NO20051497D0 - Beta-laktamaseinhibitorprodrug. - Google Patents

Beta-laktamaseinhibitorprodrug.

Info

Publication number: NO20051497D0
Authority: NO; Norway
Prior art keywords: laktamaseinhibitorprodrug; beta
Prior art date: 2002-08-23

Application number

NO20051497A

Other languages

English (en)

Other versions

NO20051497L (no

Inventor

Anthony Marfat

Dale Gordon Mcleod

Original Assignee

Pfizer Prod Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-08-23

Filing date

2005-03-21

Publication date

2005-03-21

2005-03-21 Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc

2005-03-21 Publication of NO20051497D0 publication Critical patent/NO20051497D0/no

2005-03-21 Publication of NO20051497L publication Critical patent/NO20051497L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
- C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
- C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Communicable Diseases (AREA)
Oncology (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicinal Preparation (AREA)

NO20051497A 2002-08-23 2005-03-21 Beta-laktamaseinhibitorprodrug. NO20051497L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US40564002P	2002-08-23	2002-08-23
PCT/IB2003/003582 WO2004018484A1 (en)	2002-08-23	2003-08-11	Beta-lactamase inhibitor prodrug

Publications (2)

Publication Number	Publication Date
NO20051497D0 true NO20051497D0 (no)	2005-03-21
NO20051497L NO20051497L (no)	2005-03-21

Family

ID=31946909

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20051497A NO20051497L (no)	2002-08-23	2005-03-21	Beta-laktamaseinhibitorprodrug.

Country Status (31)

Country	Link
US (1)	US7091197B2 (no)
EP (1)	EP1534717B1 (no)
JP (1)	JP2005539037A (no)
KR (1)	KR20050037583A (no)
CN (1)	CN1688589A (no)
AP (1)	AP2005003231A0 (no)
AR (1)	AR041028A1 (no)
AT (1)	ATE349452T1 (no)
AU (1)	AU2003250489A1 (no)
BR (1)	BR0313683A (no)
CA (1)	CA2494953A1 (no)
DE (1)	DE60310733D1 (no)
EA (1)	EA007540B1 (no)
EC (1)	ECSP055625A (no)
GT (1)	GT200300179A (no)
HR (1)	HRP20050162A2 (no)
IL (1)	IL166719A0 (no)
IS (1)	IS7693A (no)
MA (1)	MA27387A1 (no)
MX (1)	MXPA05001446A (no)
NO (1)	NO20051497L (no)
NZ (1)	NZ538340A (no)
OA (1)	OA12909A (no)
PA (1)	PA8579701A1 (no)
PE (1)	PE20040899A1 (no)
PL (1)	PL375988A1 (no)
TN (1)	TNSN05054A1 (no)
TW (1)	TWI250162B (no)
UY (1)	UY27947A1 (no)
WO (1)	WO2004018484A1 (no)
ZA (1)	ZA200501513B (no)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
MXPA05012895A (es) *	2003-06-05	2006-02-22	Pfizer Prod Inc	Profarmaco inhibidor de beta-lactamasa.
US20060105941A1 (en) *	2004-11-12	2006-05-18	Allergan, Inc.	Mixed antibiotic codrugs
US20090306341A1 (en) *	2005-07-29	2009-12-10	Joachim Emmert	LC/MS Blends Containing Ionizing Additives
WO2010118968A1 (en)	2009-04-16	2010-10-21	Nicox S.A.	No-donor aspirin derivatives
WO2013056163A1 (en)	2011-10-14	2013-04-18	The Regents Of The University Of California	Beta-lactamase inhibitors
AU2013207510A1 (en) *	2012-01-06	2014-07-31	The Regents Of The University Of California	Compositions, methods of use, and methods of treatment
CN109422765B (zh) *	2017-09-05	2020-08-28	香港理工大学深圳研究院	C类β-内酰胺酶抑制剂及其制备方法和应用

