AU1208999A - Compounds which inhibit tryptase activity - Google Patents
Compounds which inhibit tryptase activityInfo
- Publication number
- AU1208999A AU1208999A AU12089/99A AU1208999A AU1208999A AU 1208999 A AU1208999 A AU 1208999A AU 12089/99 A AU12089/99 A AU 12089/99A AU 1208999 A AU1208999 A AU 1208999A AU 1208999 A AU1208999 A AU 1208999A
- Authority
- AU
- Australia
- Prior art keywords
- compounds
- tryptase activity
- inhibit tryptase
- inhibit
- activity
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C257/00—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines
- C07C257/10—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines
- C07C257/18—Compounds containing carboxyl groups, the doubly-bound oxygen atom of a carboxyl group being replaced by a doubly-bound nitrogen atom, this nitrogen atom not being further bound to an oxygen atom, e.g. imino-ethers, amidines with replacement of the other oxygen atom of the carboxyl group by nitrogen atoms, e.g. amidines having carbon atoms of amidino groups bound to carbon atoms of six-membered aromatic rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/06—Benzimidazoles; Hydrogenated benzimidazoles with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached in position 2
- C07D235/16—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/20—Two benzimidazolyl-2 radicals linked together directly or via a hydrocarbon or substituted hydrocarbon radical
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
- C07D333/08—Hydrogen atoms or radicals containing only hydrogen and carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (5)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US6515497P | 1997-11-10 | 1997-11-10 | |
US60065154 | 1997-11-10 | ||
US17969598A | 1998-10-27 | 1998-10-27 | |
US09179695 | 1998-10-27 | ||
PCT/US1998/023362 WO1999024407A1 (en) | 1997-11-10 | 1998-11-03 | Compounds which inhibit tryptase activity |
Publications (1)
Publication Number | Publication Date |
---|---|
AU1208999A true AU1208999A (en) | 1999-05-31 |
Family
ID=26745272
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
AU12089/99A Abandoned AU1208999A (en) | 1997-11-10 | 1998-11-03 | Compounds which inhibit tryptase activity |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP1030844A1 (en) |
AU (1) | AU1208999A (en) |
WO (1) | WO1999024407A1 (en) |
Families Citing this family (20)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP1334719A3 (en) | 1996-02-22 | 2003-09-24 | Tularik, Inc. | Pentafluorobenzenesulfonamides and analogs |
CN1147294C (en) | 1996-07-19 | 2004-04-28 | 图拉列克股份有限公司 | Pentafluorobenzenesulfonamides and analogs |
CN100335461C (en) | 1998-09-23 | 2007-09-05 | 图拉里克公司 | Arylsulfonanilide ureas |
WO2000073270A1 (en) * | 1999-05-31 | 2000-12-07 | Daiichi Pharmaceutical Co., Ltd. | Remedies for periodontal diseases |
ATE256666T1 (en) * | 1999-06-04 | 2004-01-15 | Elan Pharma Int Ltd | COMPOSITIONS AND METHODS FOR PREVENTING CELL DEATH |
WO2001019809A1 (en) | 1999-09-14 | 2001-03-22 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Tryptase inhibitors |
DE19945787A1 (en) | 1999-09-24 | 2001-03-29 | Boehringer Ingelheim Pharma | New 2-(amidino- or aminomethyl-phenethyl)-5-sulfonylamino-benzimidazoles, are tryptase inhibitors useful e.g. for treating inflammatory or allergic disease such as asthma, urticaria or arthritis |
DE19945810A1 (en) * | 1999-09-24 | 2001-03-29 | Boehringer Ingelheim Pharma | Substituted benzimidazole derivatives, process for their preparation and their use as medicaments |
US6413990B1 (en) | 1999-09-24 | 2002-07-02 | Boehringer Ingelheim Pharma Kg | Arylsulphonamide-substituted benzimidazoles having tryptase-inhibiting activity |
