinobenzamides comme mc4-r agonistes.
ATE348097T1 (de) *	2001-04-09	2007-01-15	Chiron Corp	Guanidinoverbindungen als melanocortin-4-rezeptor (mc4-r) agonisten
ATE511840T1 (de) *	2001-10-09	2011-06-15	Amgen Inc	Imidazolderivate als entzündungshemmende mittel
US20050124652A1 (en) *	2002-02-04	2005-06-09	Rustum Boyce	Guanidino compounds
US20030195187A1 (en) *	2002-02-04	2003-10-16	Chiron Corporation	Guanidino compounds
US20030207814A1 (en) *	2002-02-04	2003-11-06	Chiron Corporation	Novel guanidinyl derivatives
JP2005524649A (ja) *	2002-02-25	2005-08-18	カイロンコーポレーション	Ｍｃ４−ｒアゴニストの鼻腔内投与
EP1551834B1 (en) *	2002-05-23	2010-08-25	Novartis Vaccines and Diagnostics, Inc.	Substituted quinazolinone compounds
WO2004014905A1 (en) *	2002-08-08	2004-02-19	Boehringer Ingelheim Pharmaceuticals, Inc.	Substituted benzimidazole compounds
DE10314761A1 (de) *	2003-03-31	2004-10-14	Basf Ag	Als Katalysator für die Hydrocyanierung von olefinisch ungesättigten Verbindungen geeignetes System
US7625909B2 (en) *	2003-05-23	2009-12-01	Novartis Vaccines And Diagnostics, Inc.	Substituted quinazolinone compounds
EP1686996A4 (en) *	2003-11-19	2008-11-12	Novartis Vaccines & Diagnostic	QUINAZOLINONE COMPOUNDS WITH REDUCED BIOACCUMULATION
ES2550755T3 (es) *	2007-08-03	2015-11-12	Romark Laboratories, L.C.	Compuestos de tiazolida sustituidos con alquilsulfonilo
CA2940954A1 (en)	2009-05-12	2010-11-18	Romark Laboratories L.C.	Nitazoxanide and tizoxanide for the treatment of rhinovirus and rhabdovirus infections
EA030679B1 (ru)	2009-06-26	2018-09-28	РОМАРК ЛЭБОРЕТЕРИЗ Эл.Си.	Соединения и способы лечения гриппа
US9115127B2 (en)	2010-08-05	2015-08-25	Amgen Inc.	Benzimidazole and azabenzimidazole compounds that inhibit anaplastic lymphoma kinase

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GB1122957A (en) *	1965-06-07	1968-08-07	Smith Kline French Lab	Substituted benzimidazoles and anthelmintic compositions containing them
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CH570759A5 (en) *	1972-10-19	1975-12-31	Ciba Geigy Ag	2-Acylamino-5-halo-1,3,4-thiadiazoles as pesticides - e.g. 2-chloroacetamido-5-bromo-1,3,4-thiadiazole
GB1400540A (en) *	1972-12-06	1975-07-16	Smith Kline French Lab	Salicylamides and compositions thereof
GB1551735A (en) *	1975-06-05	1979-09-12	Lilly Industries Ltd	Acylated aminothiazoles and aminooxadiazoles
DK351778A (da) *	1977-08-15	1979-02-16	Lilly Co Eli	Thiadiazolylbenzamider og fremgangsmaade til deres fremstilling
FR2406634A1 (fr) *	1977-10-19	1979-05-18	Fabre Sa Pierre	Immunostimulants derives d'amino thiazoles
US4343945A (en) *	1979-01-23	1982-08-10	Olin Corporation	5-Benzamido-3-trichloromethyl-1,2,4-thiadiazoles and their use as herbicides, fungicides and insecticides
MA19269A1 (fr) *	1980-09-16	1982-04-01	Lilly Co Eli	Perfectionnement relatif a des derives de n-arylbenzamides .
EP0061882A1 (en) *	1981-03-27	1982-10-06	Eli Lilly And Company	Process for preparing isoxazol-3-ylcarboxamides
US4563527A (en) *	1984-07-19	1986-01-07	Torii & Co., Ltd.	Amidine compounds
JPS61225168A (ja) *	1985-03-30	1986-10-06	Nippon Tokushu Noyaku Seizo Kk	新規ベンズアミド、その製法及び殺虫剤
JPS6229566A (ja) *	1985-07-30	1987-02-07	Taiyo Yakuhin Kogyo Kk	新規グアニジノメチル安息香酸誘導体
ES2044964T3 (es) *	1986-08-12	1994-01-16	Roussel Uclaf	Procedimiento para preparar derivados de decahidroquinolina.
IT1197259B (it) *	1986-09-23	1988-11-30	Valeas Spa	Derivati ammidici eterociclici di acidi benzoici sostituiti e composizione terapeutiche che li contengono come principi attivi

