AT383128B - METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXY AETHYLESTER OF ALPHA-AMINOBENZYLPENICILLIN - Google Patents

METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXY AETHYLESTER OF ALPHA-AMINOBENZYLPENICILLIN

Info

Publication number: AT383128B
Authority: AT; Austria
Prior art keywords: aethylester; aethoxycarbonyloxy; aminobenzylpenicillin; alpha; producing
Prior art date: 1982-06-29

Application number

AT0238483A

Other languages

German (de)

Other versions

ATA238483A (en

Inventor

Luigi Ratti

Derek Reginald Palmer

Robert Graham Tyson

Original Assignee

Astra Laekemedel Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-06-29

Filing date

1983-06-29

Publication date

1987-05-25

1982-06-29 Priority claimed from IT22141/82A external-priority patent/IT1190897B/en

1983-01-07 Priority claimed from GB838300331A external-priority patent/GB8300331D0/en

1983-06-29 Application filed by Astra Laekemedel Ab filed Critical Astra Laekemedel Ab

1986-06-04 Priority to AT151886A priority Critical patent/AT389700B/en

1986-10-15 Publication of ATA238483A publication Critical patent/ATA238483A/en

1987-05-25 Application granted granted Critical

1987-05-25 Publication of AT383128B publication Critical patent/AT383128B/en

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C68/00—Preparation of esters of carbonic or haloformic acids
- C07C68/02—Preparation of esters of carbonic or haloformic acids from phosgene or haloformates
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
- C07C69/96—Esters of carbonic or haloformic acids
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Plural Heterocyclic Compounds (AREA)

AT0238483A 1982-06-29 1983-06-29 METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXY AETHYLESTER OF ALPHA-AMINOBENZYLPENICILLIN AT383128B (en)

Priority Applications (1)

Application Number	Priority Date	Filing Date	Title
AT151886A AT389700B (en)	1982-06-29	1986-06-04	Process for the preparation of the 1- ethoxycarbonyloxyethyl ester of benzylpenicillin

Applications Claiming Priority (5)

Application Number	Priority Date	Filing Date	Title
IT22141/82A IT1190897B (en)	1982-06-29	1982-06-29	PROCEDURE FOR THE PREPARATION OF THE 1-ETHOXYCARBONYLOXYETHYL ACID ACID 6- (D (-) - ALPHA AMINOALPHA-PHENYLACETAMIDE) -PENICILLANIC
GB8226751		1982-09-20
GB8228622		1982-10-06
GB8232629		1982-11-16
GB838300331A GB8300331D0 (en)	1983-01-07	1983-01-07	Preparation of bromo carbonates

Publications (2)

Publication Number	Publication Date
ATA238483A ATA238483A (en)	1986-10-15
AT383128B true AT383128B (en)	1987-05-25

Family

ID=27516485

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
AT0238483A AT383128B (en)	1982-06-29	1983-06-29	METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXY AETHYLESTER OF ALPHA-AMINOBENZYLPENICILLIN

Country Status (23)

Country	Link
JP (2)	JPH0819052B2 (en)
AT (1)	AT383128B (en)
AU (1)	AU566803B2 (en)
BG (3)	BG38335A3 (en)
CH (2)	CH656377A5 (en)
CY (2)	CY1520A (en)
DD (1)	DD211561A5 (en)
DE (2)	DE3348299C2 (en)
DK (3)	DK160039C (en)
FI (1)	FI79115C (en)
FR (1)	FR2543957B1 (en)
GB (3)	GB2168050A (en)
GR (1)	GR78585B (en)
HU (1)	HU191534B (en)
IE (1)	IE56712B1 (en)
IL (1)	IL68992A (en)
IS (1)	IS1361B6 (en)
NL (1)	NL194081C (en)
NO (3)	NO157696C (en)
NZ (1)	NZ204736A (en)
PT (1)	PT76944B (en)
SE (2)	SE454879B (en)
YU (2)	YU43926B (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
FR2573756B1 (en) *	1984-11-23	1987-01-16	Poudres & Explosifs Ste Nale	PROCESS FOR THE PREPARATION OF BROMO-1 ETHYL AND HYDROCARBYL CARBONATES AND NOVEL BROMO-1 ETHYL AND HYDROCARBYL CARBONATES