Family Cites Families (24)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE34011B1 (en)	1969-03-13	1975-01-08	Leo Pharm Prod Ltd	New penicillin esters
IE34019B1 (en)	1969-03-18	1975-01-08	Leo Pharm Prod Ltd	New semi-synthetic penicillin esters
GB1267936A (en)	1969-05-28	1972-03-22	Beecham Group Ltd	DERIVATIVES OF alpha-AMINOPENICILLINS
US3957764A (en)	1969-11-11	1976-05-18	Lovens Kemiske Fabrik Produktionsaktieselskab	6-aminopenicillanic acid derivatives
US3862181A (en)	1970-10-28	1975-01-21	Squibb & Sons Inc	Process for preparing cephalosporins
GB1315566A (en)	1970-11-06	1973-05-02	Leo Pharm Prod Ltd	Penicillanic acid derivatives
CA996929A (en)	1971-04-05	1976-09-14	Kohzi Nakano	Acyloxyalkyl ester derivatives of penicillin
GB1426717A (en)	1972-03-13	1976-03-03	Astra Laekemedel Ab	Penicillins
GB1433131A (en)	1972-03-13	1976-04-22	Astra Laekemedel Ab	Penicillins
US4397783A (en)	1979-03-05	1983-08-09	Pfizer Inc.	Process for converting 6,6-disubstituted penicillanic acid derivatives to the 6-β-congeners
DE2927004A1 (de) *	1979-07-04	1981-05-27	Bayer Ag, 5090 Leverkusen	Penicillansaeure-1,1-dioxide, ihre herstellung und ihre verwendung als arzneimittel als arzneimittel
US4287181A (en) *	1979-10-22	1981-09-01	Pfizer Inc.	Derivatives of 6β-hydroxyalkylpenicillanic acids as β-lactamase inhibitors
US4432970A (en)	1979-11-23	1984-02-21	Pfizer Inc.	6-beta-Halopenicillanic acid 1,1-dioxides as beta-lactamase inhibitors
GB2076812A (en) *	1980-05-22	1981-12-09	Ciba Geigy Ag	Penam-dioxide compounds, processes for their manufacture, and their use
JPS5849387A (ja)	1981-09-17	1983-03-23	Sankyo Co Ltd	７−メトキシセフアロスポリン化合物およびその製法
AU559689B2 (en) *	1981-09-22	1987-03-19	Kureha Kagaku Kogyo K.K.	Penicillin derivative
US4406887A (en)	1981-10-13	1983-09-27	Bristol-Myers Company	Method for treating resistant bacteria including anaerobes
US4428935A (en) *	1982-05-24	1984-01-31	Pfizer Inc.	Penicillanic acid dioxide prodrug
US4521533A (en)	1984-07-12	1985-06-04	Pfizer Inc.	Salts of 6-alpha-(aminomethyl)penicillanic acid 1,1-dioxide esters and beta-lactam antibiotics
DE3901405A1 (de)	1989-01-19	1990-07-26	Hoechst Ag	Cephalosporinderivate und verfahren zu ihrer herstellung
JPH03206038A (ja)	1990-01-08	1991-09-09	Yoshitomi Pharmaceut Ind Ltd	抗菌剤
GB9001405D0 (en)	1990-01-22	1990-03-21	Leo Pharm Prod Ltd	New intermediates,their production and use
GB9208492D0 (en)	1992-04-16	1992-06-03	Glaxo Spa	Heterocyclic compounds
MXPA05012895A (es)	2003-06-05	2006-02-22	Pfizer Prod Inc	Profarmaco inhibidor de beta-lactamasa.

