NI201200039A - Nuevos derivados dihidro - oxazolobenzodiazepinonas, su procedi - Google Patents
Nuevos derivados dihidro - oxazolobenzodiazepinonas, su procediInfo
- Publication number
- NI201200039A NI201200039A NI201200039A NI201200039A NI201200039A NI 201200039 A NI201200039 A NI 201200039A NI 201200039 A NI201200039 A NI 201200039A NI 201200039 A NI201200039 A NI 201200039A NI 201200039 A NI201200039 A NI 201200039A
- Authority
- NI
- Nicaragua
- Prior art keywords
- oxazolobenzodiazepinones
- procedure
- dihydro derivatives
- new dihydro
- new
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D245/00—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms
- C07D245/04—Heterocyclic compounds containing rings of more than seven members having two nitrogen atoms as the only ring hetero atoms condensed with carbocyclic rings or ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A61P25/16—Anti-Parkinson drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/52—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings condensed with carbocyclic rings or ring systems
- C07D263/54—Benzoxazoles; Hydrogenated benzoxazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Epidemiology (AREA)
- Cardiology (AREA)
- Psychiatry (AREA)
- Heart & Thoracic Surgery (AREA)
- Hospice & Palliative Care (AREA)
- Psychology (AREA)
- Urology & Nephrology (AREA)
- Pain & Pain Management (AREA)
- Vascular Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
Compuestos de fórmula (I): en la que R1 representa un átomo de hidrógeno o un grupo alquilo; R2 representa un grupo alquilo; R3 representa un grupo arilo o heteroarilo. Medicamentos.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR1100682A FR2972454B1 (fr) | 2011-03-08 | 2011-03-08 | Nouveaux derives dihydro-oxazolobenzodiazepinones, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NI201200039A true NI201200039A (es) | 2012-11-09 |
Family
ID=44004482
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NI201200039A NI201200039A (es) | 2011-03-08 | 2012-03-07 | Nuevos derivados dihidro - oxazolobenzodiazepinonas, su procedi |
Country Status (44)
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| HU230684B1 (hu) * | 2014-01-21 | 2017-08-28 | Egis Gyogyszergyar Nyilvanosan Muekoedoe Reszvenytarsasag | Új dihidro-oxazino-benzodiazepin vegyületek és eljárás ezek elõállítására, illetve az ezeket tartalmazó gyógyászati készítmények |
| DE102016005291B4 (de) | 2016-04-29 | 2024-01-11 | Ksg Austria Gmbh | Verfahren zur Herstellung eines elektronischen Gerätes in der Form eines Spritzgußteils mit eingelegter Leiterplatte |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0101223B1 (en) | 1982-08-06 | 1987-04-01 | Ube Industries, Ltd. | process for producing phenylacetones |
| US5891871A (en) * | 1996-03-21 | 1999-04-06 | Cocensys, Inc. | Substituted 2,3-benzodiazepin-4-ones and the use thereof |
| CA2300142A1 (en) * | 1997-08-12 | 1999-02-18 | Peter Kotay Nagy | 1,3-dioxolo/4,5-h//2,3/benzodiazepine derivatives as ampa/kainate receptor inhibitors |
| UA67749C2 (uk) * | 1997-08-12 | 2004-07-15 | Егіш Дьйодьсердьяр Рт. | Похідна 8-заміщеного-9н-1,3-діоксол/4,5-h//2,3/бензодіазепіну з властивостями амра/каїнатного антагоніста, спосіб одержання похідних, фармацевтична композиція (варіанти), спосіб її одержання та спосіб лікування |
| GB9900222D0 (en) * | 1999-01-06 | 1999-02-24 | Merck Sharp & Dohme | Therapeutic compounds |
| HU227128B1 (en) * | 1999-07-07 | 2010-07-28 | Egyt Gyogyszervegyeszeti Gyar | New 2,3-benzodiazepine derivatives |
| JP2009513644A (ja) * | 2005-10-26 | 2009-04-02 | ザ リージェンツ オブ ザ ユニバーシティ オブ ミシガン | 治療組成物および方法 |
| HU230760B1 (hu) * | 2005-12-30 | 2018-03-28 | Egis Gyógyszergyár Nyilvánosan Működő Részvénytársaság | Dihidro-2,3-benzodiazepin-származékok optikai izomerjei, eljárás ezek sztereoszelektív szintézisére, alkalmazásuk, az ezeket tartalmazó gyógyszerkészítmények és az eljárás közbenső termékei |
| EP2298296A1 (en) * | 2009-08-25 | 2011-03-23 | CNRS Centre National De La Recherche Scientifique | Composition and method for treating cognitive impairments in down syndrome subjects |
-
2011
- 2011-03-08 FR FR1100682A patent/FR2972454B1/fr active Active
-
2012
- 2012-02-20 IL IL218215A patent/IL218215A/en active IP Right Grant
- 2012-02-21 JO JO201236A patent/JO2948B1/en active
- 2012-02-22 SG SG2012012340A patent/SG184633A1/en unknown
- 2012-02-22 PE PE2012000242A patent/PE20121682A1/es active IP Right Grant