Citations (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2161420A1 (en) *	1970-12-30	1972-07-27	Toyama Chemical Co. Ltd., Tokio	Penicillin derivatives and processes for their preparation
AT309683B (en) *	1970-09-25	1973-08-27	Beecham Group Ltd	Process for the production of new penicillins
DE1795701B2 (en) *	1967-09-29	1977-04-21	Ausscheidung aus: 17 95 423 Loevens Kemiske Fabrik Produktionsaktieselskab, Ballerup (Dänemark)	ALPHA-SUBSTITUTED BENZYL PENICILLIC ACID ESTERS

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3873521A (en) *	1970-09-17	1975-03-25	Astra Laekemedel Ab	Esters of {60 -amino penicillins
BE784800A (en) *	1971-06-15	1972-10-02	Yamanouchi Pharma Co Ltd	PROCESS FOR PREPARING NEW OXYMETHYL ESTERS OF PENICILLIN AND CEPHALOSPORIN
IL48514A (en) *	1972-02-15	1976-08-31	Mckenna A	Hexapeptide intermediate for the preparation of the lh-and fsh-releasing hormone
GB1425571A (en) *	1972-03-13	1976-02-18	Astra Laekemedel Ab	Penicillins and cephaosporins
GB1426869A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1426717A (en) *	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
SE397981B (en) *	1973-02-19	1977-11-28	Astra Laekemedel Ab	NEW TETRAALKYLAMMONIUM SALTS OF 6-AMINOPENICILLANIC ACID AND OF BENZYLPENICILLIN INTENDED TO BE USED AS INTERMEDIATE PRODUCTS IN THE PREPARATION OF CERTAIN ESTERS OF 6-AMINOPENICILLANIC ACID AND OF BENZYLPENIC
GB1565656A (en) *	1975-12-13	1980-04-23	Beecham Group Ltd	Preparation of substituted penicillin acid esters
GB1598568A (en) *	1977-04-19	1981-09-23	Glaxo Lab Ltd	Esters of(6r,7r)-3-carbamoyloxymethyl-7-((z)-2-(fur-2-yl)-2-methoxyiminoacetamido)-ceph-3-em-4-carboxylic acid
JPS5444694A (en) *	1977-09-06	1979-04-09	Kou Kamata	Aminobenzylpenicillin derivative
NO832376L (en) *	1982-06-30	1984-01-02	Glaxo Group Ltd	Cephalosporin ANTIBIOTICS.
DE3380024D1 (en) *	1982-11-04	1989-07-13	Astra Laekemedel Ab	Process for the preparation of the 1'-ethoxycarbonyloxyethyl ester of benzylpenicillin

1983
- 1983-06-15 SE SE8303414A patent/SE454879B/en not_active IP Right Cessation
- 1983-06-15 IL IL68992A patent/IL68992A/en not_active IP Right Cessation
- 1983-06-20 IE IE1445/83A patent/IE56712B1/en not_active IP Right Cessation
- 1983-06-24 DE DE3348299A patent/DE3348299C2/de not_active Expired - Lifetime
- 1983-06-24 DE DE3322783A patent/DE3322783A1/en active Granted
- 1983-06-27 GB GB08528958A patent/GB2168050A/en not_active Withdrawn
- 1983-06-28 CH CH3540/83A patent/CH656377A5/en not_active IP Right Cessation
- 1983-06-28 NZ NZ204736A patent/NZ204736A/en unknown
- 1983-06-28 DK DK296683A patent/DK160039C/en not_active IP Right Cessation
- 1983-06-28 BG BG068052A patent/BG38335A3/en unknown
- 1983-06-28 BG BG068053A patent/BG38336A3/en unknown
- 1983-06-28 HU HU832325A patent/HU191534B/en unknown
- 1983-06-28 NL NL8302286A patent/NL194081C/en not_active IP Right Cessation
- 1983-06-28 CH CH527585A patent/CH657620B/de not_active IP Right Cessation
- 1983-06-28 PT PT76944A patent/PT76944B/en unknown
- 1983-06-28 FI FI832363A patent/FI79115C/en not_active IP Right Cessation
- 1983-06-28 NO NO832351A patent/NO157696C/en not_active IP Right Cessation
- 1983-06-28 GR GR71790A patent/GR78585B/el unknown
- 1983-06-28 BG BG061516A patent/BG37527A3/en unknown
- 1983-06-28 AU AU16328/83A patent/AU566803B2/en not_active Expired
- 1983-06-29 AT AT0238483A patent/AT383128B/en not_active IP Right Cessation
- 1983-06-29 IS IS2825A patent/IS1361B6/en unknown
- 1983-06-29 YU YU1415/83A patent/YU43926B/en unknown
- 1983-06-29 DD DD83252531A patent/DD211561A5/en unknown
- 1983-12-30 FR FR8321138A patent/FR2543957B1/en not_active Expired
1985
- 1985-03-28 NO NO851255A patent/NO851255L/en unknown
- 1985-03-28 NO NO851254A patent/NO851254L/en unknown
- 1985-09-16 GB GB08522826A patent/GB2168699B/en not_active Expired
- 1985-09-16 GB GB08522827A patent/GB2169287B/en not_active Expired
1986
- 1986-02-14 YU YU218/86A patent/YU43693B/en unknown
1990
- 1990-04-30 DK DK106090A patent/DK167807B1/en not_active IP Right Cessation
- 1990-04-30 DK DK105990A patent/DK159821C/en not_active IP Right Cessation
- 1990-11-16 CY CY1520A patent/CY1520A/en unknown
- 1990-11-16 CY CY1519A patent/CY1519A/en unknown
1991
- 1991-02-26 SE SE9100548A patent/SE503843C2/en not_active IP Right Cessation
- 1991-04-30 JP JP3124442A patent/JPH0819052B2/en not_active Expired - Lifetime
- 1991-04-30 JP JP3124441A patent/JPH0730082B2/en not_active Expired - Lifetime

