DK1284974T3 - Triazolyltropanderivater som CCR5-modulatorer - Google Patents

Triazolyltropanderivater som CCR5-modulatorer

Info

Publication number: DK1284974T3
Authority: DK; Denmark
Prior art keywords: triazolyltropane; derivatives; ccr5 modulators; ccr5; modulators
Prior art date: 2000-05-26

Application number

DK01925808T

Other languages

Danish (da)

English (en)

Inventor

Manoussos Perros

David Anthony Price

Blanda L C Stammen

Anthony Wood

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-05-26

Filing date

2001-05-09

Publication date

2004-06-07

2000-05-26 Priority claimed from GB0014046A external-priority patent/GB0014046D0/en

2000-06-27 Priority claimed from GB0015835A external-priority patent/GB0015835D0/en

2001-05-09 Application filed by Pfizer filed Critical Pfizer

2004-06-07 Application granted granted Critical

2004-06-07 Publication of DK1284974T3 publication Critical patent/DK1284974T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
- C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
- C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
Bioinformatics & Cheminformatics (AREA)
Immunology (AREA)
Pulmonology (AREA)
Diabetes (AREA)
Cardiology (AREA)
Neurosurgery (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Obesity (AREA)
Oncology (AREA)
Endocrinology (AREA)
Urology & Nephrology (AREA)
Rheumatology (AREA)
Physical Education & Sports Medicine (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Hematology (AREA)
Communicable Diseases (AREA)
Virology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pain & Pain Management (AREA)
AIDS & HIV (AREA)
Psychiatry (AREA)
Molecular Biology (AREA)
Emergency Medicine (AREA)
Tropical Medicine & Parasitology (AREA)

DK01925808T 2000-05-26 2001-05-09 Triazolyltropanderivater som CCR5-modulatorer DK1284974T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB0014046A GB0014046D0 (en)	2000-05-26	2000-05-26	Compounds useful in therapy
GB0015835A GB0015835D0 (en)	2000-06-27	2000-06-27	Compounds useful in therapy

Publications (1)

Publication Number	Publication Date
DK1284974T3 true DK1284974T3 (da)	2004-06-07

Family

ID=26244452

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
DK01925808T DK1284974T3 (da)	2000-05-26	2001-05-09	Triazolyltropanderivater som CCR5-modulatorer
DK04004193T DK1526134T3 (da)	2000-05-26	2001-05-09	Triazolyltropanderivater som CCR5-modulatorer

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
DK04004193T DK1526134T3 (da)	2000-05-26	2001-05-09	Triazolyltropanderivater som CCR5-modulatorer

Country Status (51)

Country	Link
EP (3)	EP1990341B1 (cs)
JP (2)	JP3693957B2 (cs)
KR (2)	KR100523501B1 (cs)
CN (2)	CN100355753C (cs)
AP (1)	AP1965A (cs)
AR (2)	AR028622A1 (cs)
AT (2)	ATE407134T1 (cs)
AU (2)	AU2001252482B2 (cs)
BG (1)	BG65966B1 (cs)
BR (1)	BRPI0110955B8 (cs)
CA (1)	CA2408909C (cs)
CR (1)	CR10145A (cs)
CU (1)	CU23288B7 (cs)
CY (3)	CY2008006I1 (cs)
CZ (1)	CZ299102B6 (cs)
DE (3)	DE122008000011I1 (cs)
DK (2)	DK1284974T3 (cs)
DZ (1)	DZ3464A1 (cs)
EA (2)	EA007580B1 (cs)
EE (1)	EE05110B1 (cs)
EG (1)	EG24137A (cs)
ES (3)	ES2215129T3 (cs)
FR (1)	FR08C0007I2 (cs)
GE (1)	GEP20063799B (cs)
HK (3)	HK1054927A1 (cs)
HR (1)	HRP20020938B1 (cs)
HU (1)	HU225810B1 (cs)
IL (2)	IL152531A0 (cs)
IS (1)	IS2511B (cs)
LT (1)	LTC1284974I2 (cs)
LU (1)	LU91417I2 (cs)
MA (1)	MA26902A1 (cs)
ME (1)	ME00555B (cs)
MX (1)	MXPA02011631A (cs)
MY (3)	MY131019A (cs)
NL (1)	NL300338I2 (cs)
NO (3)	NO327892B1 (cs)
NZ (1)	NZ521477A (cs)
OA (1)	OA12264A (cs)
PA (1)	PA8517101A1 (cs)
PE (1)	PE20011371A1 (cs)
PL (1)	PL200551B1 (cs)
PT (2)	PT1526134E (cs)
RS (2)	RS50904B (cs)
SI (2)	SI1526134T1 (cs)
SK (1)	SK286129B6 (cs)
TN (1)	TNSN01077A1 (cs)
TR (1)	TR200400541T4 (cs)
TW (1)	TWI230160B (cs)
UY (1)	UY26727A1 (cs)
WO (1)	WO2001090106A2 (cs)