1988
- 1988-05-24 US US07/197,927 patent/US4874864A/en not_active Expired - Fee Related
1989
- 1989-05-18 IL IL90336A patent/IL90336A/xx not_active IP Right Cessation
- 1989-05-22 PT PT90623A patent/PT90623B/pt not_active IP Right Cessation
- 1989-05-22 AT AT89305142T patent/ATE77083T1/de active
- 1989-05-22 ES ES198989305142T patent/ES2032229T3/es not_active Expired - Lifetime
- 1989-05-22 EP EP89305142A patent/EP0343894B1/en not_active Expired - Lifetime
- 1989-05-22 DE DE8989305142T patent/DE68901746T2/de not_active Expired - Lifetime
- 1989-05-22 JP JP1128599A patent/JPH0667905B2/ja not_active Expired - Lifetime
- 1989-05-23 IE IE166889A patent/IE61151B1/en not_active IP Right Cessation
- 1989-05-23 ZA ZA893865A patent/ZA893865B/xx unknown
- 1989-05-23 AU AU35097/89A patent/AU602294B2/en not_active Ceased
- 1989-05-23 MY MYPI89000691A patent/MY104021A/en unknown
- 1989-05-23 FI FI892497A patent/FI91254C/fi not_active IP Right Cessation
- 1989-05-23 KR KR1019890006888A patent/KR910004207B1/ko not_active IP Right Cessation
- 1989-05-23 NZ NZ229235A patent/NZ229235A/en unknown
- 1989-05-23 NO NO892058A patent/NO173867C/no unknown
- 1989-05-23 DK DK249089A patent/DK249089A/da not_active Application Discontinuation
- 1989-05-24 HU HU892579A patent/HU201314B/hu unknown
1992
- 1992-07-01 GR GR920401416T patent/GR3005072T3/el unknown

Also Published As

Publication number	Publication date
IE891668L (en)	1989-11-24
DK249089A (da)	1989-11-27
NO892058D0 (no)	1989-05-23
HUT49860A (en)	1989-11-28
FI91254B (fi)	1994-02-28
GR3005072T3 (da)	1993-05-24
DE68901746D1 (de)	1992-07-16
ES2032229T3 (es)	1993-01-16
FI91254C (fi)	1994-06-10
PT90623A (pt)	1989-11-30
KR890017237A (ko)	1989-12-15
MY104021A (en)	1993-10-30
IL90336A (en)	1993-01-31
JPH0217177A (ja)	1990-01-22
IE61151B1 (en)	1994-10-05
EP0343894B1 (en)	1992-06-10
DE68901746T2 (de)	1992-12-17
NO173867B (no)	1993-11-08
AU3509789A (en)	1989-11-30
ZA893865B (en)	1991-01-30
PT90623B (pt)	1994-10-31
EP0343894A1 (en)	1989-11-29
FI892497A (fi)	1989-11-25
HU201314B (en)	1990-10-28
JPH0667905B2 (ja)	1994-08-31
KR910004207B1 (ko)	1991-06-24
NO173867C (no)	1994-02-16
ATE77083T1 (de)	1992-06-15
FI892497A0 (fi)	1989-05-23
AU602294B2 (en)	1990-10-04
NO892058L (no)	1989-11-27
US4874864A (en)	1989-10-17
NZ229235A (en)	1990-06-26

Publication	Publication Date	Title
DK249089A (da)	1989-11-27	Benzamid-forbindelser, der er nyttige som protease-inhibitorer
DE68920482D1 (de)	1995-02-23	1-Indolylalkyl-4-(substituierte Pyridinyl)-Piperazine.
ATE116306T1 (de)	1995-01-15	Hypoglykämische oxazolidindion-derivate.
LU91196I2 (fr)	2005-10-31	Picoxystrobin et ses dérivlés pharmaceutiquement acceptables(ACANTO).
DK345989A (da)	1990-01-13	Quinolinderivater
ES2046229T3 (es)	1994-02-01	Composicion antiulcerosa.
FI940731A (fi)	1994-04-15	Amiditetratsolit ACAT-inhibiitoreina
NO875357D0 (no)	1987-12-21	Kjemiske sammensetninger og deres bruk som brennstoff additiver.
DK0413278T3 (da)	1997-04-07	Anvendelse af xanthinderivater mod mavesår
ATE41421T1 (de)	1989-04-15	Carbonatderivate des ananasketons.
ATE65986T1 (de)	1991-08-15	Propanolabkoemmlinge.
ATE81128T1 (de)	1992-10-15	Substituierte chinoxaline.
ATE52514T1 (de)	1990-05-15	S-aralkyltrithiophosphonat-insektizide.
ATE74604T1 (de)	1992-04-15	Substituierte pyrimidochinoxaline.

Legal Events

Date	Code	Title	Description
1997-01-13	AHB	Application shelved due to non-payment