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AR009809A1 - Derivados de 10,13,15-trioxatriciclo[9.2.1(9.6)]-pentadecanona, procedimientos para su preparacion y medicamentos que contienen estos compuestos - Google Patents

Derivados de 10,13,15-trioxatriciclo[9.2.1(9.6)]-pentadecanona, procedimientos para su preparacion y medicamentos que contienen estos compuestos

Info

Publication number
AR009809A1
AR009809A1 ARP970104375A ARP970104375A AR009809A1 AR 009809 A1 AR009809 A1 AR 009809A1 AR P970104375 A ARP970104375 A AR P970104375A AR P970104375 A ARP970104375 A AR P970104375A AR 009809 A1 AR009809 A1 AR 009809A1
Authority
AR
Argentina
Prior art keywords
derivatives
preparation
trioxatriciclo
pentadecanone
procedures
Prior art date
Application number
ARP970104375A
Other languages
English (en)
Inventor
William D Willey
Original Assignee
Solvay Pharm Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Solvay Pharm Gmbh filed Critical Solvay Pharm Gmbh
Publication of AR009809A1 publication Critical patent/AR009809A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/06—Anti-spasmodics, e.g. drugs for colics, esophagic dyskinesia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H1/00—Processes for the preparation of sugar derivatives

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Genetics & Genomics (AREA)
  • Public Health (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Se describen derivados de N-desmetil-N-isopropil-eritromicina-A- espiroacetal estrechados en el anillo con propiedades agonistas de motilinagastrointestinalmente eficaces y su preparacion.
ARP970104375A 1996-10-24 1997-09-23 Derivados de 10,13,15-trioxatriciclo[9.2.1(9.6)]-pentadecanona, procedimientos para su preparacion y medicamentos que contienen estos compuestos AR009809A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19644195A DE19644195A1 (de) 1996-10-24 1996-10-24 10,13,15-Trioxatricyclo[9.2.1.1.·9·.·6·]-pentadecanon-Derivate, Verfahren zu ihrer Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
AR009809A1 true AR009809A1 (es) 2000-05-03

Family

ID=7809858

Family Applications (1)

Application Number Title Priority Date Filing Date
ARP970104375A AR009809A1 (es) 1996-10-24 1997-09-23 Derivados de 10,13,15-trioxatriciclo[9.2.1(9.6)]-pentadecanona, procedimientos para su preparacion y medicamentos que contienen estos compuestos

Country Status (27)

Country Link
US (1) US5912235A (es)
EP (1) EP0838469B1 (es)
JP (1) JP4175682B2 (es)
KR (1) KR100466495B1 (es)
CN (1) CN1093133C (es)
AR (1) AR009809A1 (es)
AT (1) ATE211745T1 (es)
AU (1) AU726092B2 (es)
BR (2) BR9705157A (es)
CA (1) CA2219311C (es)
CZ (1) CZ291768B6 (es)
DE (2) DE19644195A1 (es)
DK (1) DK0838469T3 (es)
DZ (1) DZ2322A1 (es)
ES (1) ES2170318T3 (es)
HK (1) HK1010885A1 (es)
HU (1) HU222540B1 (es)
IL (1) IL121969A (es)
MX (1) MX9707974A (es)
NO (1) NO308362B1 (es)
NZ (1) NZ328979A (es)
PL (1) PL184693B1 (es)
PT (1) PT838469E (es)
RU (1) RU2181727C2 (es)
SK (1) SK283114B6 (es)
UA (1) UA44310C2 (es)
ZA (1) ZA979059B (es)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6100239A (en) * 1996-11-26 2000-08-08 Chugai Seiyaku Kabushiki Kaisha 13-membered ring macrolide compound, medicine containing the same, and process for producing the same
DE60027015T2 (de) * 2000-08-17 2006-10-05 The Kitasato Institute Pseudoerythromycin-derivate
JP2003007917A (ja) * 2001-06-19 2003-01-10 Sanyo Electric Co Ltd 回路装置の製造方法
US6986882B2 (en) * 2002-01-17 2006-01-17 Astrazeneca Ab Therapy for functional dyspepsia
DK1633774T3 (da) 2003-06-18 2010-05-25 Tranzyme Pharma Inc Makrocykliske motilinreceptorantagonister
GB0611907D0 (en) 2006-06-15 2006-07-26 Glaxo Group Ltd Compounds
WO2007007018A1 (en) 2005-07-12 2007-01-18 Glaxo Group Limited Piperazine heteroaryl derivates as gpr38 agonists
US8536182B2 (en) 2005-07-26 2013-09-17 Glaxo Group Limited Benzylpiperazine derivatives and their medical use
CA2632779A1 (en) * 2005-12-08 2007-06-14 Pfizer Inc. Method for demethylating the 3'-dimethylamino group of erythromycin compounds
NZ573450A (en) 2006-06-28 2011-11-25 Glaxo Group Ltd Piperazinyl derivatives useful in the treatment of gpr38 receptor mediated diseases
CN101528765B (zh) 2006-09-11 2015-04-22 欧塞拉治疗有限公司 用于治疗胃肠动力障碍病症的促胃动素受体的大环拮抗剂
CA2750699C (en) 2009-02-27 2015-12-29 Raqualia Pharma Inc. Oxyindole derivatives with motilin receptor agonistic activity
US9682126B2 (en) * 2013-03-25 2017-06-20 Zeria Pharmaceutical Co., Ltd. Postprandial gastrokinetic agent