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CN101712679B (zh) *	2008-10-08	2013-04-10	中国科学院上海药物研究所	一种酰胺类化合物、其药物组合物及其制备方法和用途
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CN102140104B (zh) *	2010-02-03	2014-11-12	中国科学院上海药物研究所	1-(3-(s)-氨基丙基)-哌啶-4-氨基酰胺类化合物、其药物组合物及其制备方法和用途
BR112012024522A2 (pt)	2010-04-02	2017-08-08	Phivco 1 Llc	combinação, uso de uma combinação, composição farmacêutica, forma de dosagem única , kit, e, método para tratar um distúrbio
CN103159754A (zh) *	2011-12-19	2013-06-19	中国科学院上海药物研究所	一种氨基丙基取代托烷胺类化合物、其药物组合物及其制备方法和用途
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CN104304248B (zh) *	2014-10-23	2016-08-10	西北农林科技大学	3-芳基丙酸酯类化合物作为制备杀螨药物的应用
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CN104387379B (zh) *	2014-11-26	2017-01-11	扬州氟药科技有限公司	一种二氟亚甲基哌啶甲酰胺衍生物及其制备方法和用途
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Also Published As

Publication number	Publication date
GEP20063799B (en)	2006-04-25
CY1108451T1 (el)	2014-04-09
ES2401812T3 (es)	2013-04-24
HK1054927A1 (en)	2003-12-19
FR08C0007I2 (fr)	2009-01-15
RS50904B (sr)	2010-08-31
EE05110B1 (et)	2008-12-15
LU91417I9 (cs)	2019-01-02
CY2008006I2 (el)	2009-11-04
JP2005194283A (ja)	2005-07-21
SK16432002A3 (sk)	2004-01-08
EP1526134A2 (en)	2005-04-27
KR100523501B1 (ko)	2005-10-25
NO327892B1 (no)	2009-10-12
NO20025227L (no)	2002-10-31
AR060159A2 (es)	2008-05-28
BG107140A (bg)	2003-05-30
EP1526134A3 (en)	2006-11-29
BG65966B1 (bg)	2010-07-30
NZ521477A (en)	2004-07-30
KR100548854B1 (ko)	2006-02-02
CY2022009I1 (el)	2022-05-27
IS2511B (is)	2009-05-15
LU91417I2 (fr)	2008-04-22
NO2020019I1 (no)	2020-06-30
CN1680371A (zh)	2005-10-12
AP2002002663A0 (en)	2002-12-31
PA8517101A1 (es)	2002-10-24
EG24137A (en)	2008-08-06
IS6565A (is)	2002-09-24
JP3693957B2 (ja)	2005-09-14
WO2001090106A3 (en)	2002-03-28
NO20025227D0 (no)	2002-10-31
EP1990341B1 (en)	2013-01-23
EE200200656A (et)	2004-06-15
JP4854970B2 (ja)	2012-01-18
SK286129B6 (sk)	2008-04-07
EA007580B1 (ru)	2006-12-29
EP1284974B1 (en)	2004-03-03
ME00555A (en)	2011-12-20
CN1279040C (zh)	2006-10-11
PT1526134E (pt)	2008-10-28
AP1965A (en)	2009-03-04
TR200400541T4 (tr)	2004-04-21
BR0110955A (pt)	2003-06-03
CR10145A (es)	2008-08-19
NL300338I1 (nl)	2008-05-01
OA12264A (en)	2003-11-10
CZ299102B6 (cs)	2008-04-23
AU5248201A (en)	2001-12-03
CA2408909C (en)	2006-06-27
CY2008006I1 (el)	2009-11-04
HUP0302474A2 (hu)	2003-11-28
MY156920A (en)	2016-04-15
EA005382B1 (ru)	2005-02-24
DE60102233T2 (de)	2005-01-27
HU225810B1 (en)	2007-10-29
ME00555B (me)	2011-12-20
PE20011371A1 (es)	2002-01-18
HUP0302474A3 (en)	2007-05-29
EP1990341A1 (en)	2008-11-12
DE122008000011I1 (de)	2008-06-05
DE60102233D1 (de)	2004-04-08
NO2010007I1 (no)	2010-04-08
NL300338I2 (nl)	2008-06-02
ATE260914T1 (de)	2004-03-15
ES2215129T3 (es)	2004-10-01
CA2408909A1 (en)	2001-11-29
DE60135685D1 (de)	2008-10-16
FR08C0007I1 (cs)	2008-04-25
LTC1284974I2 (lt)	2020-11-10
IL152531A0 (en)	2003-05-29
AU2001252482B2 (en)	2006-01-19
TWI230160B (en)	2005-04-01
HK1090836A1 (en)	2007-01-05
RS51436B (en)	2011-04-30
ATE407134T1 (de)	2008-09-15
HRP20020938A2 (en)	2005-02-28
CN1437599A (zh)	2003-08-20
BRPI0110955B8 (pt)	2021-05-25
MXPA02011631A (es)	2003-03-27
AU2001252482C1 (en)	2001-12-03
YU82202A (sh)	2005-11-28
UY26727A1 (es)	2001-12-28
CU23288B7 (es)	2008-06-30
MY153023A (en)	2014-12-31
HRP20020938B1 (en)	2011-05-31
JP2003534343A (ja)	2003-11-18
DK1526134T3 (da)	2008-11-17
RS20090438A (en)	2010-05-07
CZ20023806A3 (cs)	2004-01-14
MY131019A (en)	2007-07-31
MA26902A1 (fr)	2004-12-20
EA200401056A1 (ru)	2005-04-28
TNSN01077A1 (fr)	2005-11-10
WO2001090106A2 (en)	2001-11-29
CY2022009I2 (el)	2022-05-27
HK1078573A1 (en)	2006-03-17
PT1284974E (pt)	2004-06-30
EA200201141A1 (ru)	2003-04-24
ES2311126T3 (es)	2009-02-01
AR028622A1 (es)	2003-05-14
DZ3464A1 (cs)	2001-11-29
SI1284974T1 (en)	2004-08-31
LTPA2008004I1 (lt)	2020-07-27
KR20030004417A (ko)	2003-01-14
IL152531A (en)	2010-05-17
SI1526134T1 (sl)	2008-12-31
PL359267A1 (en)	2004-08-23
NO2010007I2 (no)	2013-09-09
EP1526134B1 (en)	2008-09-03
KR20050046743A (ko)	2005-05-18
EP1284974A2 (en)	2003-02-26
PL200551B1 (pl)	2009-01-30
CN100355753C (zh)	2007-12-19
BRPI0110955B1 (pt)	2016-06-28