2003
- 2003-08-06 PA PA20038579701A patent/PA8579701A1/es unknown
- 2003-08-11 KR KR1020057002983A patent/KR20050037583A/ko active IP Right Grant
- 2003-08-11 OA OA1200500051A patent/OA12909A/en unknown
- 2003-08-11 EA EA200500398A patent/EA007540B1/ru unknown
- 2003-08-11 JP JP2004530453A patent/JP2005539037A/ja not_active Abandoned
- 2003-08-11 AT AT03792574T patent/ATE349452T1/de not_active IP Right Cessation
- 2003-08-11 EP EP03792574A patent/EP1534717B1/en not_active Expired - Lifetime
- 2003-08-11 AU AU2003250489A patent/AU2003250489A1/en not_active Abandoned
- 2003-08-11 WO PCT/IB2003/003582 patent/WO2004018484A1/en active IP Right Grant
- 2003-08-11 AP AP2005003231A patent/AP2005003231A0/xx unknown
- 2003-08-11 CN CNA038243164A patent/CN1688589A/zh active Pending
- 2003-08-11 DE DE60310733T patent/DE60310733D1/de not_active Expired - Lifetime
- 2003-08-11 MX MXPA05001446A patent/MXPA05001446A/es unknown
- 2003-08-11 BR BR0313683-3A patent/BR0313683A/pt not_active IP Right Cessation
- 2003-08-11 NZ NZ538340A patent/NZ538340A/en unknown
- 2003-08-11 CA CA002494953A patent/CA2494953A1/en not_active Abandoned
- 2003-08-11 PL PL03375988A patent/PL375988A1/xx unknown
- 2003-08-19 PE PE2003000840A patent/PE20040899A1/es not_active Application Discontinuation
- 2003-08-21 UY UY27947A patent/UY27947A1/es not_active Application Discontinuation
- 2003-08-21 AR ARP030103023A patent/AR041028A1/es unknown
- 2003-08-22 GT GT200300179A patent/GT200300179A/es unknown
- 2003-08-22 TW TW092123156A patent/TWI250162B/zh not_active IP Right Cessation
- 2003-08-25 US US10/648,408 patent/US7091197B2/en not_active Expired - Fee Related
2005
- 2005-02-07 IL IL16671905A patent/IL166719A0/xx unknown
- 2005-02-10 IS IS7693A patent/IS7693A/is unknown
- 2005-02-21 HR HR20050162A patent/HRP20050162A2/xx not_active Application Discontinuation
- 2005-02-21 ZA ZA200501513A patent/ZA200501513B/en unknown
- 2005-02-23 EC EC2005005625A patent/ECSP055625A/es unknown
- 2005-02-23 MA MA28119A patent/MA27387A1/fr unknown
- 2005-02-23 TN TNP2005000054A patent/TNSN05054A1/fr unknown
- 2005-03-21 NO NO20051497A patent/NO20051497L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
PE20040899A1 (es)	2004-12-28
AU2003250489A1 (en)	2004-03-11
CA2494953A1 (en)	2004-03-04
CN1688589A (zh)	2005-10-26
AP2005003231A0 (en)	2005-03-31
HRP20050162A2 (en)	2005-06-30
BR0313683A (pt)	2005-06-21
EA200500398A1 (ru)	2005-08-25
IL166719A0 (en)	2006-01-15
KR20050037583A (ko)	2005-04-22
ECSP055625A (es)	2005-04-18
EP1534717A1 (en)	2005-06-01
PA8579701A1 (es)	2005-05-24
JP2005539037A (ja)	2005-12-22
TWI250162B (en)	2006-03-01
DE60310733D1 (de)	2007-02-08
AR041028A1 (es)	2005-04-27
UY27947A1 (es)	2004-03-31
US20040110740A1 (en)	2004-06-10
GT200300179A (es)	2004-05-18
IS7693A (is)	2005-02-10
WO2004018484A1 (en)	2004-03-04
OA12909A (en)	2006-10-13
MXPA05001446A (es)	2005-06-06
US7091197B2 (en)	2006-08-15
EP1534717B1 (en)	2006-12-27
ZA200501513B (en)	2006-09-27
NZ538340A (en)	2006-10-27
ATE349452T1 (de)	2007-01-15
TNSN05054A1 (fr)	2007-05-14
TW200417548A (en)	2004-09-16
NO20051497L (no)	2005-03-21
MA27387A1 (fr)	2005-06-01
EA007540B1 (ru)	2006-10-27
PL375988A1 (en)	2005-12-12

Publication	Publication Date	Title
NO20053248D0 (no)	2005-07-01	Kerosenblanding.
DE60305332D1 (de)	2006-06-22	IMIDAZOi1,2-AöPYRIDINE
NO20052248D0 (no)	2005-05-09	Svivelstykkesystem.
NO20051500D0 (no)	2005-03-21	Substituerte heterocyklylpyrimidiner.
ITMI20032170A1 (it)	2004-06-22	Tagliacimosse.
FR2855029B1 (fr)	2006-04-07	Cache-pot.
NO20051497D0 (no)	2005-03-21	Beta-laktamaseinhibitorprodrug.
ITMI20030916A1 (it)	2003-11-23	Lancetta.
ITMI20031078A1 (it)	2004-11-30	Copridivano.
ITGE20030068A1 (it)	2005-03-06	Termoalgometro.
ES1055830Y (es)	2004-10-16	Mosquitera.
ES1052590Y (es)	2003-05-01	Quiosco-consigna.
ES1052011Y (es)	2003-03-01	Espetero.
ES1052029Y (es)	2003-03-01	Balin-proyectil.
ES1051110Y (es)	2002-10-16	Caja-palet.
ES1051605Y (es)	2002-12-16	Cromo-puzzle.
ES1051703Y (es)	2003-01-16	Potera.
ES1052945Y (es)	2003-06-16	Contraventana.
ES1052938Y (es)	2003-06-16	Cantonera.
ES1052654Y (es)	2003-05-01	Cubitera.
ITRM20020034A1 (it)	2002-04-23	Fiocchettatrice.
ITRM20020327A1 (it)	2003-12-10	Dnaser.
ITRE20020089A1 (it)	2004-05-13	Apparecchiatutto.
ITRE20020088A1 (it)	2004-05-13	Parcheggiafacile.
ITRM20020151U1 (it)	2004-03-21	Mobile-letto.

Legal Events

Date	Code	Title	Description
2008-03-31	FC2A	Withdrawal, rejection or dismissal of laid open patent application