Patent Citations (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE1795701B2 (en) *	1967-09-29	1977-04-21	Ausscheidung aus: 17 95 423 Loevens Kemiske Fabrik Produktionsaktieselskab, Ballerup (Dänemark)	ALPHA-SUBSTITUTED BENZYL PENICILLIC ACID ESTERS
AT309683B (en) *	1970-09-25	1973-08-27	Beecham Group Ltd	Process for the production of new penicillins
DE2161420A1 (en) *	1970-12-30	1972-07-27	Toyama Chemical Co. Ltd., Tokio	Penicillin derivatives and processes for their preparation

Also Published As

Publication number	Publication date
SE8303414D0 (en)	1983-06-15
DK106090D0 (en)	1990-04-30
ATA238483A (en)	1986-10-15
GB8522827D0 (en)	1985-10-23
CH656377A5 (en)	1986-06-30
CY1520A (en)	1990-11-16
HU191534B (en)	1987-03-30
YU141583A (en)	1986-06-30
YU43693B (en)	1989-10-31
JPH0819052B2 (en)	1996-02-28
DK105990A (en)	1990-04-30
SE9100548L (en)	1991-02-26
DK105990D0 (en)	1990-04-30
DK106090A (en)	1990-04-30
BG37527A3 (en)	1985-06-14
SE9100548D0 (en)	1991-02-26
DK159821C (en)	1991-04-29
NO851254L (en)	1983-12-30
FI832363L (en)	1983-12-30
DE3322783C2 (en)	1991-01-31
GB2168699A (en)	1986-06-25
JPH0730082B2 (en)	1995-04-05
NL194081B (en)	2001-02-01
DE3348299C2 (en)	1990-12-20
BG38336A3 (en)	1985-11-15
DK160039C (en)	1991-06-10
GB2168699B (en)	1987-04-15
DE3322783A1 (en)	1984-02-09
GB2169287B (en)	1987-04-08
CH657620B (en)	1986-09-15
DK296683D0 (en)	1983-06-28
SE503843C2 (en)	1996-09-16
AU1632883A (en)	1984-01-05
NO851255L (en)	1983-12-30
DK160039B (en)	1991-01-21
GB8522826D0 (en)	1985-10-23
PT76944B (en)	1986-04-09
DK159821B (en)	1990-12-10
DD211561A5 (en)	1984-07-18
CY1519A (en)	1990-11-16
FI79115B (en)	1989-07-31
NO832351L (en)	1983-12-30
NZ204736A (en)	1986-11-12
NO157696C (en)	1988-05-04
DK167807B1 (en)	1993-12-20
IS1361B6 (en)	1989-05-25
NO157696B (en)	1988-01-25
NL8302286A (en)	1984-01-16
JPH0717918A (en)	1995-01-20
JPH0543583A (en)	1993-02-23
SE454879B (en)	1988-06-06
FI79115C (en)	1989-11-10
GR78585B (en)	1984-09-27
PT76944A (en)	1983-07-01
IE831445L (en)	1983-12-29
GB2169287A (en)	1986-07-09
YU21886A (en)	1987-10-31
AU566803B2 (en)	1987-10-29
NL194081C (en)	2001-06-05
GB2168050A (en)	1986-06-11
FI832363A0 (en)	1983-06-28
SE8303414L (en)	1983-12-30
YU43926B (en)	1989-12-31
BG38335A3 (en)	1985-11-15
DK296683A (en)	1983-12-30
IL68992A (en)	1991-06-10
IE56712B1 (en)	1991-11-20
FR2543957B1 (en)	1986-10-24
IS2825A7 (en)	1984-07-08
GB8528958D0 (en)	1986-01-02
FR2543957A1 (en)	1984-10-12