Publication	Publication Date	Title
DK1526134T3 (da)	2008-11-17	Triazolyltropanderivater som CCR5-modulatorer
NO20026195D0 (no)	2002-12-23	Substituerte-triazolopyrimidiner som anticancer midler
NO20013149L (no)	2001-08-23	Piperidiner som CCR5-modulatorer
NO20013183L (no)	2001-08-08	Azabicykloalkaner som CCR5-modulatorer
NO20013671L (no)	2001-09-26	Substituerte bisycliske derivater nyttige som anticancer midler
DK1492789T3 (da)	2006-09-11	Tropanderivater som CCR5-modulatorer
NO20031001D0 (no)	2003-03-04	Polyarylkarboksamider nyttige som lipidsenkende midler
DK1397364T3 (da)	2007-11-26	Hidtil ukendte pyrrolderivater som farmaceutiske midler
NO20021239L (no)	2002-03-13	Pteridinoner som kinase-inhibitorer
DK1326858T3 (da)	2006-05-08	Piperidinforbindelser som anti-allergiske midler
DK1244647T3 (da)	2006-09-25	Quinzolinderivater som VIGF-inhibitorer
NO20032531D0 (no)	2003-06-04	Tetralon-derivater som antitumormidler
NO20023828L (no)	2002-09-30	Pyrimidin-4-on derivater som LDL-PLA2 inhibitorer
NO20022888L (no)	2002-08-02	Lipopeptider som antibakterielle midler
NO20041317L (no)	2004-06-29	Benzimidazolidinondenvater som muskarine midler
NO20022887L (no)	2002-08-12	Lipopeptider som antibakterielle midler
NO20015065L (no)	2001-10-18	Pyrazolobenzodiazepiner som CDK2-inhibitorer
NO20051042L (no)	2005-03-31	Pyrimidylsulfonamidderivater som kemokinreseptormodulatorer
NO20032272D0 (no)	2003-05-20	Bifenylkarboksamider nyttige som lipidsenkende midler
NO20023770L (no)	2002-08-09	Indol-3-ylderivater
NO20035183D0 (no)	2003-11-21	5-substituerte-2-arylpyridiner som CRF1 modulatorer
NO20040860L (no)	2004-04-22	Farmasoytisk sammensetning som innbefatter lumiracoxib
NO20021959L (no)	2002-05-29	Tetrahydrotiopyranftalazinon-derivater som PDE4-inhibitorer
NO20020457L (no)	2002-03-27	Benzenaminderivater som antikoagulanter
DK1263734T3 (da)	2007-01-29	3-thiomethylpyrazoler som pesticider