CA2379557C (en) * | 1999-09-24 | 2008-09-16 | Boehringer Ingelheim Pharma Kg | Arylsulphonamide-substituted benzimidazole derivatives, processes for preparing them and their use as pharmaceutical compositions |
GB9923710D0 (en) * | 1999-10-08 | 1999-12-08 | Proteus Molecular Design | Chemical compounds |
CA2392127A1 (en) | 1999-12-20 | 2001-06-28 | Byk Gulden Lomberg Chemische Fabrik Gmbh | Tryptase inhibitors |
US6924305B2 (en) | 2001-01-31 | 2005-08-02 | Altana Pharma Ag | Diazocine derivatives and their use as tryptase inhibitors |
DE10105628A1 (en) * | 2001-02-08 | 2002-08-22 | Boehringer Ingelheim Pharma | Benzimidazole derivatives, process for their preparation and their use as medicines |
US6656956B2 (en) | 2001-02-08 | 2003-12-02 | Boehringer Ingelheim Pharma Kg | Benzimidazole derivatives, processes for preparing them and their use as pharmaceutical compositions |
ATE364037T1 (en) | 2001-02-21 | 2007-06-15 | Altana Pharma Ag | TRYPTASE INHIBITORS |
AU2002253035B8 (en) | 2001-02-21 | 2008-02-21 | Altana Pharma Ag | Tryptase inhibitors |
US6962941B2 (en) | 2001-06-19 | 2005-11-08 | Altana Pharma Ag | Tryptase inhibitors |
JP2005523883A (en) * | 2001-12-13 | 2005-08-11 | 興和株式会社 | Pharmaceutical composition for prevention and treatment of delayed type hypersensitivity |
US7049333B2 (en) | 2002-06-04 | 2006-05-23 | Sanofi-Aventis Deutschland Gmbh | Substituted thiophenes: compositions, processes of making, and uses in disease treatment and diagnosis |
Family Cites Families (12)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AU527371B2 (en) * | 1980-09-16 | 1983-03-03 | Torii & Co., Ltd. | Amidine |
DE3427865A1 (en) * | 1984-07-27 | 1986-02-06 | Torii & Co., Tokio/Tokyo | Amidino compounds, process for their preparation and pharmaceutical compositions containing these compounds |
ATE114670T1 (en) * | 1991-03-06 | 1994-12-15 | Searle & Co | PHENYLAMIDE DERIVATIVES AS PLATELET AGGREGATION INHIBITORS. |
ZA928276B (en) * | 1991-10-31 | 1993-05-06 | Daiichi Seiyaku Co | Aromatic amidine derivates and salts thereof. |
JPH05213927A (en) * | 1992-02-10 | 1993-08-24 | Torii Yakuhin Kk | New furancarboxylic amidinonaphthyl ester derivative and its acid added salt |
US5525623A (en) * | 1993-03-12 | 1996-06-11 | Arris Pharmaceutical Corporation | Compositions and methods for the treatment of immunomediated inflammatory disorders |
KR100309616B1 (en) * | 1993-03-12 | 2002-02-28 | 추후제출 | Compositions and Methods for the Treatment of Immune Mediated Inflammatory Diseases |
DE4316922A1 (en) * | 1993-05-20 | 1994-11-24 | Boehringer Mannheim Gmbh | New 4-amidinophenylsulfonamides - process for their preparation and medicaments containing these compounds |
WO1996009297A1 (en) * | 1994-09-23 | 1996-03-28 | Arris Pharmaceutical Corporation | Compositions and methods for treating mast-cell inflammatory condition |
ATE222583T1 (en) * | 1995-01-05 | 2002-09-15 | Torii Pharmaceutical Co Ltd | DERIVATIVES OF SUBSTITUTED AMIDINONAPHTHYL ESTER |
WO1997037969A1 (en) * | 1996-04-10 | 1997-10-16 | Ono Pharmaceutical Co., Ltd. | Tryptase inhibitor and novel guanidino derivatives |
IL127873A0 (en) * | 1996-07-08 | 1999-10-28 | Du Pont Pharm Co | Amidinoindoles amidinoazoles and analogs thereof as inhibitors of factor xa and of thrombin |
-
1998
- 1998-11-03 AU AU12089/99A patent/AU1208999A/en not_active Abandoned
- 1998-11-03 WO PCT/US1998/023362 patent/WO1999024407A1/en not_active Application Discontinuation
- 1998-11-03 EP EP98955238A patent/EP1030844A1/en not_active Withdrawn
Also Published As
Publication number | Publication date |
---|---|
EP1030844A1 (en) | 2000-08-30 |
WO1999024407A1 (en) | 1999-05-20 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
MK6 | Application lapsed section 142(2)(f)/reg. 8.3(3) - pct applic. not entering national phase |