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3725385A (en) * 1970-11-02 1973-04-03 Abbott Lab Process for the demethylation of 3-amino macrolides
US5106961A (en) * 1987-05-26 1992-04-21 Eli Lilly And Company Erythromycin ring-contracted derivatives
US4920102A (en) * 1988-04-18 1990-04-24 Eli Lilly And Company Method for treating gastrointestinal disorders
DE4200145A1 (de) * 1992-01-07 1993-07-08 Kali Chemie Pharma Gmbh 7,10-epoxy-oxacyclododecan-derivate, verfahren und zwischenprodukte zu ihrer herstellung und diese verbindungen enthaltende arzneimittel

Also Published As

Publication number Publication date
CN1186808A (zh) 1998-07-08
NO308362B1 (no) 2000-09-04
JPH10130297A (ja) 1998-05-19
US5912235A (en) 1999-06-15
CA2219311C (en) 2007-09-04
CZ310697A3 (cs) 1998-06-17
CA2219311A1 (en) 1998-04-24
HK1010885A1 (en) 1999-07-02
PL322802A1 (en) 1998-04-27
JP4175682B2 (ja) 2008-11-05
IL121969A (en) 2000-06-29
DE59705964D1 (de) 2002-02-14
ES2170318T3 (es) 2002-08-01
KR19980032626A (ko) 1998-07-25
EP0838469A1 (de) 1998-04-29
ATE211745T1 (de) 2002-01-15
HUP9701660A3 (en) 1998-08-28
SK283114B6 (sk) 2003-02-04
CZ291768B6 (cs) 2003-05-14
AU726092B2 (en) 2000-11-02
DE19644195A1 (de) 1998-04-30
MX9707974A (es) 1998-04-30
KR100466495B1 (ko) 2005-05-27
IL121969A0 (en) 1998-03-10
NO974934D0 (no) 1997-10-24
CN1093133C (zh) 2002-10-23
DK0838469T3 (da) 2002-03-18
ZA979059B (en) 1998-05-07
PT838469E (pt) 2002-05-31
AU4278897A (en) 1998-04-30
BR9705157A (pt) 1999-09-28
DZ2322A1 (fr) 2002-12-28
RU2181727C2 (ru) 2002-04-27
NZ328979A (en) 1998-10-28
NO974934L (no) 1998-04-27
BR9705143A (pt) 2000-12-12
SK141997A3 (en) 1998-05-06
EP0838469B1 (de) 2002-01-09
PL184693B1 (pl) 2002-12-31
HU222540B1 (hu) 2003-08-28
HUP9701660A2 (hu) 1998-05-28
UA44310C2 (uk) 2002-02-15
HU9701660D0 (en) 1997-12-29

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