Publication	Publication Date	Title
AT383808B (en)	1987-08-25	METHOD FOR PRODUCING PENEMAS
AT370086B (en)	1983-02-25	METHOD FOR PRODUCING THE D-CAMPHORATE OF L-CARNITINAMIDE
AT379831B (en)	1986-03-10	METHOD FOR PRODUCING CRYSTALS
AT377259B (en)	1985-02-25	METHOD FOR PRODUCING DIHYDROPYRIDYLIMIDATE ESTERS
AT374827B (en)	1984-06-12	METHOD FOR PRODUCING CHOLESTERASE
AT389512B (en)	1989-12-27	METHOD FOR PRODUCING 3-CHLORMETHYLCHINUCLIDINE
AT367436B (en)	1982-07-12	METHOD FOR PRODUCING COPOLYMERISATS
ATA199684A (en)	1989-09-15	METHOD FOR PRODUCING 6-DEOXYANTHRACYCLINONES
AT380686B (en)	1986-06-25	METHOD FOR PRODUCING BUSPIRON
AT380480B (en)	1986-05-26	METHOD FOR PRODUCING ANTHRACYCLINGLYCOSIDES
AT382141B (en)	1987-01-12	METHOD FOR PRODUCING FORESTITE STONES
DD209438A5 (en)	1984-05-09	METHOD FOR PRODUCING SUBSTITUTED CHLOROACETANILIDES
AT375071B (en)	1984-06-25	METHOD FOR PRODUCING PHENYLPYRIDAZINE COMPOUNDS
AT383128B (en)	1987-05-25	METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXY AETHYLESTER OF ALPHA-AMINOBENZYLPENICILLIN
AT388374B (en)	1989-06-12	METHOD FOR PRODUCING N-SULFONYLARYLOXYBENZAMIDES
ATA201283A (en)	1991-04-15	METHOD FOR PRODUCING CARBOXYALKYLDIPEPTIDES
ATA319282A (en)	1983-11-15	METHOD FOR PRODUCING PURE 3-AMINO-CROTONITRILE
AT387012B (en)	1988-11-25	METHOD FOR PRODUCING NITROMETHANE
AT384024B (en)	1987-09-25	METHOD FOR PRODUCING AZINOMETHYL RIFAMYCINES
ATA151886A (en)	1989-06-15	METHOD FOR PRODUCING THE 1-AETHOXYCARBONYLOXYAETHYLESTER OF BENZYLPENICILLIN
ATA328581A (en)	1982-09-15	METHOD FOR PRODUCING 1-PHENOXY-3-AMINO-2-PROPANOLS
AT378180B (en)	1985-06-25	METHOD FOR PRODUCING ADRENOCHROME
ATA81785A (en)	1986-01-15	METHOD FOR PRODUCING ANTHRACYCLINGLYCOSIDES
ATA358482A (en)	1983-06-15	METHOD FOR PRODUCING O-TRIMETHYLSILYL-CELLULOSE
AT381309B (en)	1986-09-25	METHOD FOR PRODUCING 5Z-SHAPES OF 2,3,4-TRINOR-1,5-INTER-M-PHENYLENE-PROSTACYCLINDERIVA EN

Legal Events

Date	Code	Title	Description
2005-06-15	ELA	Expired due to lapse of time