- 2012-02-22 AU AU2012201031A patent/AU2012201031B2/en not_active Ceased
- 2012-02-24 MY MYPI2012700036A patent/MY162537A/en unknown
- 2012-02-27 CL CL2012000496A patent/CL2012000496A1/es unknown
- 2012-02-28 UY UY0001033927A patent/UY33927A/es unknown
- 2012-03-02 MA MA34658A patent/MA33641B1/fr unknown
- 2012-03-05 CA CA2771189A patent/CA2771189C/fr not_active Expired - Fee Related
- 2012-03-05 GE GEAP201212613A patent/GEP20146017B/en unknown
- 2012-03-06 EC ECSP12011711 patent/ECSP12011711A/es unknown
- 2012-03-06 AP AP2012006149A patent/AP3344A/xx active
- 2012-03-06 CR CR20120109A patent/CR20120109A/es unknown
- 2012-03-06 MX MX2012002788A patent/MX2012002788A/es active IP Right Grant
- 2012-03-07 EP EP12290077.2A patent/EP2497774B1/fr active Active
- 2012-03-07 ZA ZA2012/01681A patent/ZA201201681B/en unknown
- 2012-03-07 EA EA201200267A patent/EA021125B1/ru not_active IP Right Cessation
- 2012-03-07 ES ES12290077.2T patent/ES2442293T3/es active Active
- 2012-03-07 TW TW101107763A patent/TWI428342B/zh not_active IP Right Cessation
- 2012-03-07 RS RS20130492A patent/RS53032B/en unknown
- 2012-03-07 BR BRBR102012005137-0A patent/BR102012005137A2/pt not_active Application Discontinuation
- 2012-03-07 NZ NZ598625A patent/NZ598625A/xx not_active IP Right Cessation
- 2012-03-07 WO PCT/FR2012/000080 patent/WO2012120206A1/fr active Application Filing
- 2012-03-07 DK DK12290077.2T patent/DK2497774T3/da active
- 2012-03-07 RU RU2013144824/04A patent/RU2572556C2/ru not_active IP Right Cessation
- 2012-03-07 SA SA112330231A patent/SA112330231B1/ar unknown
- 2012-03-07 JP JP2012050550A patent/JP5475816B2/ja not_active Expired - Fee Related
- 2012-03-07 PT PT122900772T patent/PT2497774E/pt unknown
- 2012-03-07 UA UAA201202760A patent/UA112153C2/uk unknown
- 2012-03-07 SI SI201230017T patent/SI2497774T1/sl unknown
- 2012-03-07 HN HN2012000485A patent/HN2012000485A/es unknown
- 2012-03-07 SA SA112330331A patent/SA112330331B1/ar unknown
- 2012-03-07 PL PL12290077T patent/PL2497774T3/pl unknown
- 2012-03-07 US US13/413,977 patent/US8778932B2/en not_active Expired - Fee Related
- 2012-03-07 AR ARP120100728A patent/AR085691A1/es unknown
- 2012-03-07 NI NI201200039A patent/NI201200039A/es unknown
- 2012-03-08 CU CUP2012000041A patent/CU24134B1/es unknown
- 2012-03-08 CN CN201210063418.8A patent/CN102675341B/zh not_active Expired - Fee Related
- 2012-03-08 KR KR1020120023935A patent/KR101477991B1/ko active IP Right Grant
- 2012-03-08 GT GT201200066A patent/GT201200066A/es unknown
-
2013
- 2013-03-18 HK HK13103337.1A patent/HK1176355A1/xx not_active IP Right Cessation
- 2013-12-13 CY CY20131101128T patent/CY1114729T1/el unknown
-
2014
- 2014-01-16 HR HRP20140050AT patent/HRP20140050T1/hr unknown
Also Published As
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CY1120188T1 (el) | ΠΑΡΑΓΩΓΑ ΝΑΦΘΥΡΙΔΙΝΗΣ ΧΡΗΣΙΜΑ ΩΣ ΑΝΤΑΓΩΝΙΣΤΕΣ ΙΝΤΕΓΚΡΙΝΗΣ αvβ6 | |
| UA113643C2 (xx) | N-цикліламіди як нематоциди | |
| UA111626C2 (uk) | Похідні дигідрохінолін-2-ону | |
| CR20150061A (es) | Compuesto de pirazolopirimidinas | |
| UY33883A (es) | Novedosos derivados heterocíclicos | |
| BR112013002182A2 (pt) | derivados de quinolina e inibidores de melk contendo os mesmos | |
| CR20150045A (es) | Inhibidores de hepatitis c | |
| EA201290800A1 (ru) | Гетероциклическое соединение | |
| CR20140229A (es) | Nuevos derivados bicíclicos de dihidroisoquinolin-1-ona | |
| CR20120417A (es) | Inhibidores de virus flaviviridae | |
| CR20140535A (es) | Novedosas n-piridinil amidas cíclicas sustituidas como inhibidores de quinasa | |
| CR20130539A (es) | Triazolopiridinas | |
| RS54730B1 (sr) | Inhibitori beta sekretaze | |
| EA200900945A1 (ru) | Новый способ синтеза агомелатина | |
| MX2014014531A (es) | Derivados de aminoquinazolina y piridopirimidina. | |
| EA200900946A1 (ru) | Новый способ синтеза агомелатина | |
| EA201590561A1 (ru) | Пролекарства аминохиназолинового ингибитора киназы | |
| CR20130625A (es) | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina | |
| UA113086C2 (xx) | Піразольні сполуки як інгібітори sglt1 | |
| UA111333C2 (uk) | Спосіб одержання l-аргінінової солі периндроприлу | |
| CR20130597A (es) | Isoxazolinas como agentes terapèuticos | |
| BR112015006370A2 (pt) | meios e métodos para tratamento de tumores sólidos | |
| CY1121116T1 (el) | Νεα μεθοδος για την συνθεση αγομελατινης | |
| CR20150272A (es) | Derivado de hidantoina | |
| EA200900943A1 (ru) | Новый способ синтеза агомелатина |